Non-selective agents

Alprenolol Bucindolo l Carteolol Carvedilol (has additional α-blocking activity) Nadolol Propranolol Sotalol Labetalol (has additional α-blocking activity) Penbutolol (has intrinsic sympathomimetic activity) Pindolol (has intrinsic sympathomimetic activity)

Timolol

β1-Selective agents
Acebutolol (has intrinsic sympathomimetic activity) Atenolol Betaxolol Bisoprolol Celiprolol Esmolol Metoprolol Nebivolol

β2-Selective agents
Butaxamine (weak α-adrenergic agonist activity) - No common clinical applications, but used in experiments.

ICI-118,551 Highly selective β2-adrenergic receptor antagonist - No known clinical applications, but used in experiments due to its strong receptor specificity.

β3-Selective agents
SR 59230A (has additional α-blocking activity) - Used in experiments.

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