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COLINERGIC

Receptor: M1 (SNc, gg veg), M2 (cord, m netezi), M3 (m net, gl ex), M4 (SNC), N1


(neuronal), N2 (musc)
Parasimpmim: Ach, comp sint (metacolina, carbacolina, betanecolul), pilocarpina
Anticolinesterazice: rev (fizostigmina, neostigmina), irev
Parasimplitice: atropina, scopolamina,substit atropina (butilscopolamina, pirenz
epina, metantelina)
Subst gg: nicotina, ggplegice (hexametoniu, mecamilamina, trimetafan)
Curarizante: antidep (tubocurarina, galamina, pancurin), dep (sexametoniu)
ADRENERGIC
Rec: alfa1 (bronsii, perete vasc, trombocite, m radiar iris, tract gastr-intest,
capsula splenica), alfa2 (vase sang, m gastro-intest, gl sal, pancreas, SNC, pr
esin, trombocite), beta 1 (inima, intestin), beta2 (pereti vasc, bronhii, uter),
DA (SNC, postsin: rinichi, coronare, meenterice, gg simp, m net dig)
Simpatomim: directe nesel (adrenalina, noradr, dopamina), alfa1 (fenilefrina, me
toxamina), alfa2 (clonidina), beta (izoprenalina, dobutamina, solbutamol, terbut
alina, fenaterol); indirecte (efedrina, nafazolina, amfetamina)
Simpatolitice: directe alfa (fentolamina, tolazolina, prozosin), beta (propranol
ol, pinelolol, 1 metoprolol, atenolol); indirecte (guanetidina, reserpina)
ANESTEZICE GEN
- per inductie(faza de betie, de excitatie), per de anestezie propriu-zisa (somn
superf, somn prof, faza de alarma), per toxica
- volatile (halotan, metoxifluran, isofluran), gazoase (protoxid azot, cicloprop
an)
- intravenoase: barbiturice (tiopentan sodic), alte (benzdiazepine, ketamina, dr
operidol-fentonil)
ANESTEZICE LOCALE
- pot M act L bupivacaina; pot dur med lidocaina, mepivacaina; pot m dur s proca
ina, cloroprocaina

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