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CN 105251856 A (19) pe A REE RAMI PHA * (21) BIBS 201510791879. 0 (22) BHA 2015. 11.17 1) BA TRO ALR OYA RS Heh 401336 AKT EK AH 8 CD RABA ae ES Balk (74) SAURIBAAY eee BOE AED Ai Up atk) 11489 HBA (51) Int. G1 6070 213/30(2006. 01) ‘p (12) SBS ALR AER HAT (10) RIBAS CN 10525455 (43) FRB A A 2016. 01. 20 a ieHeT _mIPRITE (64) RBA Pb i ie SA BE ye NE FH 67) HE ABE AWE 1 — Fal i EEO OT EEL I Te, FOREN E45 RAT RL, PEA) LR A PBN 4, 4” — Lebo -2— Be) FASE] Ree rege SERGE AT BM, 8 LR DB RTRSSTOM, HS TR. ARB SEL Hl A OPE SZ FR tl SSA 8 FE A fal Ff BURFI WOR. 01105251556 4 RW RK + 27 1. Abi 46 CT RTT TES SOREL LRA BR () FERCURD E30 ~ — 10°C, Fs ATA AR FALUN HIRE a RSE AT BZ (2) GEER ISIE 20 ~ OC, FAL ARR (1) FOR SH a AT oe BY 4,4? —[ (ilk -2- Se) FE) Oca HEL: AF RM. ME 15 ~ 60 SER, SEE FHL, ARH SAMA BY 10°C ~ 35°C, HAMLET ROL, RMA (3) EAP (2) PAAR ER LIS OO IR SEC a TA JE pH (ARE EAT FEL, FEARS ACHE, SAA ARTI ZR AD) HEE FA TAR AR ST” DO A a DU RT RAY 5 ATA pH (AREA 10.0 ~ BE Li pH AFL 11 ~ 12. 2. ARE ARALBER 1 POTASH ATT SURPIELET ECLA FARR CL) ALAS AES TEP LA Zk PE Bf SALE 40°C ~ BOC HEAT RM 215 ~ 60 SDP YE» EEL 3E O'C ~ 40°C ARSEETT QML RMN 15 ~ GO SH ERE WATKAT REET, ART PMs (2) TE FIRB ETP a A Ek Zo RAK, AR, Be a Loy DEAE IK Z MEER » AME 28 FA YO A ALARA PE SY DL Ry Bie HA» 3. AREAL SER 2 POTASH ATT, SORPGEET RUA FARR () FERURD FB, 30 ~ 10°C FR, Fs AR AA UML BSI RARE AT BN IE IEEE Ae PL EASE HT ERE LS ~~ 45 SB CR AD is IP Ig -20 ~ 15°C, HGPRT Jy 30 ~ 45 SNP 5 (2) WEtREES -20~ 0. F a ARMED (3) EAT (2) FIAR AD SET Ch DORI AR NT SS ME WL A FA HEL IE 8 LOC ~~ 20°C, IFAT IE pi Ay 11. 0 ~ 12.0 HRBEATARIR 1 ~ 3 UK, FLAIR 3 Ok, ARO + FORA ZAC HAS HF ELBE RAK Jk» CFA ZB I AACR EL ‘PRI IE 2 1K, ABIL AR TD APARATO BER PER 28 IE 0. OSMPa ~ —0. IMPaa, 7K YEPELISE ASE EL 80°C sb AP HG VEE EME -0. O7MPa ~ -0. IMPa, HKG ANIBEL 60°C 5 (4) Fa) APR (3). POT SAR 19 BR he HA A hE, 48 PS FRE 50°C ~ 60°C IEEE ADU GUE AT ML 30 OP ~ 45 OPE a, RE I EOC ~ 40°C, THIEF A BRISA BR FFI A FE AA TEPER TE HE EAT ABE IR EE, SSE ISE OC ~ 30°C Mh 5. 0 aly My ~ 12 AEE, (RIA HCAIENE LO°C ~ 20°C Ih ELIF] 8. 0 ~ 10 AIRY ZR PB Ls, BOSE HE 90rpm ~ 120rpm, fii 9Srpm ~ LOSrpm WAKA PEE, EARL 60°C FUE HE -0. 05MPa ~ -0. IMPa, ARF PM + (5) APR C4) TARE PPA Took ZB ARK, TTR 60 ~ 90°C, FER LBC, OCMELTE 2. 0 IRE ~ 3. 0 Asin: Bemis ## Jei Meith 48 0°C~ 30°C, bik 9 20°C ~ 30°C: Ly A> FET ZETA » AB HE AE FP a Ti PNA oh GT th LGR LFS PPR A BI ADL RY RGN PTS HFS 19 FR 799-0. OSMPa ~ -O. LMPa, 7 YEPELEE WN 40°C ~ 70°C, FIR BY TH Py 5. 0 “AEE ~ 10 “sii, HEHE Ay 8.0 ~ 10. ANiih , iBE Ae CHAR FAS 7 HSE INT Td SH OC 2 CN 105254556 4 RW RK + 2/24 75-0. O7MPa ~ -0. IMPa, 50°C ~ 60°C, 6. 0 “Asti ~ 8. O SNP Aria LAL Hh OL TY WGA AH TAS ABEL 0.1% © 4 HEAR ALSER 3 TRY) A A718: SREIELE TP PPR AER CL) bent 5 SRC HEY 6 ~ 421, Rid 5:10 5. HEAR ABER 3 ARAYA 46 AT, SORMIECET, PRE R (1) dnl 5 ASR (2) 4,4? ~[ (iki -2- 3 ) FPS ] RADE ELLY (5 ~ 8) 3H 6: 1 6. HEAR ALSEOR 3 FAA Hi a AT, SORMIECET PRR (2) 4 tutu 45 PBR (2) 4, 4? ~[ Clk -2— 3 ) RS] SADE Cy (12 ~ 8) 21, HEN 10:1. TARE BA BEAR 3 FATA HY i eH HG IE CET, ra A aR (2) 4, a? CC We -2- BE) FAA) SUSE 3) dey LTE TAL EL 1 4 ~ 6) , EAI 1:5. 8. HRA BC A BEAR 3S FATA 9 Hl HH, SNE LET, Pred A MR (2) A a, a? CC We -2- BE) FARE) RUSE C4) TEAR EAR REEL 1 (2 ~ 3), Phi 122. 9. HEED ALSER 3 ATR A 7 ids, JONIECET. BRE (3) “PAO UL 10. ARAB ALSER 3 ATR NUH ae 7, SORMIEET, PRA E (3) PINAR RUEIIZ, 2M. ON 105254556 4 i mB 18H MSS Or NE AT Loco] As Az Jak Tinh ILE ANIM, AS Ae Ne TY RN i RT, EL Pel hey A EO A HT BREAK [0002] EF (constipation) AENPR IS DLN SE Ai AK, 3 Be HEE Bae b> Fe ER DFAT HERA E.R — A BIA, SIP SEE TE, TELA BRILL AI SS BE, VAIL AA Mak Aa TW (BRL AS PE AR A Pe ED, A 2 HEIRS AL IIA EPR HE SE AD PEL PY aC Eh BRL IG A SEITE BD WE EAE RA Ro [0003] DLR BEMRHY (GER BAY :Sodium picosulfate, 424 Hy <4, 4 —CHLBE ~2- HE SFP AE ) SARS DURE RAG AN)» HLM TC Se RCRA, AIR ES ARPS Hl. BAIT Pe FREED, CUBE TUF ARUN, LA SSRI NEL Be BGA HN» CEA i A FY SE IM LAT HR AS RAPD A» TR Aa HBR PF SY 7 TOC, 1S FS BATE EY. SEA BERETS USEABLE AUST TE ANCA AA SAE PEELE, PG SSHEAA THE, 2 2 al DRE PES a SES PE PAL AL AL Se AL TA 5 AS PE FAS HOTS AS PO BER AIRE CALE) AOA TE EP OBER 5 EP) ALD TE PTT EADIE, WILDS OTC Bi ARAL, LEME SETTT AAD RA PEAU AT AEE. Sh FEDS I PR a fe & BB BT Pe A SA EA A AR HE. (ooo4] TL RY BiB ARS th AIR AL HEI? ARE, SE EIT, AS RR ER I TES HF a i» ARR NL A BE HEL ASH He A SPI LT Ele pba HA PB a PM HUD BE) EZ, HEEL ABS EE IR AG DC PRGHART LL. ASiShe ABCAIS SEEA 2e TDINY BRE ZA LF) TH GE IK, TK 5 ASP RPE ABE REPU YI 2s FL 1 A SB NS FL OP TL eb FLEA SEA RELATE 5 ELAS Se AE Pe SP FL, CAL aE AR PAL ee PR) 5 AT IBA AK 2a ETA A, SO A OM 41, EY | EF AL A. E28 RSE, TAY RT 8 AR AOE YB EAR SSE PSE EA» ABS PLE EAI, EET ILL WE A BEE A [000s] DL AYRE AY. RAT AA De Angeli AHF, IFT 1966 4 ETAT. FMT, i KAI De Angeli Zi) 3 HITE 1968 421 1970 HE AE SEM HRS TREAT AY TR ARI Al EAS OW 28986 USS55RG43 « MA ART FER REND 2S al 8 SEE 7S A), TEAL Laxoberal (ITB 4 AG HF AL, M1980 4 5 AAPM AA Al. era ASA A 252 a) 3] BER, IEF 1980 4F 5 AVL Laxoberon (Iii ZR LAVERY. [oooe] LATER AH LARS — EAL As BOY hy I LAL BAST AE] AR 4 CN 105254556 A i mB 2/8 Hi LT ba Ao Pr ee PEA ABE [0007] HHi-E-eAY 1152199 eae TOL] wT tl ev IA. 4, 4” — CC eee -2- RE) HE] SRP A SRF MU YE HSE A eR A SS BAA ok, AT BR BE AT a GSI A A ok CBIR, TCR EL BIOL AR kK. A CH515902, 68543613, DE 1904322 #1 4 Al] US3528986 te Ae FELAB IAD Ay ttl eT FE 7K OC A BEI Ne (ooos] 4 A] US3528086 IFT FACAKMLBE BUH PIMA, 4, 4° ~[ Citi -2- 3) FE] OLA A RBI TM TEE EA RMS, TEI Aa. ATL AY ee LAL EAS FE EAE AE LA RAT EEE. ARF SE, CL 7 AI RESELL AUK ARI A A RUC PE pH AEE RE, FRSA ACD SHG 6 TRAIN ATE ERR ELIE, APIA SERIAL pl. MAS SUF MASS ME BY, 4, 4? LCi -2~ Sa) FS ] POY ASR IARR WARS eM ET, FPN A RS FAUT RA IR RAI ZF ADE USHER DT ah HE, BED WRT TR B49 1 9 BAP HE A, 4? [ CME ~2~ AE) ASE] SET LE, A RAR, BLA Tah ELBE SUR SEE P 7 2k IR, ELL ERT BT 5 HA AY LL Hi OC RAT th PAAR AAT 0. 126 «ALAA US3528086 A 2 BA ARS SPB, HEAL: BE YR A HE A Ea PU BA STE AS a Ae EME HE LH BL AUK AAC TR Oo PE Be, EE PB BAe RE [000s] ZEJHTY Helvetica Chimica Acta (1968 4 51 4e3% 5 JH 1164 ~ 1168 HL) HE 2 F444? [Cite -2- aE) FR) PED AL AR 2- CH) RANK 2, 6- LG AAEM, RS TERA ERT ACY [o0s0] (3) FEA PAIR, FEA ASE, EEE Coost] (4) FLATS ie ERE A ALY, HAD IBGD (oos2] (5) HiT, ARTS TEGAN AC Coosa] (6) PY Hi AS BL Wily, WE, oC HR IB [0054] (7) Fe. Ala IF: (ooss] (8) Acith Aas, HEM ZG Hah AS SLAY Be RB AE 8 ON 105254556 4 i mB 6/8 PREC BB Coos] fi 1 yDC my RAR HK Coos7] FL 2 Ay PAL ae Ee ll 4H (I a i EO HE HPLC PE Coos] Fi 3 Ay RAYS HG GAL 1 fil ob VTE BY RHINE USE HE MPLC PRAM, RRT (LEASH RABI TEs Coos] Fei 4 Day AR FAL SSe ini i 2 hil G49 YC NA AU MEAG TE PLC PRM, RRT LEASH RABI TEs Cooco] Fl 5 Day AR FLSA ini i 3 fil hs 9) OY A NP A MEAG TE PLC PRM, RRT LEAHY RABI TEs Coos] FH 6 RAL SEHMGt A 4 tl 4 th IDE FY Ha AAU EHO HE HPLC PALS , RRT (AL AAD Bunt ial ABTHAK [oos2] xf Let [0063] i) 4 2 = fE 2000m1 = FRM A 750m1 FE AML BE, ETEK A 4, 4° 0 CE We -2- BE) FAA] MUA) 100 Fe, MESES 5 Hstbl (A RHEL SE O ~ 5°C, PP ASNT A SR I 102 i» HRA BE Se He RL AAAS Ay, BEL Rea ec SE EAT I. RTT BS, HLS, (RULE 7 A. [0064] AFSC ANEIBLERL A SL Pk ric tee BaF, DA 30.26 (FRA STREET Hd FL 2 WEE FD RATE A RUHL 5 ACAI ATE OIE HL TE, FIA RBI ph. WA = BE HURASS RMN 4, 4” - [Cee -2- BE) PE) A). AE 40 ~ 45 ERE TE A 3.4L BRST FAST REI, BA ITE A ZB LAL A ERE EAL a, TE, EGET 40 BE AEE FPR 4 5 EE HOY REA 8 (ooes] FH 1 AyFc NE HC LGA TRE, Co mt bas Co Om) ATL FRSC ETA (UAE PR PLC 3 ) PRET ALE ST, AULA CE te = Tmin Zea We, ASAE AWE ZE t= 13min AAT MAE, RRT (ELBA RINT TA], GSD RR ARI = 13 FRARK AMARA (ooes) — Seitifsil 1: [0067] AUCH FAERIE PREY LOOL SHE BCSPS Be EME HH I AUILUE 30ke, 1 OR BEML THLE {ERIE -30 ~ -10°C, HEIN RE 6. Oke, HALA EMA SLA AE INTE HEARIEEPE 30 ~ 45 3} Ph. Fetal (dk RARE -20 ~ -10°C, HIM 4, 4? (ibe -2- 3) FARE J] EHH, ATES 4, 4” -[ (ite -2- 3) FARE] BUY 5. Oke AUMLBE 50kg 1 AACA ARTLDCEE 2.0 ANY. STE FLUE Heth AR HLBE 25°C ~ RULE 10 Is Inf ~ 12 Avi}. Bi MEe HEP AAA LAE ASL 55°C , HEHE -0. OTMPa, WRF ARM ET WEAVER O'C~ 10°C, Beil (KR LHE OC ~ 10°C, EIN AUR EL, TAA pHi. OC BASE Fa SLih), AA AE ROR A Ak 52. Ske AAC 10. Oke He Acie Te FEE AZIRZMG 25. Oke/ UHERE IK» Befil 0. O7MPa ~ -0. IMPa, Miz LAE ALEL 70°C, THLE ARAB AHH ET DMA FEAR Z.BE 10. Oke/ UAE ART 5 PR AR RIE T= 2 RAR IM AK 9 i mB 8H FRBNY 60. Okg, 428th) RUB ME 50°C ~ 60°C, RILBEHE 30 SF h~ 45 S40, MERLE 10°C ~ 40°C. FAL BEE NA EA EBA 10. Oke, TEPER 0. 50kg. tA AIAME 10°C ~ 20°C, Be MUR 28 95rpm, ARELIR EL THR 8.0 AMY. BhoLy, Heth BEE HE 0. O7MPa, HAR TLE ASILEL 60°C FARE AUR BLIP IMA FER ZBF 30ke, EAR Ike, ARIF 75°C (RMB 2.0 ht. MEL 20°C, Bits, AA ZN 10. Oke VERA, ALNE TE THT BT ARE. Bet 28) -0. O7MPa, HOA ULE 50°C LEE TPR 6. O IFES. TPR NE MICHA 4) fe Oa CP, ARIK AR ASE 0. (loose) FA 2 ApH Ima A 1 LAUT: SER, Aa ANH ba Ao UE PR A FR ERGBH ET (UAE TPR PLC 3 ) YSERA EME PBT, AULA CE te = Tmin Aaa We, FLEA Hed EE ACS HU [0069] [0070] UR FETT TRAY LOOL J WE SE PIMA MEE 30K, HV EL EA HR WE -15 ~ -10°C, etl fA RULE -15 ~ 10°C, RUN 6. Oke, HAN PEP AE AL, BEAR. HEINE RDS 45 3} PP. PE A RUBE -15 ~ -10°C Mn 4, 4” - [Catt We -2- BE) FAA ] RU URL UE Yasin, PAPE BL 4, 4” -[ (ibe -2- 2E ) FRE) UR 5. Oke A MCE 5Okey He A Ae il Td Me i Te HE RATE 3.0 lM BEAL A Hl (AS FUEL IE 30°C ~ 35°C, PRIA 12 Ahh. JQ ESE HE Al Me ACU HE ASL 55°C, PEAR HE 0. IMP a RFE AAR MEET. HAMEL -10°C~ OC. Hetil RELHE -10°C ~ O'C TINA AULA, TAT pHLL. 0 LASER FE ERTL ) FIT AUR BATE BOR ALA ak 52. Ske AUSUSULAN 10. Oke TRAIL 61M HEIN A ZARZM 25. Oke/ HEAR. BEB EE NE -0. MPa, HK LIE ALL 70°C , URAL. MAZEL 10. Oke / RAK, ERE RAT PMA, 7K PAY 60. Oke, He fh AUIS 60°C, (RULDEE 45 30h, MELE 30°C ~ 40°C. ALR BEI IN AFAR TURAN 10. Oke, TEPER 0. 50kg. BETA RULIS 10°C ~ 20°C, SRMEMPEHE 105rpm, 1% HIRE THR 10 Ast. Cy, EAL IEE PE 0. MPa, HbA HAE ANAL 60°C, WLP AS 6 FP 3 Fe FSC RUME IM A FEAR ZOE 30ke, BUCA Ike, AFT 85°C, (RULES 3.0 At. BE LE 30°C, Ly, OAK E 10. Oke BEIA, LIE A 1-9 OL By Wie RAL Ah 0 BRA ILE -O. MPa, FAA LHE 60°C , WUE TPR 8.0 AsiiL. TPRSE NE, CHISTES SE LF] RTE, JS 8 AB GE 0.1%. (oo71] FA 3 Ay 4e MSHA) 2 TART SER A ANH ba Ao PR FRSC ETA (UAE PR PLC 3 ) PRET ALE ST, AULA CE te = Tmin Zea We, ELSPA RS IU AC A UE (0072) Seif 3 = [0073] UCR, ZERIT TRY LOOL ASDA Be MEME CH I A 32k a, YOU HEE EA AR ELE - 16°C, etb (FRU —16°C FRA 7. Oke, GEARS ERA AA Ime EARLBETE 35 4). A (A ARLE -16°C SATA 4, 4” —( Coie -2- 2) FE) RCS WUC TESGB, PARES HH 4, 4” —[ (bbe -2- 2 ) FPS ] ALM) 5. Oke AIMLHE 5Okg Tee AC TTA + HATIME HERALD 2. 5 clit. GAPE FLL F2etHl RANE 30°C, (RIE 12 NIN. BEES HE PRANK ALL 55 CHCA HE -0. O8MPa, RAR AR IBUELE EP. HABE OC. Hil) {B ARLFE O°C HR AAC PATEK, LY pl. OC LASER ALRGT ) , AR SUSU ANT OR BE 10 CN 105254556 A i mB 8/8 5 Ske AAACN 10. Oke 12 AACA MT LIA ZARZMH 25. Oke/ PRS BE 0. O8MPa, HAGE ALEL 70°C WER ZETA ALT «IMA FE7K ZRF 10. Oke / HEART ARK, WEEE TET BAR IMA Tork PY 65. Oke, fA RADE 55°C, FREE 35 PH, RULE 25°C 6 FARR ABME TIM A TEAK CPE 10. Oke, TR HERE 0. 5Okeeo H(A FAME 15°C, SQ BEMEHE HE LOOrpm, PRL EE THR 9 Ait. TBSLs, BEML IEE RE ~0. OBMPa, Her ELIE AS GEE 60°C, REE ARI PEE To TAL EME IN CAR ZLI 30kg, BEAK L. 2ke, AFT 80°C, PRILDEFE 2.5 “Nit. BEI 25°C, Bt, JOKZAF 10. Oke Bete, PLM OL AY HER AGL «Pet PCE /R -0. O8MPa, AMZIELAE 55°C, WUE THR TNL. PRR TEHE, WICKED AS na PETC OY RAN, BAR ALL 0. 1% [0074] HAW iP 3 TORRENT ARB, A WA Bl bt CeO) eA FRSC ET (UAE PR PLC 3 ) PEATE OPT, AULA CE te = Tmin ZA Whe, FLIP A Re EE ACS Coos] Skitefal 4 (oo7e] UR F, CETTE TRAY LOOL J WE SE PIMA MEE 25k, HO EE HR CREM TA AU RE -16 CNR BEM 5. Oke, RENEL ALE RL EA. ARIE: 35 5 Ph. PEL AME -15°C Hin 4, 4” CC mbtme -2- 3) A) SUH Mm iver 4, 4” ~[ CLE ~2- 38) FALE ] AUN) 5. Oke AUMLME 50ke TE AAC BT A HAI E ERADEHE 2. 5 clit. GAVE FLL, eH RANE 30°C, (RIE 12 IN. BeBe HE Ei OK RANE 55°C, WCF HE 0. O8MPa, WOR ZR TIMUR ET. UR ELE OC. Ea LAS FRMLNE 0°C HEIN SUL ANTE, HAY pH. OC LASEIR ALT ) , TRUE NER RAUL 7K 52. Ske AUASULAN 10. Okey Tee AR TAR EIA ZAZA 21. Oke/ UHR. PE FCASNE 0. O8MPa, A ACHLIE ARERL 70°C, WUE AREF. MA EK ZAM 8. Ske/ WAR TUK, RRA. ARUN IM ATE AMY 50. Oke, PEM {A RULE 55°C, PRELBGEE 35 4} Ph, ERLE 25°C. ALR MEME AE ACCA 8. Ske, HEHE 0. 50ke. FEI AULKE 15°C, JCSLMEAG HE L00rpm, FREI TPR 8. 0 “IEE ~ 10 hf. SLs, BEM LAE HE -0. O8MPa, HVE 60°C, APT. UR MEME IA FCA ZY 25ke, AULA Ike, ETE HLA 80°C, PRUDEE 2. 5 vi}. BERLE 25°C, Ls, LAZY 10. Oke Dei, IEA TAL AY BAL As MICE NE 0. OBMPa, AUK TELE 55°C, WUE TBR 7. 0 ATER SE HE, WICH 49 85 SENET BY BARI, AR ALEL 0. 1% © [0077] 5 yi i A TREAT ERB, A A Bl bat PO A A a Fie cea: CUA PRY BK IPL is) ASEREATAUNE DOT, OUD CE te= Tmin Zea th We, ELSPA RS IU AC A UE Cooma) PAE REA BH AAS SE A Bal AT PA aR BH MELAS AY ZA AS A BB SEAS FEAR HHA ACEH» ALAA ABB Pm i DE A 0s he de Ae eB AAEAR AMR SET Z A 1/3 ot ot i CN 105254856 A li3 12 2/3 ot ot i CN 105254856 A CN 105254856 A be ot ot

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