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Joycemay G.

Andaya III – ABSP 09/03/2018

DRUGS ACTING IN THE NERVOUS SYSTEM

DIRECT ACTING PARASYMPATHETIC AGONIST

Muscarinic Agonist

Bethanecol Carbacol Pilocarpine Muscarine

Nicotine Agonist

Nicotine Varenicline HLC Succinylcholine

Arecoline Lobeline

INDIRECT ACTING PARASYMPATHETIC AGONIST

Amino Alcohol

Edrophonium
Joycemay G. Andaya III – ABSP 09/03/2018

Organocarbamates

Physostigmine Neostigmine Pyridostigmine Ambenomium

Miscellaneous AchE Inhibitors

Tacrine Donepizil Galantamine Rivastigmine

Organophosphates

Ecothiophate Isoflurophate Parathion Malathion

Sarin Soman Tabun


Joycemay G. Andaya III – ABSP 09/03/2018

PARASYMPATHETIC AGONIST

Selective Antimuscarinic Agonist

Darifenacin Fesoterodine Solifenacin Tolteridone

Pirenzipine Telezepine

Non Selective Antimuscarinic Agonist

Atropine Ipratropium Scopolamine Benztropine

Biperiden Trihexyphenidyl
Joycemay G. Andaya III – ABSP 09/03/2018
Anti-Nicotinic Ganglionic Blockers

Hexamethonium Trimethaphan Mecamylamine

Anti-Nicotinic Neuromuscular Blockers

Non-Depolarizing

Atracurium Cistacurium Mivacurium

Pancurium Tubocurarine Vecuronium

Depolarizing

Succinycholine
Joycemay G. Andaya III – ABSP 09/03/2018
DIRECT ACTING NON SELECTIVE SYMPATHETIC AGONIST

Norepinephrine Epinephrine Dopamine

DIRECT ACTING ɑ1-SYMPATHETIC AGONIST

Phenyleprine Tetrahydrozoline Oxymetazoline

Naphazoline Xylometazoline

DIRECT ACTING ɑ2-SYMPATHETIC AGONIST

Clonidine Apraclonidine Brimonidine


Joycemay G. Andaya III – ABSP 09/03/2018

Guanabenz Guanfacine Methyldopa

Dexmedetomidine Tizanidine

DIRECT ACTING B-SYMPATHETIC AGONIST

Dobutamine

DIRECT ACTING B2-SYMPATHETIC AGONIST

Albuterol Bambuterol Salmeterol

Terbutaline Ritodrine

DIRECT ACTING D1-SYMPATHETIC AGONIST


Joycemay G. Andaya III – ABSP 09/03/2018

Fenoldopam

DIRECT ACTING D2-SYMPATHETIC AGONIST

Bromocriptine

INDIRECT ACTING NEUROTRANSMITTER RELEASERS

Amphetamine Methamphetamine Ephedrine Propylhexedine

Tyramine Phenylpropanolamine Phentermine Fenfluramine

INDIRECT ACTING REUPTAKE BLOCKERS


Joycemay G. Andaya III – ABSP 09/03/2018

Cocaine TCA Reserpine Guanethedine

Methyrosine

NON-SELECTIVE a-BLOCKERS

Phentolamine Phenoxybenzamine

DIRECT ACTING B-NON SELECTIVE AGONIST

Isoproterenol

a1-SELECTIVE BLOCKERS
Joycemay G. Andaya III – ABSP 09/03/2018

Prazosin Doxazosin Terazosin Tamsulosin

a2-SELECTIVE BLOCKERS

Yohimbine

NON-SELECTIVE B-BLOCKERS

Propanolol Timolol Betaxolol

INTRINSIC SYMPATHETIC ACTIVITY

Pindolol Acebutolol Carteolol Bopindolol


Joycemay G. Andaya III – ABSP 09/03/2018

Oxyprenolol Celiprolol Penbutolol

MEMBRANE STABILZING ACTIVITY

Pindolol Acebutolol Labetalol Propanolol

Metoprolol

B1-SELECTIVE BLOCKER

Nadolol Esmolol Metoprolol Nebivolol

B2-SELECTIVE BLOCKER MIXED a AND B BLOCKERS

Butoxamine Carvedilol Labetalol

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