You are on page 1of 3
Antipsihotici: farmakokinetika/farmakodinamika oralnih i kratkodjelujuéih intramuskularnih formulacija ‘ Eliminacjs Troovacki Oraina Vilemeje do Vezanje Metabolix! naziv loraspolotivest rajvige azine proteina enzimitvansporten— Metabotta olualvot ‘Antipsinotic! prve generacije Neromin Thorsin 93 ann sossoos maijmmmneiraan, SORICPENORSCIZ Rik pss i cs E Tufenasin Prosi .7% smeao:2sata 99% CYPaDG (alan) supstat — BHofemain, 6 ag saiperis! aldol gasp mine sorcaue Weeevcepara PAG aloperdl eran : jopenidel wool 708 rang 2-8 sath 39%-93% (mol); SON—60% hidroksimetabolitom Meareatt C¥Paka oD, C¥FEDS 5, Samet ohana ‘Loksapin ‘Loksitan 99% 15-3 sata om mani, supstrat CYPSA4 —(amoksapin), 8 Bifara: podernih 5 {ca labor (epots Sst crminl ah open exPabe an C¥PAS a gosipetenarn peensin —Tolafon 20-40% Penton r-gaata oiieggr (Hank EWPAC9 an), Cicer ome Reena grasa (iol) supstrat hnmmed Cnt ggg cxPite tained, cvPane bee stent) Fimonid ——Omp_—= 350% eat ox Gem CVPGAS eva) nln eine, ngs spstat piper vP20s (avn supsteat—Meruidain vostro Tordads —-Melladl ——ag-gghs sasate 68-99% Lnjcetinlior Jetted ordain, sree CvPsci9 (an supsteat—Slidain 50%: pepeaviina Thiotiene —Navane 5, S08 nesta 90% CPUAR lam supsrat —_Nijednanijezailjefena sata eprtnn Ni deemsitriuoperan,7- “Tiwoperain Stein Negev sos) vo%=008 PIAL ini suprat—hidrokrtaopemainy 9.12 ‘Antipsihotic| druge generacije xP (giav), CVPSA Aspipeml Abii sat >on AFD an Debideosipipezal 758 ideoaripipeanats 46st aim etabotenocina Grab CxPiAa gle, CYPADS—_Nesktvog: No} (oo supra CYP3Ag akan, Nene Ascrapin——Sapiris——g58. as-is ys mollglokeronidacja Senin Nemesis agate Uoriagevrspesh —— tenapinN tarball Crise (gla, crabs Nesktivaa: (+> (esa supaea CYPaAs — lukuroad, N-desnet Acenwin Seeuudo—-Nijepeimenjino—Nijedastuppo oll aktnidacje—henapn Nedesmetl= agate UGrayeveabesh —— tenapia Nkarbamol, fabio sukaron Revs 5% sta 09K CVPSM4 (pnw), CYPADSNentivoo: DMax eat (qhoad sopszat Rloapia operon Lrasidon ‘anaapin Paliperton oetapin iperidon prasdon ‘Trgovacki naziv Vroyae ozs, Facts, Vener Fanapt 2yprene Seroquel Risperdal Geadon Oratna bioraspolozivest ‘ito sri 0% 0% sve 100% Apsluio: 70% “bles vodooeu ma oral otopine 94% rai shrsnom: Vrijeme je do najvibe razine osat sonata (easpon 6 a) geste ‘Usmenc: 6st laren pore 15 sta ‘Trenutae patane date aden een: 6 sa Vezanje proteina our od 9% 0% os 80% sox Motabolicki ‘enzimitranspertor, c¥P gg gon, spat CrPade (ol) CovPinsigaei, cvPane {eran CvPaCt9 esa, CyPacs (man C¥Pads (eon) CFP3Ag Gd ‘exP206 pad, supetrat (CaPaAt taal sb Inhibitor Crea cvP Ag awn supra, (CrP sh ator ‘cvPiaa (gavni, c¥PaD6 (eo spt etabolrane evan ‘ularonidacjon Pgikoprotela/ ABC De (ah, supra ahs ad CHP awn, supstat (CrP2D8 (mel) ‘cvPaps avn), C¥PaAt (Goan supateat protin/ABCB!,¥ ‘Seaton on, (CyPaDeclabnhblor orP Aa (mod ups CrPsA id peta, seh ida Motabotita Desnetiavipraia (CAR) didesmat Keipssn (DDCAR) (ake) hidvokera deen Heald ineakien gat, msag26 (aka tD-20209, 1D Soazo (maka) 0- lsonid, 48° dest eaten (aeakivaa) Nejasna akon: Novaioy Muna, Mis Asia: nortan. 7 Hdrokskeeagin ‘ealtvan: retin slo aw Petal site Bacio Ain: 9-hidras Fsperidon ‘Aka: besiainaa ‘ala ge enrol aon (alive, zrasidon ‘loa Some {Sihidreirasidon Eliminaciski polugivot u fedraslin aviprain 2 dane Dean ia dena DDDCAR: 1 tedna 4-5 sa (tain Sanja at) Opsetn ‘metabolic Hoperdan 8 a, Pat a6sai P9529 oli meaboiator loperdon sta, P87 st Pos at arasidon 3840 a0 w.g28: 75-1050 sosat gatas 24-sisats sceriea bt icects0 ‘eifminat) Roetapin: 7st ork: 12a irks Feperdon: 21-0 omeno: 7a Trgovacki Oraina Vrileme jedo Vezanje Metaboli¢ki Eliminaciski haziv Bloraspolotivest hajvge azine proteina enzimitransportet—‘Metabotta potutvatu teen porioon lpm porate: lege oe a5 “979), Chald-Pogh Wasa A odgovaraChilL-Pugh olen ed 5-6, Has B odgovara Child-Pugh ena 7-9, «Masa C odgovaraChd-Pugh eat od 10-35, ‘rare. CxC1~ktensKetinin; CYP ~itokrom P4s0; MDD ~ vlk depres poremets; UCT ~ win §-

You might also like