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Rx option?

Rx Product desirable properties


High
Solubility (Bioavailability)
Stability (Shelf-life)
Free Energy
Polymorphs
Rx option?

Transformation
Amorphous Rx issue? Crystalline

Rx issue?
Pharmaceutical Conversion Pharmaceutical
Solids Solids
Rx Approaches on Solids
1. Nonaqueous Solvate
2. Anhydrate Low
3. Hydrate Free Energy
4. Cocrystal
5. Size Reduction Polymorphs
6. Salt Selection

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