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732

PHARMACOLOGICAL
CLASSIFICATION OF
DRUGS
FIRST EDITION

PREPARED BY

TARIQ AHMAD
DEPARTMENT OF PHARMACY
UNIVERSITY OF LAHORE

TARIQ AHMAD

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

SPECIAL THANX FOR SUPPORT & HELP TO


DR AQEEL AHMAD
DEPARTMENT OF PHARMACY
UNIVERSITY OF LAHORE

DR SHAFIQ AHMAD ZAHID


DEPARTMENT OF PHARMACY
UNIVERSITY OF LAHORE

SAJID MEHMOOD
(TECHNICAL SUPPORT)
DEPARTMENT OF CS
COMSATS

REFERENCE BOOKS
GOODMAN & GILLMANS
THE PHARMACOLOGICAL BASIS OF THERAPEUTICS
LIPPINCOTTS
ILLUSTRATED REVIEWS OF PHARMACOLOGY
BERTRAM G. KATZUNGS
BASIC & CLINICAL PHARMACOLOGY
PHARMAGUIDE

732

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

INDEX
1) DRUGS OF AUTONOMIC
NERVOUS SYSTEM
2) DRUGS OF CENTRAL
NERVOUS SYSTEM

1.
2.
3.
4.
5.
6.
7.
8.
9.
10.
11.
12.

3) DRUGS OF
CARDIOVASCULAR SYSTEM

13.
14.
15.
16.

17.
4) DRUGS ACTING ON BLOOD

18.

5) DRUGS OF GASTRO
INTESTINAL TRACT

19.
20.
21.
22.

6) DRUGS OF RESPIRATORY
SYSTEM

23.
24.
25.

7) DRUGS OF RENAL FUNCTION

26.

8) CHEMOTHERAPEUTIC
DRUGS

27.
28.
29.
30.
31.
32.
33.

9) DRUGS OF INFLAMMATON &


PYREXIA
10) DRUGS OF
IMMUNOMODULATION
11) DRUGS OF HORMONAL
DISORDERS
12) DERMATOLOGY
13) DRUGS OF OTHER DISEASES
& SYSTEMS

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CHOLINERGIC DRUGS
ADRENERGIC DRUGS
CNS STIMULANTS
NEUROLEPTIC DRUGS
ANXIOLYTIC, HYPNOTIC & SEDATIVE DRUGS
OPIOID ANALGESICS & ANTAGONISTS
ANAESTHETICS
DRUGS USED TO TREAT PARKINSONISM
DRUGS USED TO TREAT EPILEPSY
DRUGS USED TO TREAT DEPRESSION &
ANXIETY DISORDERS
DRUGS USED TO TREAT PSYCHOSIS & MANIA
5-HYDROXYTRYPTAMINE (SEROTININ)
RECEPTOR DRUGS
ANTI ANGINAL DRUGS
DRUGS USED IN CONJESTIVE HEART FAILURE
ANTI ARRHYTHMIC DRUGS
ANTI HYPERTENSIVE DRUGS
ANTI HYPER LIPIDEMIC DRUGS
DRUGS USED TO TREAT DISEASES OF BLOOD

4
5
6
6
7
7
8
9
9
9

DRUGS USED TO TREAT PEPTIC ULCER


ANTI DIARRHOEAL DRUGS (ANTI MOTILITY)
ANTI CONSTIPATIVE DRUGS (LAXATIVES)
DRUGS USED IN INFLAMMATORY BOWL
DISEASE
ANTI EMETICS
DRUGS USED TO TREAT ASTHMA
DRUGS USED TO TREAT OTHER RESPIRATORY
DISEASES
DIURETICS

16
16
16
17

10
10
11
12
13
13
14
15

17
18
18
20

ANTI BACTERIAL DRUGS


ANTI AMOEBIC DRUGS (ANTI PROTOZOAL)
ANTI FUNGAL DRUGS (ANTI PROTOZOAL)
ANTI MALARIAL DRUGS (ANTI PROTOZOAL)
ANTI VIRAL DRUGS
ANTI CANCER DRUGS
ANTI INFLAMMATORY, ANALGESIC &
ANTIPYRATIC DRUGS
34. AUTACOIDS & AUTACOID ANTAGONISTS
35. IMMUNOSUPRESSANT

21
23
23
24
24
25
26

36. ANTI DIABETIC DRUGS


37. STEROID HORMONES
38. DRUGS USED IN DERMATOLOGICAL DISEASES

29
29
31

39. DRUGS USED TO TREAT OBESITY


40. DRUGS USED TO TREAT ERECTILE
DYSFUNCTION
41. DRUGS USED TO TREAT AIDS

32
32

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

27
28

32

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

1) DRUGS OF AUTONOMIC NERVOUS SYSTEM

1. CHOLINERGIC DRUGS (PARASYMPATHETIC)


RECEPTORS
M1

M3,M5
M2,M4

Nm

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AGONISTS
ACETYLCHOLINE
MIOCHOL-E
BETHANCHOL
GENERIC,
URECHOLINE
CARBACHOL
TOPICAL: ISOPTOCARBACHOL,
CARBOPTIC
INTRAOCULAR:
MIOSTAT, CARBASTAT
METHACHOLINE
PILOCARPINE
GENERIC,
ISOPTOCARPINE
ACETYLCHOLINE
MIOCHOL-E
BETHANCHOL
GENERIC, URECHOLINE
CARBACHOL
TOPICAL: ISOPTO
CARBACHOL,
CARBOPTIC
INTRAOCULAR:
MIOSTAT, CARBASTAT
METHACHOLINE
PILOCARPINE
GENERIC, ISOPTOCARPINE
ACETYLCHOLINE
MIOCHOL-E
CARBACHOL
TOPICAL: ISOPTOCARBACHOL,
CARBOPTIC
INTRAOCULAR:
MIOSTAT, CARBASTAT
NICOTINE

ANTAGONISTS
PIRENZEPINES
ATROPINE
GENERIC
OPHTHALMIC:
GENERIC, ISOPTOATROPINE
IPRATROPIUM
GENERIC, ATROVENT
PROPANTHELINE
GENERIC, PROBANTHINE
SCOPOLAMINE
GENERIC

ATROPINE
GENERIC
OPHTHALMIC:
GENERIC, ISOPTO ATROPINE
IPRATROPINE
GENERIC, ATROVENT
PROPANTHELINE
SCOPOLAMINE
GENERIC

ATRACURIUM
SUCCINYLCHOLINE
TUBOCURARINE

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
Ng

ACETYLCHOLINE
MIOCHOL-E
CARBACHOL
TOPICAL: ISOPTOCARBACHOL,
CARBOPTIC
INTRAOCULAR:
MIOSTAT, CARBASTAT
NICOTINE

HEXAMETHONIUM
TRIMETHAPHAN

2. ADRENERGIC DRUGS (SYMPATHETIC)


RECEPTORS
1

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AGONISTS
PHENYLEPHRINES
GENERIC, NEOSYNEPHRINE
DOPAMINE
GENERIC, INTROPIN
EPINEPHRINE
GENERIC,
ADRENALINECHLORIDE
NOREPINEPHRINE
GENERIC, LEVOPHED
APRACLONIDINE
IOPIDINE
CLONIDINE
DOBUTAMINES
GENERIC, DOBUTREX
DOPAMINE
GENERIC, INTROPIN
EPINEPHRINE
GENERIC,
ADRENALINECHLORIDE
ISOPROTERENOL
GENERIC, ISUPREL
NOREPINEPHRINE
METAPROTERENOLS
ALBUTEROL
EPINEPHRINE
GENERIC,
ADRENALINECHLORIDE
ISOPROTERENOL
GENERIC, ISUPREL
TERBUTALINE (TERIL)

ANTAGONISTS
PRAZOSINS
GENERIC, MINIPRESS

YOHIMBINES
PHENOXY BENZAMINE
DIBENZYLINE
METOPROLOLS
GENERIC, LOPRESSOR,
TOPROL
PROPRANOLOL
GENERIC, INDERAL
TIMOLOL
ORAL: GENERIC,
BLOCADREN
OPTHALMIC: GENERIC,
TIMOPTIC
BUTOXAMINES
PROPRANOLOL
GENERIC, INDERAL
TIMOLOL
ORAL: GENERIC,
BLOCADREN
OPTHALMIC: GENERIC,
TIMOPTIC

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

2) DRUGS OF CENTRAL NERVOUS SYSTEM

3. CNS STIMULANTS
1) PSYCHOMOTOR
STIMULANTS

2) PSYCHOTOMIMETIC
DRUGS

AMPHETAMINE
CAFFEINE (CAFERGOT)
METHYLPHENIDATE
NICOTINE
THEOBROMINE
THEOPHYLLINE (THEO PLUS)
FENPHENCYCLIDINE (PCP)
LYSERGIC ACID DIETHYLAMIDE (LSD)
TETRA HYDRO CANNABINOL (THC)

4. NEUROLEPTIC DRUGS
1) PHENOTHIAZINE

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2) BENZISOXAZOLES

CHLORPROMAZINE (THORAZINE)
FLUPHENAZINE (PERMITIL)
PROCHLOR PERAZINE (CLORPAZINE)
PROMETHAZINE
THIORIDAZINE
RISPERIDONE

3) DIBENZODIAZEPINES

CLOZAPINE (CLOZARIL)

4) BUTROPHENONES

HALOPERIDOL (HALDOL)

5) THIOXANTHENES

THIOTHIXENE (NAVANE)

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

5. ANXIOLYTIC, HYPNOTIC & SEDATIVE DRUGS


1) BENZODIAZEPINES

2) BENZODIAZEPINE
ANTAGONIST
3) BARBITURATES

4) NON BARBITURATE
SEDATIVES
5) OTHER ANXIOLYTIC
DRUGS

i)

ANXIOLYTICS
ALPRAZOLAM (XANAX)
CHLORDIAZEPOXIDE (LIBRIU)
CLONAZEPAM (KLONOPIN)
CLORAZEPATE (TRANXENE)
DIAZEPAM (VALIUM)
LORAZEPAM (ATIVAN)
ii)
HYPNOTICS
ESTAZOLAM
FLURAZEPAM (DALMANE)
MIDAZOLAM (VERSED)
QUAZEPAM
TEMAZEPAM (RESTORIL)
TRIAZOLAM
FLUMAZENIL

AMOBARBITAL (AMUTAL)
PHENOBARBITAL (LUMINAL)
PENTOBARBITAL (NEMBUTAL)
SECOBARBITAL (SECONAL)
THIOPENTAL
ANTI HISTAMINES
CHLORAL HYDRATE (NOCTEC)
ETHANOL
BUSPIRONE (BUSPAR)
HYDROXYZINE
ZOLPIDEM

6. OPIOID ANALGESICS & ANTAGONISTS


1) AGONISTS

2) ANTAGONISTS

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a) STRONG AGONISTS
FENTANYL (SUBLIMAZE)
HEROIN (diacetylmorphine)
MORPHINE
MEPRIDINE (DEMEROL)
METHODONE
b) MODERATE AGONISTS
CODEINE
PROPOXYPHENE
NALAXONE (NARCAN)
NALTREXONE
NALMEFENE (REVIX)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
3) MIXED AGONISTSANTAGONISTS

BUTORPHANOL (STADOL)
NALBUPHINE (NUBAIN)
PENTAZOCINE (TALWIN)

7. ANAESTHETICS
1) ADJUNCTS TO
ANAESTHETICS

2) GENERAL
ANAESTHETICS

3) LOCAL ANAESTHETICS

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a) PRE ANAESTHETIC MEDICATION


ANTI CHOLINERGICS
ANTI EMETICS
BARBITURATES
BENZODIAZEPINES
OPOIDS
b) MUSCLE RELAXANTS
ATRACURIUM (TRACRIUM)
SUCCINYLCHOLINE (ANECTINE)
VECURONIUM (NORCURON)
a) INHALANT ANAESTHETICS
ENFLURANE (ETHRANE)
HALOTHANE (GENERIC, FLUOTHANE)
ISOFLURANE (FORANE)
METHOXY FLURANE (PENTHRANE)
NITROUS OXIDE
SEVOFLURANE
b) INTRAVENOUS ANAESTHETICS
i.
BARBITURATES
METHO HEXITAL (BREVITAL)
THIAMYLAL (SURITAL)
THIOPENTAL (PENTOTHAL)
ii.
BENZODIAZEPINES
DIAZEPAM (GENERIC, VALIUM)
LORAZEPAM (GENERIC, ATIVAN)
MIDAXOLAM (VERSED)
iii.
OPIOIDS
FENTANYL
MORPHINE
iv.
NEUROLEPTIC
DROPERIDOL & FENTANYL
v.
DISSOCIATIVE
KETAMINE (KETALAR)
vi.
PROPOFOL (DIPRIVAN)
vii.
ETOMIDATE
BUPIVACAINE (GENERIC, MARCAINE)
LIDOCAINE (GENERIC, XYLOCAINE)
PROCAINE (GENERIC, NOVOCAIN)
TETRACAINE (PONTOCAINE)

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

8. DRUGS USED TO TREAT PARKINSONISM

AMANTADINE (SUMMETREL)
ANTI MUSCARINIC AGENTS
BROMOCRIPTINE (PARLODEL)
CARBIDOPA (LODOSYN)
DEPRENYL
LEVODOPA (DOPAR, LARODOPA)

9. DRUGS USED TO TREAT EPILEPSY

CARBAMAZEPINE (TEGRETOL)
CLONAZEPINE (KLONOPIN)
CLORAZEPATE (TRANXENE)
DIAZEPAM (GENERIC, VALIUM)
ETHOSUXIMIDE (ZARONTIN)
GABA PENTIN
LAMOTRIGINE
PHENOBARBITAL (GENERIC, LUMINAL)
PHENYTOIN (GENERIC, DILANTIN)
PRIMIDONE (GENERIC, MYSOLINE)
VALPROIC ACID (GENERIC, DEPAKENE

10. DRUGS USED TO TREAT DEPRESSION & ANXIETY DISORDERS


1) NOREPINEPHRINE
REUPTAKE INHIBITORS

2) SELECTIVE SEROTONIN
REUPTAKE INHIBITORS

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a) TERTIARY AMINE TRICYCLICS


AMITRIPTYLINE (GENERIC, ELAVIL)
AMOXAPINE (ASENDIN)
DESIPRAMINE (NORPRAMIN)
DOXEPIN (GENERIC, SINEQUAN)
IMIPRAMINE (GENERIC, TOFRANIL)
MAPROTILINE (LUDIOMIL)
TRIMIPRAMINE (SURMONTIL)
b) SECONDARY AMINE TRICYCLICS
MAPROTILINE (LUDIOMIL)
NORTRIPTYLINE (PAMELOR, MOTIVAL)
PROTRIPTYLINE (VIVACTIL)
CITALOPRAM (CELEXA)
FLUOXETINE ( PROZAC)
FLUVOXAMINE (LUVOX)
NETAZODONE
PAROXETINE (PAXIL)

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

3) ATYPICAL
ANTIDEPRESSANTS

4) MONOAMINE OXIDASE
INHIBITORS

SERTRALINE (ZOLOFT)
TRAZODONE (GENERIC, DESYREL)
VENLAFAXINE (EFFEXOR)
BUPROPION (WELLBUTRIN)
MIRTAZAPINE (REMERON)
NEFAZODONE (SERZONE)
TRAZODONE (DESYRIL)
ISOCARBOXAZID (MARPLAN)
PHENELZINE (NARDIL)
SELEGILINE (ELDEPRYL)
TRANYLCYPROMINE

11. DRUGS USED TO TREAT PSYCHOSIS & MANIA


1) PHENOTHIAZINS

2) THIOXANTHENES
3) OTHER HETROCYLIC
COMPOUNDS

4) LITHIUM SALTS
(FOR MANIA & AS MOOD
STABILIZING AGENT)

CHLORPROMAZINE (THORAZINE)
FLUPHENAZINE (PERMITIL)
MESORIDAZINE (SERENTIL)
PERPHENAZINE (TRILAFON)
RIFLUOPERAZINE (STELAZINE)
THIORIDAZINE (SERENTIL)
CHLORPROTHIXENE (TARACTAN)
THIOTHIXENE (NAVANE)
CLOZAPINE (CLOZARIL)
HALOPERIDOLE (HALDOL)
LOXAPINE (LOXITANE)
OLANZIPINE (ZYPREXA)
PIMOZIDE (ORAP)
RESPERIDONE (RISPERDAL)
LITHIUM CARBONATE (CAMCOLIT, LITRISON, LOCAM)
LITHIUM CITRATE
LITHIUM SULFATE

12. 5-HYDROXYTRYPTAMINE (SEROTONIN) RECEPTOR DRUGS


1) AGONISTS

2) ANTAGONISTS

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BUSPIRONE (BUSPAR)
IPSAPERONE
RIZATRIPTAN (MAXALT)
SUMATRIPTAN (IMITREX)
ZOLMITRIPTAN (ZOMIG)
DOLASETRON (ANZEMET)
GRANISETRON (KYTRIL)
KETANSERIN (SUFREXAL)
ONDANSETRON (ZOFRAN)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

10

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

3) DRUGS OF CARDIOVASCULAR SYSTEM

13. ANTI ANGINAL DRUGS


1) ORGANIC NITRATES AND
NITRITES

2) -BLOCKERS

3) Ca2+ CHANNEL BLOCKERS

4) ANGIOTENSIN
CONVERTING ENZYME
(ACE) INHIBITOR
5) OTHER CORONARY
VASODILATORS

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AMYL NITRATE (GENERIC)


ISOSORBIDE DINITRATE (GENERIC, ISORDIL)
ISOSORBIDE MONONITRATE (ISMO)
NITRO GLYCERINE OR GLYCERINE TRINITRATE
SUBLINGUAL: GENERIC
ORAL SUSTAINED RELEASE: GENERIC, NITROTIME
PARENTERAL: GENERIC
TRANSDERMAL PATCHES: GENERIC, NITREK,
NITRO-DUR, TRANSDERM-NITRO
TOPICAL OINTMENT: GENERIC, NITRO-BID
PENTA ERYTHRITOL TETRA NITRATE
ACETBUTOLOL
ATENOLOL (TENORMIN, ATELOR)
METOPROLOL
PROPRANOLOL
AMLODIPINE (AMLOCARD, AMLOPIN)
DILTIAZEM (CALCARD)
FELODIPINE
NICARDIPINE
NIFEDIPINE (ADALAP)
NITREDIPINE
VERAPAMIL (CALAN)
CAPTOPRIL (CATOPER, APTIL)
ENALAPRIL (CARDACE, CARDIL)
PERINDOPRIL
DIPYRIDAMOL (PERSANTIN)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

11

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

14. DRUGS USED IN CONJESTIVE HEART FAILURE


1) CARDIAC GLYCOSIDES

2) -BLOCKERS

3) RENIN ANGIOTENSIN
SYSTEM BLOCKERS

4) DIURETICS

5) DIRECT VASODILATORS

6) INOTROPIC AGENTS

7) ALDOSTERONE
ANTAGONISTS
8) -ADRENERGIC AGONIST
(FOR ACUTE HEART
FAILURE ONLY)

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a)

DIGITOXIN (GENERIC, CRYSTODIGIN)


DIGOXIN (LANOXIN)
OUABAIN
ATENOLOL
CURVEDILOL
METOPROLOL
PROPRANOLOL
ACE INHIBITOR
CAPTOPRIL (CATOPER, APTIL)
ENALAPRIL (CARDIL)
FOSINOPRIL
LISINOPRIL
QUINAPRIL (QUINE)
RAMIPRIL
b) ANGIOTENSIN TYPE 1 RECEPTORS BLOCKERS
CONDESERTAN
LOSARTAN (COZAAR, HYZAAR)
TELMISARTAN
VALSARTAN (DIOVAN, VALTREX)
BUMETANIDE
FUROSIMIDE (LASIX)
HYDRO CHLORO THIAZIDE
METOLAZONE
HYDRALAZINE
ISO SORBIDE DINITRATE
SODIUM NIRO PRUSSIDE
AMRINONE (INOCOR)
DIGITOXIN
DIGOXIN (GENERIC, LANOXIN)
DOBUTAMINE (DOBUTREX)
MILRINONE
SPIRONOLACTONE

DOBUTAMINE (DOBUTREX)
DOPAMINE (GENERIC, INTROPIN)
ISOPERANALINE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

12

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

15. ANTI ARRHYTHMIC DRUGS


1) Na+ CHANNEL
BLOCKERS

2) -ADENO RECEPTOR
BLOCKERS
(Ca+ BLOCKERS INDIRECTLY)
3) Ca+ CHANNEL BLOCKERS
(Ca+ BLOCKERS DIRECTLY)
4) K+ CHANNEL BLOCKERS

5) OTHER S

DISOPYRAMIDA (GENERIC, NORPACE)


PROCAINAMIDE (GENERIC, PROCAN SR)
QUINIDINE (GENERIC, QUINIDEX)
LIDOCANE (GENERIC, XYLOCAINE)
MEXILETINE(MEXITIL)
TOCAINIDE
FLECIAINIDE (TAMBOCOR)
PROPAFENONE
ESMOLOL
METOPROLOL
PROPANOLOL
DILTIAZEM (CARDIZEM)
VERAPAMEL (CALAN)
AMIODAPRONE (CORDARONE)
DOFETILIDE
SOTALOL
ADENOSINE (ADNOCARD)
DIGOXIN

16. ANTI HYPERTENSIVE DRUGS


1) ACE INHIBITORS
(ANGIOTENSIN
CONVERTING ENZYME)

2) ANGIOTENSIN II
RECEPTOR
ANTAGONISTS
3) Ca2+ CHANNEL BLOCKERS

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a)

BENAZEPRIL
CAPTOPRIL (CAPOTEN)
ENALAPRIL (VASOTEC)
FOSINOPRIL (MONOPRIL)
LISINOPRIL (PRINVIRIL, ZESTRIL)
MOEXIPRIL (UNIVASC)
QUINAPRIL (ACCUPRIL)
RAMIPRIL (ALTACE)
TRANDOLAPRIL (MAVIK)
IRBESARTAN
LOSARTAN (COZAAR)
TELMISARTAN
VALSARTAN (DIOVAN, VALTREX)
DIPHENYL ALKYL AMINS:
VERAPAMIL (CALAN)
b) BENZO THI AZEPINES:
DILTIAZEN (DILZEM, ETIZEM)
c) DI HYDRO PYRIDINES:
AMLODIPINE
FELODIPINE
ISRADIPINE

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

13

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

4) -ADRENO RECEPTOR
BLOCKERS
5) CENTRALLY ACTING
ADRENERGIC DRUGS
6) VASODILATORS
7) -BLOCKERS

8) DIURETICS

NICARDIPINE
NIFEDIPINE (ADALAT)
NISOLDIPINE
DOXAZOSIN (DOXCIL)
PRAZOSIN (MINIPRES)
TERAZOSIN (HYTRIN)
CLONIDINE (GENERIC, CATAPRES)
-METHYL DOPA
HYDRALAZINE (GENERIC, APRESOLINE)
MINOXIDIL (LONITEN)
ATENOLOL
LABETALOL
METOPROLOL
NADOLOL (NAFACIN)
PROPRANOLOL
TIMOLOL
(CONSULT DIURETIC DRUGS)

17. ANTI HYPER LIPIDEMIC DRUGS


1) HMG-COA REDUCTASE
INHIBITORS (STATINS)
(3-HYDROXY-3-METHYL
GLUTARYL CO ENZYME A
REDUCTASE)
2) FIBRATES
3) NIACIN
4) BILE ACID SEQUESTANTS

5) CHOLESTEROL
ABSORPTION
INHIBITORS

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ATORVASTATIN (LIPITOR)
FLUVASTATIN
LOVASTATIN (MEVACOR)
PRAVASTATIN (PRAVACHOL)
RUSUVASTATIN
SIMVASTATIN (SIMVACOR, VASTIN)
FENO FIBRATES
GEM FIBRATES (LOPID)
NICOTINIC ACID (NICOTRIM)

CHOLESTYRAMINE (QUESTRAN)
COLESEVELAM
COLESTIPOL (COLESTID)
EZITIMIDE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

14

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

4) DRUGS ACTING ON BLOOD

18. DRUGS USED TO TREAT DISEASES OF BLOOD


1) PLATELET INHIBITORS

2) ANTI COAGULANTS

3) THROMBOLYTIC AGENTS

4) TREATMENT OF
BLEEDING

5) TREATMENT OF ANEMIA

6) TREATMENT OF SICKLE
CELL ANEMIA

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ASPIRIN (DISPRIN, ANAPRIN, ANTICLOT, Ec-PRIN)


DIPYRIDAMOLE
TICLOPIDINE
ENOXAPRIN
HEPARIN (GENERIC, CALCIPARINE)
WARFARIN (GENERIC, COUMADIN)
ALTEPLASE (tPA)
ANISTREPLASE
STREPTOKINASE
UROKINASE
AMINOCAPROIC ACID
PROTAMINE SULFATE
TRENEXAMIC ACID
VITAMIN K
CYANOCOBALAMIN (B12) (GENERIC, CYNOTONE)
ERYTHROPOIETIN (EPREX, ESSENTIALE)
FOLIC ACID
IRON (IRZAPYRIN, ISMO 20)
HYDROXY UREAS

TARIQ AHMAD | tareeqahmad@hotmail.com


DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

15

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

5) DRUGS OF GASTRO INTESTINAL TRACT

19. DRUGS USED TO TREAT PEPTIC ULCER


1) H2 BLOCKERS

2) PROTON PUMP
INHIBITORS

3) MUCOSAL
STRENGTHENED
4) ANTI BIOTICS
5) ANT ACIDS

CIMETIDINE (TAGMET)
FAMOTIDINE (PEPSID)
NIZATIDINE (AXID)
RANITIDINE (ZANTAX)
ESOMEPRAZOL
LANSOPRAZOLE (LANZID, LANZIT, LANZAC)
OMEPRAZOLE (OMEZOL, OMEGA)
RABEPRAZOLE
MISOPROSTAL (MITOMYCIN, MITISTATE)

AMOXACILINE
CALITHSOMYCINE
ALUMINIUM HYDROXIDE Al (OH)3
MAGNESIUM HYDROXIDE Mg (OH)2
SODIUM BICARBONATE
NaHCO3

20. ANTI DIARRHOEAL DRUGS (ANTI MOTILITY)

DIFENOXIN
DIPHENOXYLATE (LOMOTIL, MOTILEX)
LOPERAMIDE (LOPRIN)

21. ANTI CONSTIPATIVE DRUGS (LAXATIVES)


1) IRRITANT AND
STIMULANT

2) BULKING AGENT

732

ALOE
BISACODYL (GENERIC, BICOLAX)
CASCARA
CASTER OIL
SENNA
AGAR
BRAN
HYDROPHILLIC COLLOIDS
METHYL CELLULOSE
POLY ETHYLENE GLYCOL (COLONIC LEVAGE)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

16

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

3) STOOL SOFTNERS

PSYLLIUM SEEDS
SALINE CATHARTICS
DOCUSATE SODIUM
GLYCERINE SUPPOSITORIES
MINERAL OIL

22. DRUGS USED IN INFLAMMATORY BOWL DISEASE


1) ANTI INFLAMMATORY
DRUGS

AZA THIOPRINE (IMPURA)


(6-MEROCAPTO PURINE OR 6MP OR PURINETHOL)
CYCLOSPORIN (CYCLOZ)
GLUCOCORTICIODS & ACTH
MESALAZINE (ASACOL, MESAZINE)
SULFASALAZINE (SALAZINE, SALAZODINE)

23. ANTI EMETICS


1) SEROTONIN 5-HT3
ANTAGONISTS
2) DOPAMINE BLOCKERS

3) ANTI HISTAMINE

732

DULASETION
GRANISETRON
ONDANSETION
DOMPERIDONE (EMIDONE, MOTIL, MOTILIUM)
DROPERIDOL
HALOPERIDOL (HALOTHANE, HAPRO, HARTEN)
BELLADONA ALKALOIDS (BENADRYL)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

17

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

6) DRUGS OF RESPIRATORY SYSTEM

24. DRUGS USED TO TREAT ASTHMA


1) -ADRENERGIC AGONISTS
(USED AS INHALENTS)

a) SHORT ACTING
ALBUTEROL (PROVENTIL)
LEVALBUTEROL (XOPENEX)
METAPROTERENOL (ALUPENT)
PIRBUTEROL (MAXAIR)
TERBUTALINE (BRETHAIRE)
b) LONG ACTING
BITOLTEROL (TORNALATE)
SALMETEROL XINAFOATE (SEREVENT)
BECLOMETHASONE DIPROPIONATE (BECLOVENT
VANCERIL)
FLUTICASONE PROPIONATE (FLOVENT)
TRIA AMACINOLONE ACETONIDE (AZMACORT)
a) LEUKOTRIENE RECEPTOR ANTAGONISTS
MONTELUKAST (SINGULAIR)
ZAFIRLUKAST (ACCOLATE)
b) LEUKOTRIENE SYNTHESIS INHIBITORS
ZILEUTON (ZYFLO)
CROMOLYN SODIUM
NEDOCROMIL SODIUM
THEOPHYLLINE (THEO PLUS)

2) GLUCOCORTICOIDS
(CORTICOSTEROIDS)
(USED AS INHALENTS &
SYSTEMIC AS WELL)
3) LEUKOTRIENE RECEPTOR
ANTAGONISTS &
LEUKOTRIENE SYNTHESIS
INHIBITORS
4) CROMOLYN &
NEDOCROMIL
5) BRONCHODILATORS
6) CHOLINERGIC
ANTAGONISTS

IPRATROPIUM (ATROVENT)

25. DRUGS USED TO TREAT OTHER RESPIRATORY DISEASES


1) DRUGS USED TO TREAT
RHINITIS

2) DRUGS USED TO TREAT


CHRONIC OBSTRUCTIVE
PULMONARY DISEASE

732

-ADRENERGIC AGONISTS
ANTIHISTAMINES
CORTICOSTEROIDS
CROMOLYN
-ADRENERGIC AGONISTS
CORTICOSTEROIDS
IPRATROPIUM (CHOLINERGIC ANTAGONIST)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

18

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
3) DRUGS USED TO TREAT
COUGH

732

(OPIATES)
BENZONATATE (TESSALON)
CARAMIPHEN
DEXTROMETHORPHAN
DIPHENYL HYDRAMINE
NOSCAPINE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

19

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

7) DRUGS OF RENAL FUNCTION

26. DIURETICS
1) CARBONIC ANHYDRASE
INHIBITORS
2) LOOP DIURETICS
3) THIAZIDES

4) POTASSIUM SPARING
DIURETICS
(ALDOSTERONE ANTAGONISTS)
5) OSMOTIC DIURETICS

732

ACETAZOLAMIDE
DICHLORPHENAMIDE
METHAZOLAMIDE
ETHACRYNIC ACID (EDECRIN)
FUROSEMIDE (LASIX)
CHLOROTHIAZIDE (DIURIT)
CHLORTHALIDONE (HYGROTON)
HYDROCHLOROTHIAZIDE (COZEAL)
INDAPRAMIDE
(LAZOL)
METOLOZANE
(ZYROKOT)
AMILORIDE (MIDAMOR)
TRIAMTERENE (MAXZIDE)

MANNITOL (GENERIC, NAOLAX)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

20

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

8) CHEMOTHERAPEUTIC DRUGS

27. ANTI BACTERIAL DRUGS

732

1)

SULPHONAMIDES

2)

CO-TRIMOXAZOLE

3)

QUINOLONES &
FLOROQUINOLONES

4)

AMINO GLYCOSIDES

a) ORAL ABSORABLE
i. SHORT ACTING
SULFAMETHIZOLE (PROKLAR)
SULFISOXAZOLE (PEDIAZOLE)
ii. INTERMEDIATE ACTING
SULFADIAZINE (GENERIC, ANTRIMA)
SULFAMETHOXAZOLE
iii. LONG ACTING
SULFADOXINE (METAFIN)
b) TOPICAL
i. DERMAL USE
SILVER SULFADIAZINE
MEFINIDE
ii. MUCOSAL USE
SULFACETAMIDE
TRIMETHOPRIM : SULPHAMETHOXAZOLE
1
:
5
(BACTRIM, AMOXAZOLE)
a) QUINOLONES
CINUXACIN
NALIDIXIC ACID (NALACID)
b) FLOROQUINOLONES
CIPROFLOXACIN (LUCID, CIPROXIN)
LEVOFLOXACIN (LEVOCIL)
LOMEFLOXACIN (LOMOTIL)
NORFLOXACIN (NOROXIN)
OFLOXACIN (OFLOX, TARIVID)
SPARFLOXACIN (SPARAXIN)
a) AMINO GLYCOSIDES CAUSING COCLEAR NERVE
DAMAGE
AMIKACIN (AMIKIN)
KANAMYCIN (KANACYN)
b) AMINO GLYCOSIDES CAUSING VERTIBULAR
NERVE DAMAGE
GENTAMYCIN (GENERIC, GENTICYN)
STREPTOMYCIN (GENERIC, STRIKE)
TOBERAMYCIN (ABBOCIN)
c) AMINO GLYCOSIDES USED TOPICALLY
NEOMYCIN (GENERIC, CICATRIN)
PAROMOMYCIN

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

21

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

732

5)

PENICILLINS

6)

CEPHALOSPORIN

a) NARROW SPECTRUM PENICILLINS


i) SHORT ACTING PENICILINS
PENICILLIN G (BENZYL PENICILLIN)
PENICILLIN V (PHENOXY METHYL
PENICILLIN)
ii) PENICILLINASE RESISTANT PENICILLINS
CLOXACILLIN (GENERIC, AMPICLOX)
FLUCLOXACILLIN (FLUCOL)
METHICILLIN
NAFICILLIN
iii) LONG ACTING PENICILLINS
PROCAINE PENICILLIN (KANACILLIN)
BENZATHIN (LAPEN)
b) BROAD SPECTRUM PENICILLINS
AMPICILLIN (GENERIC, AMPICLOX)
AMOXYCILLIN (GENERIC, AMOXIL)
BACAMPICILLIN (BACILLOCID)
c) ANTI PSEUDOMONAL PENICILLINS
CARBENICILLIN
PIPERACILLIN
d) -LACTAMASE INHIBITOR
CLAVULANIC ACID
SULBACTUM
TAZOBACTAM (TAZOCIN)
a) FIRST GENERATION CEPHALOSPORIN
CEPHRADIN (BIOCEF)
CEPHALOTHIN
CEPHALEXIN (CEFLIN)
CEFADROXIL (CEDROX)
CEFAZOLIN (KEFZOL)
CEPHAPIRIN
b) SECOND GENERATION CEPHALOSPORIN
CEFACLOR (CECLOR)
CEFPROXIL
CEFUROXIME (CEFUZINE)
CEFPRODOXIME
LORACARBEF
c) THIRD GENERATION CEPHALOSPORIN
CEFOTAXIME (CLAFORAN)
CEFTRIAXONE (CEFCIN)
CEFIXIME (CEFIX)
CEFOPERAZONE (CEFOBID)
CEFTAZIDIME
MOXALACTUM
d) FORTH GENERATION CEPHALOSPORIN
CEFEPIME (CEFGARD, CEFIM, CEFIX)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

22

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
7)

TETRACYCLINES

8)

MACROLIDES

9)

CHLORAMPHENICOL

a) SHORT ACTING TETRACYCLINES


TETRACYCLINE
OXY TETRACYCLINE
CHLOR TETRACYCLINE
b) INTERMEDIATE ACTING TETRACYCLINES
DEMECLOCYCLINE
METHACYCLINE
c) LONG ACTING TETRACYCLINES
DEOXY CYCLINE
AZITHROMYCINE (AZIT)
CARBOMYCINE
CLARITHROMYCINE (CLARICID)
ERYTHROMYCINE (ERYTHROCINE, EMYCINE)
PRITIM

28. ANTI AMOEBIC DRUGS (ANTI PROTOZOAL)


1) LUMENAL DRUGS

DILOXAMIDE (DILOXAZOLE)

2) SYSTEMIC DRUGS

CHLOROQUINE (QUINE)
DEHYDRO EMETINE
EMETINE
METRONIDAZOLE (FLAGYL, AMEZOLE, FLEZOLE)

3) MIXED DRUGS

29. ANTI FUNGAL DRUGS (ANTI PROTOZOAL)


1)

2)

3)

1)

732

( ACCORDING TO THEIR CHEMICAL NATURE )


POLYENES
AMPHOTERICIN-B (AMPICIL)
NATAMYCIN
NYSTATIN (NINSTAT)
AZOLE DERIVATIVES
FLUCONAZOLE (DERECON, FLUGAL)
ITRACONAZOLE
KETOCONAZOLE
MISCELLANEOUS DRUGS
FLUCYPTOCINE
GRIESEOFULRIN
( ACCORDING TO THEIR SITE OF ACTION )
DRUGS FOR
AMPHOTERICIN-B (AMPICIL)
SUBCUTANEOUS &
FLUCONAZOLE (DERECON, FLUGAL)
SYSTEMIC MYCOSIS
FLUCYTOCINE
KETOCONAZOLE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

23

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
2) DRUGS FOR SUPERFICIAL
MYCOSIS

CLODRIMAZOLE
GRISEOFULVIN
MYSTATIN

30. ANTI MALARIAL DRUGS (ANTI PROTOZOAL)


1) QUININE & ITS SALTS
2) 9-AMNO ACRIDINES

MEPOCRINE

3) 4-AMINO QUINOLONES

CHLOROQUINE (QUINE)

4) 8-AMINO QUINIDINES

PRIMAQUINE

5) BIGUANIDES

PROGUANID

6) DIAMINO PYRIMIDINES

PYRIMETHAMINE
TRIMETHOPRIM (ANTRIMA)

7) SULPHONAMIDES &
DAPSONE

31. ANTI VIRAL DRUGS


1) DRUGS INHIBITING
EARLY PROTEIN
SYNTHESIS
2) DRUGS INHIBITING LATE
PROTEIN SYNTHESIS
3) DRUGS INHIBITING
NUCLEAC ACID
SYNTHESIS

4) DRUGS INHIBITING
BOTH NUCLEAC ACID &
PROTEIN SYNTHESIS
5) DRUGS INHIBITING
ADSORPTION &
PENETRATION OF
SUSCEPTIBLE CELLS

732

GUANIDINE
HYDROXY BENZYL BENZIMIDAZOLE

FLURO PHENYL ALANINE


METHESAZONE
5-FLURO URACIL (GENERIC, CURACIL, FLURACIL)
ACYCLOVIR (ZOVIRAX)
CYTARABIN
GANCICLOVIR (CYTOVENE)
RIBAVIRIN (REBETOL)
INTERFERONES (INTRON)

AMANTADINE (SYMMETREL)
GAMMA-GLOBULIN

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

24

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

32. ANTI CANCER DRUGS


1) ANTI METABOLITES

2) ANTI BIOTICS

3) ALKYLATING AGENTS

4) MICROTUBULE
INHIBITORS

5) STEROID HORMONES &


THEIR ANTAGONISTS

6) OTHERS

732

5-FLUROURACIL (GENERIC, CURACIL, FLURACIL)


6-MERCAPTOPURINE
6-THIOGUANINE
CYTARABINE
FLUDARABINE
METHOTREXATE
BLEOMYCINE
DACTINOMYCIN (DAFLON, DALACIN C, DALACIN T)
DAUNORUBICIN
IDARUBICIN (ZAVEDOS, IDOGIL)
PLICAMYCIN
CARMUSTINE & LOMUSTINE
CYCLOPHOSPHAMIDE & IFOSFAMIDE
MECHLORETHAMINE
STREPTOZOTOCIN
NAVELBINE
PACLITAXEL (TAXOL)
VINBLASTINE (VELBE)
VINCRISTINE (ONCOVIN)
AMINOGLUTETHIMIDES
ESTROGENS
FLUTAMIDE
GOSERELIN
LEUPROLIDE
PREDNISONE
TAMOXIFEN (TAMOXIN)
ASPARAGINASE
CISPLATIN (ZORID) & CARBOPLATIN
ETOPOSIDE
INTERFERONS (INTRON)
PROCARBAZINE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

25

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

9) DRUGS OF INFLAMMATON & PYREXIA

33. ANTI INFLAMMATORY, ANALGESIC & ANTIPYRATIC DRUGS


1) NON SELECTIVE
CYCLOOXYGENASE
(COX) INHIBITOR

i.

ii.

iii.

iv.

v.

vi.

vii.

viii.
2) SELECTIVE
CYCLOOXYGENASE-2
(COX-2) INHIBITORS
3) DRUGS USED TO TREAT
GOUT

732

SALICYLIC ACID DERIVATIVES


ASPIRIN (DISPRIN, ANAPRIN, Ec-PRIN)
DIFLUNISAL (DOLOBID)
OLSALAZIN
SALSALATE (DISALCID)
SULFASALAZIN
PARA-AMINO PHENOL DERIVATIVES
ACETAMINOPHEN (PARACETAMOL,
PANADOL, DISPROL)
ARYL PROPIONIC ACIDS
FENOPROFEN (NELFON)
FLURBIPROFEN
IBUPROFEN (BRUFEN)
KETOPROFEN (ORUDIS)
NAPROXEN (ALEVEA)
OXAPRAZIN
INDOLE ACETIC ACID
INDOMETHACIN (INDOCIN)
SULINDAC (CLINORIL)
ENOLIC ACIDS
MELOXICAM (MOBIC)
PIROXICAM (FELDENE)
FENAMATES
MECLOFENAMIC ACID
MEFENAMIC ACID (PONSTAN)
HETROARYL ACETIC ACIDS
DICLOFENAC (DICLORAN)
KETOROLAC (TORADOL)
TOLMETIN (TOLECTIN)
ALKANONES
NABUMETONE (RELAFEN)
CELECOXIB (CELEBREX)
ETODOLAC (LODINE)
NIMESULID
ROFECOXIB (VIOXX)
ALLOPURINOL
COLCHICINE
PROBENECID
SUPFIN PYRAZON

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

26

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
4) DRUGS USED TO TREAT
ARTHRITIS

CHLOROQUINE
D-PENICILLAMINE
GOLD SALTS
METHOTREXATE (GENERIC, UNITREXATE)

34. AUTACOIDS & AUTACOID ANTAGONISTS


1) PROSTAGLANDINS

2) H1 ANTI HISTAMINES

3) H2 ANTI HISTAMINES

4) DRUGS USED TO TREAT


MIGRAINE HEADACHE

732

CARBOPROST
DINOPROST
DINOPROSTONE
MISOPROSTOL
CYCLIZINE (MIGRIL)
DI MENHYDRINATE
DI PHEN HYDRAMINE
MECLIZINE
CIMETIDINE (CIMET)
FAMOTIDINE (FENCID, FAMTINE, ZEPSIN)
NIZATIDINE
RANITIDINE (PEPTAC, ZANTACNULCER)
-BLOCKERS
DI HYDRO ERGOTAMINE
ERGOTAMINE
METHY SERGIDE
SUMATRIPTAN

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

27

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

10)

DRUGS OF IMMUNOMODULATION

35. IMMUNOSUPRESSANT
1) NON SELECTIVE
IMMUNOSUPRESSANT
2) ANTI BODIES
3) SELECTIVE
IMMUNOSUPRESSANT

732

AZATHIOPRINE (AMORIN, IMURAN)


MICOPHENOLATE MOFETIL
ANTI LYMPHOCYTE & ANTI THYMOCYTE GLOBULIN
MUROMONAB-CD3
CYCLOSPORIN (SANDIMMUN)
TACROLIMUS

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

28

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

11)

DRUGS OF HORMONAL DISORDERS

36. ANTI DIABETIC DRUGS


1) INSULIN

2) ORAL HYPOGLYCEMIC
DRUGS

INSULIN ZINC SUSPENSION


ISOPHENE INSULIN (HUMULIN-N, INSULATARD)
PROTAMINE ZINC INSULIN
SEMILENTE INSULIN
ULTRALENTE INSULIN
ZINC INSULIN
ACETOHEXAMIDE
CHLORPROPAMIDE (DIABENESE, DIABTUS)
GLIPIZIDE (GLIPASE, GLIZID)
GLYBURIDE
METFORMIN (GENERIC, DIABIN, GLUCODAL)
TOLAZAMIDE
TOLBUTAMIDE

37. STEROID HORMONES


1) ESTROGENS

2) ANTI ESTROGENS
3) PROGESTINS

4) ANTI PROGESTINS
5) ANDROGENS

732

CHLOROTRIANISENE
DI ETHYL STILBESTROL
ESTRADIOL
ESTRIOL
ESTRONE
ETHINYL ESTRADIOL
MESTRANOL
QUINESTROL
CLOMIPHENE
TAMOXIFEN (GENERIC, TAMOFEN, TAMOXIN)
HYDROXYPROGESTRON
MEDROXYPROGESTRON
PROGESTRON (GENERIC, MENSTROGEN)
NORETHINDRONE
NORGESTREL
MIFEPRISTONE
DANAZOL (DANATRIS, DANOCRINE)
FLOXYMESTERONE
NANDROLONE (ABOLON, DURALONE)
STANOZOLOL
TESTOSTERONE CYPIONATE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

29

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION
6) ANTI ANDROGENS

7) CORTICOSTEROIDS

8) INHIBITORS OF
ADRENOCORTICOID
BIOSYNTHESIS

732

CYPROTERONE ACETATE
FINASTERIDE (GENESIS, PROSCAR)
FLUTAMIDE (FLUTAMIDE GADOR)
BECLOMETHAZONE
BETA METHAZONE
CORTISONE (COTRIMAX)
DEXAMETHOSONE (DECADRON)
DESOXYCORTICOSTERONE
HYDROCORTISONE
METHYLPREDNISOLONE
PREDNISONE
PREDNISOLONE(GENERIC, STERON)
AMINOGLOTETHIMIDE
KETOCONAZOLE (KETO, KONAZOLE)
MEFIPRISTONE
SPIRONOLACTONE (STEMETIL)

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

30

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

12)

DERMATOLOGY

38. DRUGS USED IN DERMATOLOGICAL DISEASES


1) GLUCOCORTICOIDS

2) TREATMENT OF
PRURITIS

732

a) TOPICAL
BETA METHOSONE (DIPROLENE)
CLOBETASOL (TEMOVATE)
DIFLORASONE (FLORONE)
HYDROCORTISONE (HYTONE)
TRIAMCILONE (ARISTOCORT)
b) SYSTEMIC
PREDNISONE
PREDNISOLONE
a) TOPICAL
ANTIHISTAMINES
CAPSAICIN
DOXEPIN
MENTHOL
PHENOL
b) SYSTEMIC
ANTIHISTAMINES
DOXIPIN
STEROIDS

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

31

PHARMACOLOGICAL CLASSIFICATION OF DRUGS


FIRST EDITION

13)

DRUGS OF SOME OTHER DISEASES

39. DRUGS USED TO TREAT OBESITY


1) ANOREXIC AGENTS
2) LIPASE INHIBITORS

PHENTERMINE
SIBUTRAMINE
ORLISTAT

40. DRUGS USED TO TREAT ERECTILE DYSFUNCTION

SILDENAFIL (VIAGRA)
ALPROSTADIL (CAVERJECT)

41. DRUGS USED TO TREAT AIDS


1) HIV PROTEASE
INHIBITORS

2) REVERSE
TRANSCRIPTASE
INHIBITORS

3) OTHERS

732

a)

AMPRENAVIR (AGENERASE)
INDINAVIR (CRIXIVAN)
NELFINAVIR (VIRACEPT)
RITONAVIR (NORVIR)
SAQUINAVIR
NON NUCLEOSIDE REVERSE TRANSCRIPTASE
INHIBITORS
DELAVIRDINE (RESCRIPTOR)
EFAVIRENZ (SUSTIVA, STOCRIN)
NEVIRAPINE (VIRAMUNE)
b) OTHER REVERSE TRANSCRIPTASE INHIBITORS
ABACAVIR (ZIAGEN)
ADEFOVIR (PREVEON, HEPSERA)
DIDANOSINE (VIDEX)
LAMIVUDINE (EPIVIR)
STAVUDINE (ZERIT)
ZALCITABINE (HIVID)
ZIDOVUDINE

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DEPARTMENT OF PHARMACY, UNIVERSITY OF LAHORE

32

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