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Inflammation

NSAIDS
Non-Selective COX Inhibitors
Salicylates (Aspirin)
Diflunisal
Acetaminophen (Tylenol)
Indoles
Indomethacin
Sulindac
Propionic acid deriv & analogs
Ibuprofen
Flurbiprofen
Naproxen
Oxaprozin
Ketoprofen
Fenoprofen
Enolic Acids
Piroxicam
Heteroaryl Acetic Acids
Ketorolac
Selective COX-2 Inhibitors
Celecoxib
Rofecoxib
Meloxicam
Valdecoxib

Histamine
H1 Receptor Antagonists (antihistamines)
Ethanolamine derivs: diphenhydramine
Ethylenediamine derivs: tripelennamine
Piperazine derivs: cyclizine
Phenothiazine derivs: promethazine
Alkylamine derivs: chlorpheniramine
Piperidine derivs: loratidine
fexofenadine
Azelastine
H2 Receptor Antagonists
Cimetidine
Ranitidine
Famotidine
Nizatidine
Serotonin (5-HT)
Serotonin Receptor Antagonists
Cyproheptadine
Ketanserin
Ondansetron
Ergot Alkaloids
Ergotamine
Methysergide
Triptans
Sumatriptan
Rizatriptan
Naratriptan
Zolmitriptan
Ergonovine
Bromocriptine

Dyshemoglobinemias
Carbon monoxide
O2
Hyperbaric O2
Cyanide
Hydroxocobalamin
Hyperbaric O2
Methemoglobin
Methylene blue - tetramethyl thionine
chloride
n-acetylcysteine
Exchange transfusion
Hyperbaric O2
Sulfhemoglobinemia
Supportive only

Autonomics
Cholinergic Receptor-Activating Drugs
Direct-Acting
Bethanechol
Muscarine
Nicotine
Pilocarpine
Cevimeline
Varenicline
Indirect-Acting
Neostigmine
Tacrine
Pyridostigmine
Donepezil
Physostigmine
Edrophonium
Echothiophate
Soman
Cholinergic Receptor-Inhibiting Drugs
Antimuscarinic
Dicyclomine
Tropicamide
Tolterodine
Ipratropium
Tiotropium
Benztropine
Scopolamine
Atropine
Ganglionic Blockers
Hexamethonium
Mecamylamine
NMJ Blockers
Succinylcholine
Tubocurarine
Mivacurium
Botulinum Toxin A
Adrenergic Indirect Agents
Tyramine
Amphetamine
Adrenergic Mixed Agents
Ephedrine
Hydroxyamphetamine
1 agonists
Phenylephrine
Ergotamine
Ergonovine
Bromocriptine
Methysergide
2 agonists
Clonidine
-methyldopa
1 agonists
Dobutamine
2 agonists
Albuterol
Terbutaline
1+2 agonists
Isoproterenol
D1 agonists
Fenoldopam
Mixed agonists
NE (1, 1, (2))
Epi (1, 1, 2, (2))
1 blocker
Prazosin
2 blocker
Yohimbine
blocker - nonselective
Phentolamine
Phenoxybenzamine
1st gen: nonselective blocker
Propranolol
2nd gen: 1 selective
Metoprolol
Atenolol
3rd gen-A: nonselective w/ additional
Carvedilol
Labetalol
3rd gen-B: 1 selective w/ additional
Betaxolol
Neuron Blocking Drugs
-methyltyrosine
Reserpine
Guanethidine

Lipids
Niacin
Fibrates
Clofibrate
Gemfibrozil
Fenofibrate
Ciprofibrate
Benzafibrate

Anticoagulants
Indirect Thrombin Inhibitors
Unfractionated heparin (UFH)
Low-molecular-weight heparin (LMWH)
Dalteparin
Enoxaparin
Tinzaparin
Fondaparinoux
Idraparinoux
Direct Thrombin Inhibitors
Hirudin
Lepirudin
Bivalirudin
Argatroban
Oral Anticoagulants
Warfarin
Activated Protein C
Fibrinolytics Drugs
Streptokinase
Urokinase
Tissue Plasminogen Activator
Reteplase
Tenecteplase
Antiplatelet
Aspirin
Dipyridamole
Clopidogrel
GPIIb-IIIa Antagonists
Abciximab
Eptifibatide
Tirofiban

Cancer
Alkylating agents
Nitrogen mustards
Mechlorethamine
Cyclophosphamide
Ifosfamide
Nitrosoureas
Carmustine
Lomustine
Streptozocin
Triazenes
Dacarbazine
Temozolomide
Platinum Analogs
Cisplatin
Carboplatin
Oxaliplatin
Antimetabolites
Folic Acid
Methotrexate
Pemetrexed
Pyrimidine Analog
5-Fluorouracil
Cytarabine
Gemcitabine
Purine Analog
6-Mercaptopurine
DNA intercalating agents
Dactinomycin
Anthracyclines
Daunorubicin
Doxorubicin
Epirubicin
Idarubicin
Bleomycin
Microtubule inhibitors
Vinca Alkaloids
Vinblastine
Vincristine
Taxanes
Paclitaxel
Docetaxel
Topoisomerase inhibitors
Epipodophyllotoxins
Etoposide
Teniposide
Camptothecin Analogs
Irinotecan
Topotecan
Hormones & their antagonists
Glucocorticoids
Prednisone
Dexamethasone
SERMs
Tamoxifen
Fulvestrant
Estradiol
Raloxifene
Aromatase Inhibitors
Aminoglutethamide
Anastrozole
Androgen deprivation
Leuprolide
Goserelin
Flutamide
Bicalutamide
Misc
Hydroxyurea
Retinoids
Arsenic Trioxide
Thalidomide
Interferons
Tyrosine Kinase Inhibitors
Imatinib
Gefitinib
Erlotinib
Monoclonal Antibodies
Rituximab
Trastuzumab
Cetuximab

Bronchodilators: inhaled 2-agonists


Albuterol
Terbutaline
Salmeterol
Methylxanthines
Theophylline
Anticholinergics
Ipratropium
Inhaled corticosteroids
Oral corticosteroids
Cromolyn Na
Leukotriene modifiers
Zafirlukost
Zileuton

Arthritis
NSAIDs
Indomethacin
COX-2 Inhibitors
DMARD
Glucocorticoids
Gold salts
Antimalarial drugs
Chloroquine
Hydroxychloroquine
Sulfasalazine
Immunosuppressives
Methotrexate
Leflunomide
Biological Response Modifiers
Etanercept
Infliximab
Adalimumab
Anakinra
Abatacept
Tocilizumab

Gout
Acute Gouty Arthritis:
Colchicine
NSAIDs
Indomethacin
Naproxen
Sulindac
Celecoxib
Corticosteroids
Chronic Tophaceous Gout:
Uricosuric Acids
Probenecid
Sulfinpyrazone
Allopurinol

Bile Acid Sequestrants (Resins)


Cholestyramine
Colestipol
Colesevelam
HMG-CoA Reductase Inhibitors (Statins)
Metastatin
Lovastatin
Simvastatin
Pravastatin
Fluvastatin
Atorvastatin
Rosuvastatin

Desmopressin
Aquaretics
Lithium
Fluoride
Demeclocycline
Saluretics
Loop Diuretics
Furosemide
Bumetanide
Torsemide
Ethacrynic acid
(dichlorophenoxyacetic acid)
Thiazide Diuretics
Chlorothiazide
Hydrochlorothiazide
Thiazide-like
Chlorthalidone
Quinethazone
Metolazone
Indapamide
Potassium-sparing diuretics
Spironolactone
Triamterene
Amiloride
Osmotic Diuretics
Mannitol
Excess glucose, urea
Isosorbide
Carbonic Anhydrase Inhibitors
Acetazolamide
Methazolamide
Dichlorphenamide
Aminophylline (theophylline)

Derm
Hydrocortisone
UV light
Methotrexate
Infliximab
Retinoids
1st gen:
Retinol
Tretinoin
Isotretinoin
2nd gen:
Etretinate
Acitretin
3rd gen:
Arotinoids (tazarotene)
Soriatane

ORAL
Oral Insulin Secretagogues
Sulfonylureas
Glyburide
Glipizide
Glimepiride
Glinides
Repaglinide
Nateglinide
Biguanides
Metformin
Thiazolidinediones (TZDs)
Rosiglitazone
Pioglitazone

Ezetimibe

HTN
Diuretics
Thiazides
Loops
K+ Sparing
Sympathetic
CNS Drugs
Methyldopa
Clonidine
Ganglion blocking drugs
Adrenergic blocking
Guanethidine
Reserpine
Blockers
Blockers

Alpha Glucosidase Inhibitors


Acarbose
Miglitol
INSULIN
Short Acting
Lispro
Aspart
Glulisine
Regular Insulin
Intermediate Acting
NPH
NPL
NPA
Determir
Long Acting
Glargine

Malaria
Vasodilators
Direct
Hydralazine
Na Nitroprusside
Minoxidil
Ca+ Channel Blockers
Dihydropyridines
Amlodipine
Nifedipine
Felodipine
Isradipine
Nondihydropyridines
Verapamil
Diltiazem
Angiotensin
ACE-Inhibitors
Captopril
Enalapril
Lisinopril
Ramipril
Quinapril
Fosinopril
ARBs
Losartan
Irbesartan
Valsartan
Candesartan
Olmesartan
Telmisartan

Antiarrhythmics
Class I: Na+ channel blockers
Class IA: Quinidine
Class IB: Lidocaine
Class IC: Flecainide

Class II: blockers


Estmol
Propanolol
Class III: K+ channel blockers
Amiodaron
Sotalol

Quinoline Derivatives
Quinine/Quinidine
Chloroquine
Mefloquine
Primaquine
Artemisinin Compounds
Artemether
Artesunate
Antifolates
Chloroguanide (w/ Atovaquone)
Pyrimethamine
Sulfonamides
Sulfones
Antibiotics

Steroids
Hypoadrenalism:
Glucocorticoids
Short-acting
Hydrocortisone
Cortisone
Intermediate-acting
Prednisone
Prednisolone
Methylprednisolone
Triamcinolone
Long-acting
Paramethasone
Betamethasone
Mineralocorticoids
Fludrocortisone
Cushings:
Aminogethimide
Ketoconazole
Mitotane
Liddle's Syndrome:
Amiloride
Triamterene

Parathyroid/Bone

Misc
Adenosine
Mg
Digitalis
Atropine

Angina
Stress Tests
Dobutamine
Adenosine
Dipyridamole
Antiplatelet
Aspirin
Ticlopidine
Clopidogrel
Prasugrel
Dipyridamole
Lipid-Lowering
ACE-Inhibitors
Blockers
Nitrates
Isosorbide dinitrate
Mononitrate

GI
Ulcers:
Neutralize Acid
Antacids
CaCO3
NaHCO3
MgOH
MgCO3
AlOH
Acid Production
Anticholinergic
Atropine
Propantheline
Metantheline bromide
H2 Receptor Blocker
Cimetidine
Ranitidine
Famotidine
Nizatidine
H+/K+ ATPase Inh (PPI)
Omeprazole
Lansoprazole
Rabeprazole
Esomeprazole
Pantoprazole
Mucosal Resistance
Coat Ulcer Crater
Bismuth Salths
Sucralfate
PGE2 Analogs
Misoprostol
Kill H. pylori
Triple Therapy
Quadruple Therapy
Reflux Esophagitis + Gastritis:
Symptoms w/o esophagitis
Alginic acid antacids
Promotility drugs
Cisapride
Metoclopramide
H2 Receptor Blockers
w/ esophagitis
H2 Receptor Blockers
Promotility
PPIs
Vomiting:
Phenothiazines
Prochlorperazine
Promethazine
Benzamide deriv
Trimethobenzamide
Metochlorpramide
THC
5HT3 receptor antagonist
Ondansetron
Granesitron
Dolasetron
Gastroparesis:
Promotility

Class IV: Ca+ channel blockers


Diltiazem
Verapamil

Osteoporosis:
Bisphosphonates
Alendronate
Risedronate
Ibandronate
Zolendronate
SERMs
Tamoxifen
Raloxifene
Calcitonin
Teriparatide
Paget's:
Bisphosphonates
Etidronate
Pamidronate
Zolendronate
Alendronate
Risendronate
Calcitonin

Diarrhea:
GI motility
Anticholinergics
Opioid Agonists
Loperamide
Diphenoxylate
Codeine Sulfate
Colloid
Metamucil
Pectin
Kaopectate
Antibiotics
Constipation:
Irritant/Stimulant:
Castor Oil
Cascara sagrada
Osmotic cathartics
Mg citrate, Mg sulfate
Milk of magnesia
Bulk-forming
Psyllium seed
Metamucil
Lubricant & Softeners
Mineral Oil
Dioctyl Na sulfosuccinate
Inflammatory Bowel Dz:
Acute
Anti-inflammatories
Mesalamine
Sulfasalazine
Olsalazine
Corticosteroids
Antibiotics
Chronic
Immunosuppressives
Azathrioprine
Corticosteroids
Infliximab
Cyclosporine
Irritable Bowel Syndrome:
Bulk forming
Opioids
Loperamide
Anticholinergics
Dicyclomine
hydrochloride
Hyoscyamine sulfate
Antidepressants
5HT3 rec antagonists
Alosetron
5HT4 rec agonists
Tegaserod maleate

Lead/Heavy Metals
CaNa2EDTA
BAL (Dimercaprol)

Reproduction

DMSA/Succimer

Antimicrobials
Cell Wall Synthesis Inhibitors:
Penicillins
Penicillin
Pen G
Pen V
Penicillinase Resistant Penicillins
Oxacillin
Dicloxacillin
Methicillin
Nafcillin
Aminopenicillins
Ampicillin
Amoxicillin
Extended Spectrum Penicillins
Piperacillin
-Lactamase Inhibitors
Unasyn (Ampicillin/Sulbactam)
Zosyn (Piperacillin/Tazobactam)
Augmentin (Amoxicillin/Clavulanate)
Cephalosporins
1st Gen
Cefazolin
Cephalexin
2nd Gen
Cefuroxime
3rd Gen
Ceftazidime
Ceftriaxone
Cefixime
4th Gen
Cefipime
Cyclic Polypeptides
Daptomycin
Carbapenems
Imipenem
Monobactams
Aztreonam
Vancomycin
Fosfomycin
Protein Synthesis Inhibitors:
Aminoglycosides
Gentamicin
Tobramycin
Amikacin
Streptomycin
Neomycin
Kanamycin
Netilmicin
Tetracyclines
Doxycycline
Tigecycline
Oxazolidinones
Linezolid
Clindamycin
Macrolides
Erythromycin
Azithromycin
Clarithromycin
Nucleic Acid Synthesis
Inhibitors:
Fluoroquinolones
Ciprofloxacin
Levofloxacin
Metronidazole
Rifampin
Anti-Herpes
Purine analogs
Acyclovir
Famciclovir
Valacyclovir
Ganciclovir
Pyrimidine analogs
Sorivudine

Ca+ channel blockers

Acute MI
Oxygen
Nitrates

Aspirin
Blockers
Fibrinolytics
Streptokinase
Alteplase
Reteplase
Tenecteplase-tPA

ACE-Inhibitors
Anticoagulants
Heparin

Natural Estrogens
Estradiol
Estrone
Estriol
Anti-Estrogen
Tamoxifen
Clomiphene citrate
Synthetic Estrogens
Steroidal
Ethinyl estradiol
Mestranol
Quinestrol
Nonsteroidal
Diethylstilbestrol
Chlorotrianisene
Methallenestril
Progestins
Natural
Prometrim
Crinone
Synthetic
Medroxyprogesterone
Norethindrone
Norgestrel
Megestrol
Mifepristone

CHF
ACE-Inhibitors

Erectile Dysfunction:
Sildenafil citrate
Vardenafil HCl
Tadalafil

Deferoxamine

Anti-HPV
Imiquimod
Cidofovir
Anti-Influenza A, B, H1N1
Oseltamavir
Zunamavir
Peramivir
Anti-HIV
Nucleoside RT
Inhibitors
Zidovudine
Didanosine
Zalcitabine
Stavudine
Lamivudine
Abacavir
Non-Nucleoside RT
Inhibitors
Nevirapine
Delaviridine
Efavirenz
Etravirine
Protease Inhibitors
Saquinavir
Ritonivir
Indinavir
Nelfinavir
Fusion Inhibitors
Enfuvirtide
Maraviroc
Antimetabolites:
Sulfonamides
Sulfamethoxazole
(SMX)
Sulfones
Dapsone
Trimethoprim
Pyrimethamine

Blockers
Digoxin
Hydralazine

Thyroid
Hyperthyroid
Carbimazole
Methimazole
Propylthiouracil

Nitrates
Hypothyroid
Levothyroxine
Liothyronine
Liotrix

MAOIs
Tranylcypromine
Phenelzine
Amine Reuptake Inhibitors
Tricyclics
Imipramine -> Desipramine
Amitriptyline -> Nortriptyline
SSRIs
Fluoxetine -> Norfluoxetine
Paroxetine
Sertraline
Escitalopram
Citalopram
SNRIs
Duloxetine
Venlafaxine
Atypicals
Tetracyclics & Unicyclics
Bupropion
Mirtazapine
5HT2A antagonists
Nefazodone
Trazodone
Bipolar
Lithium
Anti-convulsants
Carbamazepine
Valproate
Antidepressants
MAOI
Benzos or antipsycho
Olanzapine
Risperidone
Aripiprazole

Antiepilepsies
Valproate
Sodium
Phenytoin
Carbamazepine
Oxcarbamazepine
Lamotrigine
Calcium
Ethosuximide
GABA analogs
Gabapentin
Pregabalin
Glutamate
Felbamate
Topiramate
GABA-A agonists
Phenobarbital
Vigabatrine
Tiagabine
Benzodiazepines
Lorazepam
Diazepam
Midazolam
Levetiracetam

Anxiolytics
Benzodiazepines
Benzos
Diazepam
Chlordiazepoxide
Lorazepam
Flurazepam
Alprazolam
Midazolam
Triazolam
Pseudo-benzos
Zolpidem
Eszopiclone
Benzo antagonist
Flumazenil
Barbiturates
Phenobarbital
Thiopental
Also use
SSRIs
Busiprone

ALS/Parkinson's
ALS drugs
Riluzole
Baclofen
Tizanidine
Parkinson's
DA precursors
Carbidopa
Levodopa
DA receptor antagonists
Ropinirole
Pramipexole
Pergolide
Bromocriptine
MAO-B inhibitors
Selegiline
Rasagiline
COMT inhibitors
Entacapone
Tolcapone
Anticholinergics
Benztropine
Trihexyphenadyl
Rescue Therapy
Apomorphine
Adjuvants
Amantadine
Deep Brain Stim

Neuroleptic
(antipsychotics)
Typicals
Chlorpromazine
Thiordazine
Fluophenazine
Trifluoperazine
Haloperidol
Atypicals
SGAs
Tricyclics
Clozapine
Olanzapine
Quetiapine

Isoniazid (INH)
Pyrazinamide (PZA)

Non-tricyclics
Risperidone
Ziprazidone

Streptomycin
Ethambutol
Bactrim (TMP/SMX)
Pyrimethamine/Dapsone

Cell Membrane Function Inhibitors:


Polyenes
Nystatin
Amphotericin B

Tx neuroleptic malignant syndrome


Dantrolene
Bromocryptine
Amantadine
Tx hyperprolactinemia
Bromocryptine
Pergolide

Alzheimer's

Polymyxins
Polymyxin B
Colistin

Anti-Cholinesterases
Tacrine
Donepezil
Rivastigmine
Galantamine

Echinocandins
Capsofungin

Glutaminergic
Memantine

Azoles
Imidazoles
Clotrimazole
Miconazole
Ketoconazole

Other
& secretase inhibitors
A vaccine
NSAIDs
Vit E & C
Ginko
Selegiline (MAOI)
NGFs
B6, B12, Folate
Estrogen replacement
Clioquinol
Behavioral
Antidepressants
Antipsychotics
Sedatives

Triazoles
Fluconazole
Itriconazole
Voriconazole

ARBs
Diuretics

Antidepressants

Foscarnet

Prussian Blue

Analgesia: morphine

Diuretics

Incretin Hormones
Glucagon-like peptide 1
GLP-1 Receptor Antagonists
Exenatide
DPP-4 Inhibitors
Sitagliptin
Saxagliptin
Amylin Hormone
Pramlitide

Asthma
Anticoagulants

Diabetes

Allyamines
Terbinafine
Naftifine
Tolnafate

Multiple Sclerosis
Acute MS Attack
Corticosteroids
Methylprednisolone
Oral Prednisone
1st line for CIS & RR-MS
Avonex
Rebif
Betaseron
Glatiramer acetate
2nd line for RR-MS
Natalizumab
Mitoxantrone
1 Progressive MS
Immunosuppressants
Pulse Steroids
IVIG
2 Progressive MS
Mitoxantrone
Immunosuppressants
Azathioprine
MTX
Cyclophosphamide

Narcotics
Morphine
Codeine
Tramadol
Fentanyl
Methadone
Oxycodone
Meperidine
Propoxyphene
Antagonists
Naloxone
Naltrexone

Headache
Acute specific
Ergotamine
Dihydroergotamine
Triptans- many
Acute non-specific
Analgesics
Antiemetics
NSAIDs
Steroids
Anxiolytics
Opioids
Preventative
Antidepressants
Amitriptyline
Anti-HTN
Propranolol
Timolol
Nadolol
Atenolol
Verapamil
Antiepileptics
Divalproex Na
Topiramate

Ophthalmology
Glaucoma
1st line
Timolol
Latanoprost
Brimondine
Dorzolamide
Prostaglandin analogs
Latanoprost
Bimatroprost
Travoprost
Unoprostone
Carbonic Anhydrase Inhibitors
Oral
Acetazolamide
Ethoxzolamide
Metahazolamide
Topical
Dorzolamide
Brinzolamide
Ca channel blocker
Nifedipine
Parasympathetic
Muscurinic
Agonist
ACh (Miochol)
Carbachol
Methacoline
Pilocarpine
Antagonist
Atropine
Scopolamine
Homatropine
Cyclopentolate
Tropicamide
Nicotinic
Agonist
Endrophonium
Sympathetic
Direct Agonist
Phenylephrine
L-epinephrine
Dipivalyl
Brimondine
Indirect Agonist
Cocaine
Hydroxyamphetamine
Antagonist
Timolol
Betaxolol
Levobunolol
Dapiprazole

Anesthetics
General
Inhalational
Vapors
Halothane
Enflurane
Isoflurane
Sevoflurane
Desflurane
Gases
Nitrous Oxide
Xenon
Intravenous
Barbiturates
Thiopental
Propofol
Etomidate
Ketamine
Benzodiazepines
Midazolam
Diazepam
Lorazepam
Antagonist
Flumazenil
Opioids
Morphine
Meperidine fentanyl
Remifentanil
Skeletal Muscle Relaxants
Non-depolarizing-competitive
Long acting
Doxacurium
Pancuronium
Intermediate
Atracurium
Cisatracurium
Vecuronium
Rocuronium
Short acting
Mivacurium
Reversal
Neostigmine
Sugammadex
Depolarizing
Succinylcholine
Local
Amides
Lidocaine
Etidocaine
Mepivacaine
Bupivacaine
Prilocaine
Articaine
Dibucaine
Ropivacaine
Esters
Procaine
Propoxycaine
Tetracaine
Cocaine
Benzocaine
Dyclonine

Non-Med Drugs
Alcohol
Stimulants
Amphetamines
Cocaine
Club Drugs
Nicotine
Hallucinogens
LSD (lysergic acid diethylamide)
Mescaline (peyote)
Psilocybin (psilocin)
Substituted amphetamines
MDMA
DOM
PCP
Ketamine
Marijuana
DMT (dimethyltryptamine)
Disulfuram
Fomepizol

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