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Antimicrobials

ANTIBACTERIALS
Beta Lactams and Other Cell Wall Inhibitors
Penicillins
Penicillin G (benzyl pcn)
Benzathine pcn G
Penicillin V (pnenoxymethy pcn)
(broader spectrum)
Ampicillin
(w/ or w/o Sulbactam)
Amoxicillin
(w/ or w/o Clauvulanic Acid)
(anti-Pseudomoal)
Carbenicillin
Ticarcillin
(w/ or w/o Clavulanic acid)
Piperacillin
Azlocillin
Mezlocillin
(penicillinase-resistant: anti-Staph)
Methicillin
Oxacillin
Dicloxacillin
Cloxacillin
Naficillin
-lactamase inhibitors
Clavulanic Acid
Sulbactam
Tazobactam
Cephalosporins
(1st gen)
Cefazolin
Cefadroxil
Cephalexin
Cephalothin
Cephapirin
Cephadrine
(2nd gen)
Cefaclor
Cefamandole
Cefonicid
Ceforanide
Cefotetan
Cefoxitin
Cefuroxime
Cefuroxin axetil
(3rd gen)
Cefixime
Cefoperazone
Cefotaxime
Ceftazidime
Ceftizoxime
Ceftriaxone
Moxalactam
Monobactams
Aztreonam
Carbapenems
Imipenem
(w/ cilastatin)
Other Cell wall Inhib
Vancomycin
Bacitracin

Cycloserine
Membrane Active
Polymixin B
Colistimethate
*Polymixin E (colistin)
Protein Synthesis Inhibitors
Aminoglycosides
Streptomycin
Gentamicin
Tobramycin
Neomycin
Kanamycin
Amikacin
Netilmicin
Tetracyclines
Tetracycline
Chlorotetracycline
Demeclocycline
Doxycycline
Minocycline
Oxytetracycline
Spectinomycin
Macrolides and Lincosamides
Erythromycin
Lincomycin
Clindamycin
Chloramphenicol
Folate Antagonists
Sulfonamides
Sulfisoxazole
Sulfadiazine
Sulfamethoxazole
Sulfasalazine
(Salicylazosulfapyridine)
Sulfacetamide
Silver Sulfadiazine
Mafenide
Sulfadoxine
Trimethoprim-Sulfamethoxazole
(Bactrim & Septra)
Sulfacytine
Nucleic Acid Inhibitors (DNA Gyrase Inhibtors)
Quinolones
Nalidixic Acid
Ciprofloxacin
Norfloxacin
*Ofloxacin
*Temafloxacin
Nitrofurantoin
Rifampin
ANTIMYCOBACTERIAL
Rx TB
First line
Isoniazid (INH)
Rifampin
Ethambutol
Streptomycin
Pyrazinamide
Second line
Ethionamide
Para-Aminosalicylic acid

Cycloserine
Kanamycin, Amikacin
Capreomycin
*Viomycin
Rx Leprosy
Dapsone
Rifampin
Clofazimine
Minocycline
Clarithromycin
Fluoroquinones
*Acedapsone
*Amithiozone
ANTIFUNGAL
Polyene ABX
Amphotericin B
Nystatin (Mycostatin)
Imidazoles
Miconazole
Clotrimazole
Ketoconazole
Itraconazole
Misc.
Flucytosine
Griseofulvin
Triazoles: Fluconazole
*Tolnafate
ANTIPROTOZOAL AGENTS
Rx Malaria
Chloroquine
Primaquine
Quinine
Antifolates
Pyrimethamine
*Proguanil
*Sulfadoxine
*Dapsone
Tetracycline
Doxaclycline
Mefloquine
Fansidar
Rx Amebiasis
Metronidazole (Flagyl)
Diloxanide furoate
Paromomycin
Iodoquinol (diiodohydroxyquin)
Chloroquine
Rx Leishmaniasis
Sodium Stibogluconate
Pentamidine
Rx Trypanosomiasis
Melarsoprol
Nifurtimox
Pentamidine
Suramin
Rx Giardiasis
Metronidazole
Quinacrine
Rx Trichomoniasis
Metronidazole
Rx Toxoplasmosis
Pyrimethamine + Sulfonamide

Clindamycin + Pyrimethamine
Pyrimethamine alone (high dose)
Rx Pneumocystis Carinii
Trimethoprim-sulfamethoxazole
Pentamididne
Dapsone
ANTIHELMINTHIC
Nematodes (Roundworms)
Mebendazole
Thiabendazole
Pyrantel Pamoate
Diethylcarbamazine
*Levamisole
*Albendazole
*Ivermectin
Trematodes (Flukes)
Praziquantel
Oxamniquine
*Metrifonate
*Bithionol
*Dehydroemetine
Cestodes (Tapeworms)
Niclosamide
Praziquantel
ANTIVIRAL
Rx Herpes
Acyclovir
Famcyclovir
Ganciclovir
Vidarabine (ARA-A)
Idoxuridine
Foscarnet
Rx Respiratory Viral
Amantidine
Ribavirin
Rimantidine
Rx HIV
Azidothymidine (AZT)
DDI
DDC
Endogenous Factor
Interferon
ANTINEOPLASTIC AGENTS
Alkylating Agents
Nitrogen Mustards [bis(chloroethyl)amines]
Mechlorethamine
Cyclophosphamide
Melphalan
Chorambucil
Alkyl Sulfonate deriv
Busulfan
Nitrosureas
Carmustine (BCNU)
Lomustine (CCNU)
Semustine
Streptozocin
Triazene deriv
Dacarbazine (DTIC)
Ethylemine deriv
Triethylenethiophoramide
Aziridines
Thitepa

Triethyleenemelamine
Platinum Complexes
Cisplatin
Carboplatin
Hydrazine
Procarbazine
*Dacarbazine
Antimetabolites
Methotrexate(MTX)
5-Fluorouracil (5-FU)
Cytarabine
(Cytosine arabinoside, Ara-C)
6-Mercaptopurine (6-MP)
6-Thioguanine (6-TG)
related purine analogs
Alzathioprine
Allopurinol
Plant Alkaloids
Vinca Alkaloids
Vincristine
Vinblastine
Podophyllotoxins
Etoposide (VP-16)
Teniposide
Paclitaxel (taxol)
Antibiotics
Dactinomycin
Anthracyclin ABX
Daunorubicin
Doxorubicin (adriamycin)
Mitoxantrone
Bleomycin
Plicamycin (mithramycin)
Mitomycin C
Hormonal Rx
Prednisone
Progestins
hydroxyprogesterone
medroxyprogesterone
megesterol
Androgens
fluoxymesterone
testosterone
Estrogens
ethinyl estradiol
DES
Tamoxifen
Flutamide
Aminoglutethimide
Leuprolide
*Goserelin
*Nafarelin
Misc Agents
L-Asparaginase
Hydroxyurea
Mitotane

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