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U.S.

Department of Justice
Drug Enforcement Administration
Diversion Control Division
Drug & Chemical Evaluation Section

Lists of:

Scheduling Actions
Controlled Substances
Regulated Chemicals

July 2023
Foreword
The first three sections of this booklet list the names of the substances which are described in the Code of Federal
Regulations (CFR) as well as some of those which generate frequent inquiries. The substances are first arranged
alphabetically, then by Drug Enforcement Administration (DEA) drug code number, and finally by Controlled Substances
Act (21 U.S.C. §801 et seq.) (CSA) schedule.
These lists describe the basic or parent chemical and do not describe the salts, isomers, salts of isomers, esters,
ethers, and derivatives which may be controlled substances. These are not comprehensive lists so please note that a
substance need not be listed as a controlled substance to be treated as a scheduled substance for criminal prosecution.
The “Other Names” column, provides some examples of alternate names for certain compounds, and in some
instances provides examples of “positional isomers”. If outside parties want to ensure that a compound is not
considered a scheduled substance or listed chemical, they should write the DEA, Drug and Chemical Evaluation
Section (DRE), Diversion Control Division, 8701 Morrissette Drive, Springfield, Virginia 22152, for an official
determination.
A substance (not included on these lists) may also be regulated as a controlled substance analogue. A controlled
substance analogue is a substance which is intended for human consumption, is structurally substantially similar to a schedule
I or schedule II substance, is pharmacologically substantially similar to a schedule I or schedule II substance, or is
represented as being similar to a schedule I or schedule II substance and is not an approved medication in the United States.
See 21 U.S.C. § 802(32)(A) for the definition of a controlled substance analogue and 21 U.S.C. § 813 for the schedule.
The next two sections of this booklet list the Federal Register notices through which the DEA has directed substances
to be added, deleted or transferred between schedules of the CSA. The scheduling changes are listed first in alphabetical
order by substance and then in chronological order by effective date. With the exception of anabolic steroids, section 812 of
the CSA lists only those substances which were controlled in 1970 when the law was enacted. Since then, over 200
substances have been added, removed, or transferred from one schedule to another. The current official list of controlled
substances can be found in section 1308 of the most recent issue of Title 21 Code of Federal Regulations Part 1300 to end (21
CFR § 1308) and the final rules which have been published in the Federal Register subsequent to the issuance of the CFR.
The CFR and the Federal Register are available on the U.S. Government Printing Office web site at
https://www.gpo.gov/fdsys/. This information is accessible, also, on the Diversion Control Division’s website at
https://www.deadiversion.usdoj.gov/.
The last section of this booklet identifies the “List I” and “List II” chemicals. Certain commercial transactions
involving these chemicals are regulated by the CSA. See 21 CFR §§ 1309, 1310 and 1313 for details.
These lists are intended as general references and are not comprehensive listings of all controlled substances and
regulated chemicals.
Drug and Chemical Evaluation Section
Diversion Control Division
Drug Enforcement Administration

Telephone: 202-307-7183 • FAX: 202-353-1263

July 2023
Abbreviations
2C-B = 4-Bromo-2,5-dimethoxyphenethylamine
2C-T-7 = 2,5-Dimethoxy-4(n)-propylthiophenethylamine
BZP = N-Benzylpiperazine
DMT = Dimethyltryptamine
DOM = 4-Methyl-2,5-dimethoxyamphetamine
GBL = Gamma butyrolactone
GHB = Gamma hydroxybutyric acid, gamma hydroxybutyrate,
4-hydroxybutanoic acid, sodium oxybate
LAAM = Levo-alphacetylmethadol
LSD = Lysergic acid diethylamide, lysergide
MDA = 3,4-Methylenedioxyamphetamine
MDE = 3,4-Methylenedioxy-N-ethylamphetamine
MDMA = 3,4-Methylenedioxymethamphetamine
MPPP = 1-Methyl-4-phenyl-4-propionoxypiperidine
P2P = Phenyl-2-propanone, phenylacetone
PCC = 1-Piperidinocyclohexanecarbonitrile
PCE = N-Ethyl-1-phenylcyclohexylamine
PCH = 1-Phenylcyclohexylamine
PCP = 1-(1-Phenylcyclohexyl)piperidine, phencyclidine
PEPAP = 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine
PHP = 1-(1-Phenylcyclohexyl)pyrrolidine
SPA = (-)-1-Dimethylamino-1,2-diphenylethane
TCP = 1-[1-(2-Thienyl)cyclohexyl]piperidine
TCPy = 1-[1-(2-Thienyl)cyclohexyl]pyrrolidine
THC = Tetrahydrocannabinols
THG = Tetrahydrogestrinone
Scheduling Actions
Alphabetical Order
Scheduling Actions
- Alphabetical Order -
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE

(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 04-16-19 84 FR 15505 4/16/2019 I


TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144) *
(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 03-31-21 86 FR 16669 4/16/2021 I
TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144) **
(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 04-07-22 87 FR 20318 4/7/2022 I
TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144)
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144) *
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-15-15 80 FR 27854 5/15/2015 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144) **
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-11-16 81 FR 29142 5/11/2016 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1- 01-30-15 80 FR 5042 1/30/2015 I
YL)METHANONE (THJ-2201) *
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1- 10-16-17 82 FR 47971 10/16/2017 I
YL)METHANONE (THJ-2201)
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-UR-
144, XLR11) *
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-15-15 80 FR 27854 5/5/2015 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-UR-
144, XLR11) **
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-11-16 81 FR 29142 5/11/2016 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-UR-
144, XLR11)
1-(1-(1-(4-BROMOPHENYL)ETHYL)PIPERIDIN-4-YL)-1,3- 03-01-21 86 FR 11862 3/1/2021 I
DIHYDRO-2H-BENZO[D]IMIDAZOL-2-ONE (BRORPHINE) *
1-(1-(1-(4-BROMOPHENYL)ETHYL)PIPERIDIN-4-YL)-1,3- 03-06-23 88 FR 13692 4/5/2023 I
DIHYDRO-2H-BENZO[D]IMIDAZOL-2-ONE (BRORPHINE)
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 08-31-18 83 FR 44474 8/31/2018 I
ONE (N-ETHYLPENTYLONE, EPHYLONE) *
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 08-27-20 85 FR 52915 8/31/2020 I
ONE (N-ETHYLPENTYLONE, EPHYLONE) **
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 06-14-21 86 FR 31427 6/14/2021 I
ONE (N-ETHYLPENTYLONE, EPHYLONE)
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-10-18 83 FR 31877 7/10/2018 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA) *
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-13-20 85 FR 42296 7/10/2020 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA) **
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 06-10-21 86 FR 30775 6/10/2021 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA)

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 1 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 04-16-19 84 FR 15505 4/16/2019 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25) *
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 03-31-21 86 FR 16669 4/16/2021 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25) **
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 04-07-22 87 FR 20318 4/7/2022 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25)
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-10-18 83 FR 31877 7/10/2018 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA) *
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-13-20 85 FR 42296 7/10/2020 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA) **
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 06-10-21 86 FR 30775 6/10/2021 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA)
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
3,17-dione)
2-(2-(4-BUTOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-YL)- 04-12-22 87 FR 21556 4/12/2022 I
N,N-DIETHYLETHAN-1-AMINE (BUTONITAZENE) *
2-(2-(4-ETHOXYBENZYL)-1H-BENZIMIDAZOL-1-YL)-N,N- 04-12-22 87 FR 21556 4/12/2022 I
DIETHYLETHAN-1-AMINE (ETODESNITAZENE; ETAZENE) *
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I
METHOXYBENZYL)ETHANAMINE (25B-NBOMe) *
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I
METHOXYBENZYL)ETHANAMINE (25C-NBOMe) *
2-(4-ETHOXYBENZYL)-5-NITRO-1-(2-(PYRROLIDIN-1- 04-12-22 87 FR 21556 4/12/2022 I
YL)ETHYL)-1H-BENZIMIDAZOLE (N-PYRROLIDINO
ETONITAZENE) *
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) 11-15-13 78 FR 68716 11/15/2013 I
ETHANAMINE (25I-NBOMe) *
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-20-02 67 FR 59163 9/20/2002 I
T-7) *
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-10-03 68 FR 53289 9/20/2003 I
T-7) **
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
T-7)
2,5-DIMETHOXY-4-CHLOROAMPHETAMINE (DOC) 04-11-22 04-11-22 87 FR 21069 I
2,5-DIMETHOXY-4-CHLOROAMPHETAMINE (DOC) 04-11-22 08-29-22 87 FR 52712 I Withdrew
2022
proposed
rule
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
2,5-DIMETHOXY-4-IODOAMPHETAMINE (DOI) 04-11-22 04-11-22 87 FR 21069 I
2,5-DIMETHOXY-4-IODOAMPHETAMINE (DOI) 04-11-22 08-29-22 87 FR 52712 I Withdrew
2022
proposed
rule
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
2'-FLUORO ORTHO-FLUOROFENTANYL 04-27-21 86 FR 22113 4/27/2021 I

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 2 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
3,4-DICHLORO-N-[(1- 04-14-16 81 FR 22023 5/15/2016 I
DIMETHYLAMINO)CYCLOHEXYLMETHYL]BENZAMIDE)
(AH-7921)
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N- 11-14-16 81 FR 79389 11/14/2016 I
METHYLBENZAMIDE (U-47700) *
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N- 04-20-18 83 FR 17486 4/20/2018 I
METHYLBENZAMIDE (U-47700)
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-15-87 52 FR 38225 10/15/1987 I
MDEA) *
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-13-88 53 FR 40061 10/13/1988 I
MDEA) **
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
MDEA)
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I
(METHYLONE) *
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 04-12-13 78 FR 21818 4/12/2013 I
(METHYLONE)
3,4-METHYLENEDIOXYPYROVALERONE (MDPV) * 10-21-11 76 FR 65371 10/21/2011 I
3-ALPHA-HYDROXY-3-BETA-METHYL-5-ALPHA-PREGNAN-20- 06-01-22 87 FR 32991 6/1/2022 V
ONE (GANAXOLONE)
3-FLUORO-N-METHYLCATHINONE (3-FMC) * 03-07-14 79 FR 12938 3/7/2014 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) ** 03-04-16 81 FR 11429 3/4/2016 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
3-METHYLFENTANYL * 03-25-85 50 FR 11690 4/25/1985 I
3-METHYLFENTANYL ** 04-24-86 51 FR 15474 4/25/1986 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I
3-METHYLTHIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
3-METHYLTHIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
4,4′-DIMETHYLAMINOREX (4,4′-DMAR; 4,5-DIHYDRO-4- 04-07-20 08-12-21 86 FR 44270 9/13/2021 I
METHYL-5-(4-METHYLPHENYL)-2-OXAZOLAMINE)
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) * 07-18-19 84 FR 34291 7/18/2019 I
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) ** 07-18-21 86 FR 37672 7/18/2021 I
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) 06-01-22 87 FR 32996 6/1/2022 I
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE * 01-06-94 59 FR 00671 1/6/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE ** 12-21-94 59 FR 65710 1/6/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 07-18-19 84 FR 34291 7/18/2019 I
CHLORO-A-PVP) *
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 07-18-21 86 FR 37672 7/18/2021 I
CHLORO-A-PVP) **
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 06-01-22 87 FR 32996 6/1/2022 I
CHLORO-A-PVP)
4-FLUORO-N-METHYLCATHINONE (4-FMC) * 03-07-14 79 FR 12938 3/7/2014 I
4-FLUORO-N-METHYLCATHINONE (4-FMC) ** 03-04-16 81 FR 11429 3/4/2016 I

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 3 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
4-FLUORO-N-METHYLCATHINONE (4-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE (4-OH-DiPT) 01-14-22 01-14-22 87 FR 2376 I
4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE (4-OH-DiPT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4'-METHYL ACETYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4-MEAP) 07-18-19 84 FR 34291 7/18/2019 I
*
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4-MEAP) 07-18-21 86 FR 37672 7/18/2021 I
**
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4-MEAP) 06-01-22 87 FR 32996 6/1/2022 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-07-14 79 FR 12938 3/7/2014 I
MePPP) *
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 81 FR 11429 3/4/2016 I
MePPP) **
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
MePPP)
4-METHYLAMINOREX * 10-15-87 52 FR 38225 10/15/1987 I
4-METHYLAMINOREX ** 10-13-88 53 FR 40061 10/13/1988 I
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) * 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) ** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE) * 10-21-11 76 FR 65371 10/21/2011 I
5-METHOXY-ALPHA-METHYLTRYPTAMINE (5-MeO-AMT) 01-14-22 01-14-22 87 FR 2376 I
5-METHOXY-ALPHA-METHYLTRYPTAMINE (5-MeO-AMT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
5-METHOXY-N,N-DIETHYLTRYPTAMINE (MeO-DET) 01-14-22 01-14-22 87 FR 2376 I
5-METHOXY-N,N-DIETHYLTRYPTAMINE (MeO-DET) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) ** 04-01-04 69 FR 17034 4/1/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
5-METHOXY-N-METHYL-N-ISOPROPYLTRYPTAMINE (5-MeO- 01-14-22 01-14-22 87 FR 2376 I
MiPT)
5-METHOXY-N-METHYL-N-ISOPROPYLTRYPTAMINE (5-MeO- 01-14-22 07-27-22 87 FR 45076 I Withdrew
MiPT) 2022
proposed
rule
6β-NALTREXOL ((5a,6β)-17-(CYCLOPROPYLMETHYL)-4,5- 01-24-20 85 FR 4215 1/24/2020 II -> 0
EPOXYMORPHINAN-3,6,14-TRIOL)

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 4 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-17-15 80 FR 42381 7/17/2015 I
PHENYLACETAMIDE) *
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 06-07-17 82 FR 26349 6/7/2017 I
PHENYLACETAMIDE)
ACETYL-ALPHA-METHYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
ACETYL-ALPHA-METHYLFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-14-17 82 FR 32453 7/14/2017 I
PHENYLACRYLAMIDE) *
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-29-18 83 FR 61320 11/29/2018 I
PHENYLACRYLAMIDE)
ALFAXALONE (5α-PREGNAN-3α-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II
ALPHA-ETHYLTRYPTAMINE * 03-12-93 58 FR 13533 3/12/1993 I
ALPHA-ETHYLTRYPTAMINE ** 03-07-94 59 FR 10720 3/12/1994 I
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I
ALPHA-METHYLTHIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
ALPHA-METHYLTHIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) * 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) ** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) * 07-18-19 84 FR 34291 7/18/2019 I
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) ** 07-18-21 86 FR 37672 7/18/2021 I
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) 06-01-22 87 FR 32996 6/1/2022 I
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) * 07-18-19 84 FR 34291 7/18/2019 I
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) ** 07-18-21 86 FR 37672 7/18/2021 I
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) 06-01-22 87 FR 32996 6/1/2022 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) * 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) ** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV
AMINEPTINE (7-[(10,11-DIHYDRO-5H- 07-22-22 11-17-22 87 FR 68895 12/19/2022 I
DIBENZO[A,D]CYCLOHEPTEN-5-YL)AMINO]HEPTANOIC
ACID)
AMINOREX * 09-21-92 57 FR 43399 9/21/1992 I
AMINOREX ** 08-24-93 58 FR 44611 9/21/1993 I
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 5 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
APPROVED CANNABIDIOL DRUGS , AS DEFINED IN 21 CFR 09-28-18 83 FR 48953 9/28/2018 V
1308.15(f)
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired
11/29/86
BETA-HYDROXY-3-METHYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXY-3-METHYLFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I Expired
5/29/87
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I
BETA-HYDROXYFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXYFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
BETA-HYDROXYTHIOFENTANYL * 05-12-16 81 FR 29492 5/12/2016 I
BETA-HYDROXYTHIOFENTANYL 05-08-19 84 FR 20023 5/8/2019 I
BETA-METHYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
BETA'-PHENYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
BREXANOLONE (3Α-HYDROXY-5Α-PREGNAN-20-ONE), 06-17-19 84 FR 27938 6/17/2019 IV
ALLOPREGNANOLONE
BRIVARACETAM (BRV; UCB-34714; BRIVIACT) 05-12-16 81 FR 29487 5/12/2016 V
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0
Superseded
10/97
BUTYLONE * 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE ** 03-04-16 81 FR 11429 3/4/2016 I
BUTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
BUTYRYL FENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 6 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
CENOBAMATE [(1R)-1-(2-CHLOROPHENYL)-2-(TETRAZOL-2- 03-10-20 85 FR 13741 3/10/2020 V
YL)ETHYL]CARBAMATE
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
CROTONYL FENTANYL ((E)-N-(1-PHENETHYLPIPERIDIN-4- 10-02-20 85 FR 62215 10/2/2020 I
YL)-N-PHENYLBUT-2-ENAMIDE)
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4- 01-04-18 83 FR 469 1/4/2018 I
YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE) *
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4- 10-25-19 84 FR 57323 10/25/2019 I
YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE)
DARIDOREXANT (QUVIVIQ) 04-07-22 87 FR 20313 4/7/2022 IV
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
en-17-ol, madol)
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification
of CIV
control
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification
of CII
control
DRONABINOL IN ORAL SOLUTION IN DRUG PRODUCT 03-23-17 82 FR 14815 3/23/2017 II
APPROVED FOR MARKETING BY U.S. FOOD AND DRUG
ADMIN.
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 7 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I
ELUXADOLINE 08-11-15 11-12-15 80 FR 69861 12/17/2015 IV
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-16-19 84 FR 15505 4/16/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA) *
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 03-31-21 86 FR 16669 4/16/2021 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA) **
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-07-22 87 FR 20318 4/7/2022 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA)
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II
EUTYLONE (1-(1,3-BENZODIOXOL-5-YL)-2- 04-10-23 88 FR 21101 4/10/2023 I
(ETHYLAMINO)BUTAN-1-ONE)
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
FENFLURAMINE 05-06-97 05-06-97 62 FR 24620 IV -> 0
FENFLURAMINE 05-06-97 05-15-03 68 FR 26247 IV
Withdrew
97
proposed
rule
FENFLURAMINE 07-19-22 12-23-22 87 FR 78857 12/23/2022 IV -> 0
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENTANYL CARBAMATE 05-04-21 86 FR 23602 5/4/2021 I
FENTANYL-RELATED SUBSTANCES, AS DEFINED IN 21 CFR 02-06-18 83 FR 5188 2/6/2018 I
1308.11(h)*
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 11-03-17 82 FR 51154 11/3/2017 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE *
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 10-30-19 84 FR 58045 11/3/2019 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE **
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 03-30-20 85 FR 17494 3/30/2020 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 8 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III
products
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
ISOTONITAZENE (N,N-DIETHYL-2-(2-(4 08-20-20 85 FR 51342 8/20/2020 I
ISOPROPOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-
YL)ETHAN-1-AMINE) *
ISOTONITAZENE (N,N-DIETHYL-2-(2-(4 11-04-21 86 FR 60761 12/6/2021 I
ISOPROPOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-
YL)ETHAN-1-AMINE)
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
LASMIDITAN [2,4,6-TRIFLUORO-N-(6-(1-METHYLPIPERIDINE- 01-31-20 85 FR 5557 1/31/2020 V
4-CARBONYL)PYRIDINE-2-YL-BENZAMIDE]
LEMBOREXANT 04-07-20 85 FR 19387 4/7/2020 IV
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted
RX
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) * 05-31-85 50 FR 23118 7/1/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) ** 06-17-86 51 FR 21911 7/1/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 9 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted
RX
MESOCARB (N-PHENYL-N'-(3-(1-PHENYLPROPAN-2-YL)- 08-11-21 11-22-22 87 FR 71247 12/22/2022 I
1,2,3-OXADIAZOL-3-IUM-5-YL)CARBAMIMIDATE)
METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
METHASTERONE (2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III
ANDROSTAN-17BETA-OL-3-ONE)
METHCATHINONE * 05-01-92 57 FR 18824 5/1/1992 I
METHCATHINONE ** 04-29-93 58 FR 25934 5/1/1993 I
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I
METHIOPROPAMINE (N-METHYL-1-(THIOPHEN-2- 09-02-21 12-09-22 87 FR 75470 1/9/2023 I
YL)PROPANE-2-AMINE
METHOXETAMINE 12-07-21 06-07-22 87 FR 34166 7/6/2022 I
METHOXYACETYL FENTANYL (2-METHOXY-N-(1- 10-26-17 82 FR 49504 10/26/2017 I
PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE) *
METHOXYACETYL FENTANYL (2-METHOXY-N-(1- 10-25-19 84 FR 57323 10/25/2019 I
PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE
(MDMB–FUBINACA) *
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
FUBINACA) **
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
FUBINACA)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA) *
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA) **
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB) *
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB) **
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 04-16-19 84 FR 15505 4/16/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA) *

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 10 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 03-31-21 86 FR 16669 4/16/2021 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA) **
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 04-07-22 87 FR 20318 4/7/2022 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA)
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA) *
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA) **
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA)
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 07-10-18 83 FR 31877 7/10/2018 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA) *
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 07-13-20 85 FR 42296 7/10/2020 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA) **
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 06-10-21 86 FR 30775 6/10/2021 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA)
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
MPPP * 07-10-85 50 FR 28098 8/12/1985 I
MPPP ** 08-11-86 51 FR 28695 8/12/1986 I
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
MT-45 (1-CYCLOHEXYL-4-(1,2- 12-13-17 82 FR 58557 1/12/2018 I
DIPHENYLETHYL)PIPERAZINE))
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-16-13 78 FR 28735 5/16/2013 I
CARBOXAMIDE (APINACA, AKB48) *
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-15-15 80 FR 27854 5/15/2015 I
CARBOXAMIDE (APINACA, AKB48) **
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-11-16 81 FR 29142 5/11/2016 I
CARBOXAMIDE (APINACA, AKB48)
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 04-10-17 82 FR 17119 4/10/2017 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE
(ADB–FUBINACA) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 04-08-19 84 FR 13796 4/8/2019 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE
(ADB–FUBINACA) **
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 01-24-20 85 FR 4211 1/24/2020 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (ADB-
FUBINACA)
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 02-05-16 81 FR 6171 2/5/2016 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 01-30-18 83 FR 4411 1/30/2018 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA) **

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 11 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 01-29-19 84 FR 444 1/29/2019 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA)
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-10-14 79 FR 7577 2/10/2014 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-05-16 81 FR 6175 2/5/2016 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA) **
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 09-06-16 81 FR 61130 9/6/2016 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 02-10-14 79 FR 7577 2/10/2014 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 02-05-16 81 FR 6175 2/5/2016 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA) **
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 09-06-16 81 FR 61130 9/6/2016 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 07-10-18 83 FR 31877 7/10/2018 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 07-13-20 85 FR 42296 7/10/2020 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA) **
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 06-10-21 86 FR 30775 6/10/2021 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1- 01-30-15 80 FR 5042 1/30/2015 I
(CYCLOHEXYLMETHYL)1H-INDAZOLE-3-CARBOXAMIDE (AB-
CHMINACA) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1- 10-16-17 82 FR 47971 10/16/2017 I
(CYCLOHEXYLMETHYL)1H-INDAZOLE-3-CARBOXAMIDE (AB-
CHMINACA)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H- 01-30-15 80 FR 5042 1/30/2015 I
INDAZOLE-3-CARBOXAMIDE (AB-PINACA) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H- 10-16-17 82 FR 47971 10/16/2017 I
INDAZOLE-3-CARBOXAMIDE (AB-PINACA)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLBUTANAMIDE 04-20-18 83 FR 17486 4/20/2018 I
(BUTYRYL FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 02-01-18 83 FR 4580 2/1/2018 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL) *
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 01-30-20 85 FR 5321 2/1/2020 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-25-20 85 FR 75231 11/25/2020 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2- 11-29-16 81 FR 85873 11/29/2016 I
CARBOXAMIDE (FURANYL FENTANYL) *
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2- 11-29-18 83 FR 61320 11/29/2018 I
CARBOXAMIDE (FURANYL FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 02-01-18 83 FR 4580 2/1/2018 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL) *

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 12 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 01-30-20 85 FR 5321 2/1/2020 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-25-20 85 FR 75231 11/25/2020 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 02-01-18 83 FR 4580 2/1/2018 I
(VALERYL FENTANYL) *
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 01-30-20 85 FR 5321 2/1/2020 I
(VALERYL FENTANYL) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 11-25-20 85 FR 75231 11/25/2020 I
(VALERYL FENTANYL)
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1- 02-01-18 83 FR 4580 2/1/2018 I
PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL) *
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1- 11-29-18 83 FR 61320 11/29/2018 I
PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL)
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-25-20 85 FR 75231 11/25/2020 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)*
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 01-30-20 85 FR 5321 2/1/2020 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)**
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL) *
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 10-25-19 84 FR 57323 10/25/2019 I
YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL)
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 05-03-17 82 FR 20544 5/3/2017 I
YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL) *
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-29-18 83 FR 61320 11/29/2018 I
YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL)
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL) *
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 01-30-20 85 FR 5321 2/1/2020 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL) **
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-25-20 85 FR 75231 11/25/2020 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL)
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 04-16-19 84 FR 15505 4/16/2019 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA) *
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 03-31-21 86 FR 16669 4/16/2021 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA) **
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 04-07-22 87 FR 20318 4/7/2022 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA)
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 04-10-17 82 FR 17119 4/10/2017 I
3-CARBOXAMIDE (5F–APINACA, 5F–AKB48) *
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 04-08-19 84 FR 13796 4/8/2019 I
3-CARBOXAMIDE (5F-APINACA, 5F-AKB48) **
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 01-24-20 85 FR 4211 1/24/2020 I
3-CARBOXAMIDE (5F-APINACA, 5F-AKB48)
N,N-DIETHYL-2-(2-(4- METHOXYBENZYL)-5-NITRO-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (METONITAZENE) *

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 13 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N,N-DIETHYL-2-(2-(4-FLUOROBENZYL)-5-NITRO-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (FLUNITAZENE) *
N,N-DIETHYL-2-(2-(4-METHOXYBENZYL)-1H-BENZIMIDAZOL- 04-12-22 87 FR 21556 4/12/2022 I
1-YL)ETHAN-1-AMINE (METODESNITAZENE) *
N,N-DIETHYL-2-(5-NITRO-2-(4-PROPOXYBENZYL)-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (PROTONITAZENE) *
N,N-DIISOPROPYLTRYPTAMINE (DiPT) 01-14-22 01-14-22 87 FR 2376 I
N,N-DIISOPROPYLTRYPTAMINE (DiPT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
N,N-DIMETHYLAMPHETAMINE * 08-03-88 53 FR 29232 8/3/1988 I
N,N-DIMETHYLAMPHETAMINE ** 08-02-89 54 FR 31815 8/2/1989 I
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 07-10-18 83 FR 31877 7/10/2018 I
CARBOXYLATE (NM2201; CBL2201) *
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 07-13-20 85 FR 42296 7/10/2020 I
CARBOXYLATE (NM2201; CBL2201) **
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 06-10-21 86 FR 30775 6/10/2021 I
CARBOXYLATE (NM2201; CBL2201)
NAPHYRONE * 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE ** 03-04-16 81 FR 11429 3/4/2016 I
NAPHYRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
N-ETHYLHEXEDRONE * 07-18-19 84 FR 34291 7/18/2019 I
N-ETHYLHEXEDRONE ** 07-18-21 86 FR 37672 7/18/2021 I
N-ETHYLHEXEDRONE 06-01-22 87 FR 32996 6/1/2022 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE * 10-15-87 52 FR 38225 10/15/1987 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE ** 10-13-88 53 FR 40061 10/13/1988 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORFENTANYL (N-PHENYL-N-(PIPERIDIN-4- 09-17-19 04-17-20 85 FR 21320 5/18/2020 II
YL)PROPIONAMIDE)

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 14 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
OLICERIDINE 10-30-20 85 FR 68749 10/30/2020 II
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
ORTHO-FLUOROACRYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I
ORTHO-FLUOROBUTYRYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2- 10-26-17 82 FR 49504 10/26/2017 I
FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)) *
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2- 10-25-19 84 FR 57323 10/25/2019 I
FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL))
ORTHO-FLUOROISOBUTYRYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I
ORTHO-METHYL ACETYLFENTANYL 04-27-21 86 FR 22113 4/27/2021 I
ORTHO-METHYL METHOXYACETYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PARA-FLUORO FURANYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I
PARA-FLUOROFENTANYL * 02-07-86 51 FR 4722 3/10/1986 I
PARA-FLUOROFENTANYL ** 03-10-87 52 FR 7270 3/10/1987 I
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
PARA-METHOXYMETHAMPHETAMINE (PMMA), 1-(4- 05-15-20 06-25-21 86 FR 33508 7/26/2021 I
METHOXYPHENYL)-N-METHYLPROPAN-2-AMINE
PARA-METHYLFENTANYL 04-27-21 86 FR 22113 4/27/2021 I
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
PENTEDRONE * 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE ** 03-04-16 81 FR 11429 3/4/2016 I
PENTEDRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
PENTYLONE * 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE ** 03-04-16 81 FR 11429 3/4/2016 I
PENTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PEPAP * 07-10-85 50 FR 28098 8/12/1985 I
PEPAP ** 08-11-86 51 FR 28695 8/12/1986 I
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
PERAMPANEL [2-(2-OXO-1-PHENYL-5-PYRIDIN-2-YL-l ,2- 10-22-13 12-02-13 78 FR 72013 1/2/2014 III
DIHYDROPYRIDIN-3-YL)BENZONITRILE]
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 15 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
PHENYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III
ANDROSTANO[3,2-C]PRYAZOLE)
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-10-14 79 FR 7577 2/10/2014 I
CARBOXYLATE (5-FLUORO-PB–22; 5F–PB–22) *
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-05-16 81 FR 6175 2/5/2016 I
CARBOXYLATE (5-FLUORO-PB–22; 5F–PB–22) **
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 09-06-16 81 FR 61130 9/6/2016 I
CARBOXYLATE (5-FLUORO-PB-22; 5F-PB-22)
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-10-14 79 FR 7577 2/10/2014 I
(PB–22; QUPIC) *
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-05-16 81 FR 6175 2/5/2016 I
(PB–22; QUPIC) **
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB- 09-06-16 81 FR 61130 9/6/2016 I
22; QUPIC)
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II
REMIMAZOLAM (4H-IMIDAZOL[1,2-A][1,4]BENZODIAZEPINE- 10-06-20 85 FR 63014 10/6/2020 IV
4-PROPIONIC ACID)
SAMIDORPHAN 04-19-21 86 FR 20284 4/19/2021 II -> 0
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
SERDEXMETHYLPHENIDATE 05-07-21 86 FR 24487 5/7/2021 IV
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
SOLRIAMFETOL (2-AMINO-3-PHENYLPROPYL CAR- 06-17-19 84 FR 27943 6/17/2019 IV
BAMATE; BENZENEPROPANOL,BETA-AMINO-, CARBAMATE
(ESTER))
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
TETRAHYDROFURANYL FENTANYL (N-(1- 10-26-17 82 FR 49504 10/26/2017 I
PHENETHYLPIPERIDIN-4-YL)-N-
PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE) *

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 16 of 17
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
TETRAHYDROFURANYL FENTANYL (N-(1- 11-29-18 83 FR 61320 11/29/2018 I
PHENETHYLPIPERIDIN-4-YL)-N-
PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE)
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
THENYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I Expired
11/29/86
THIAFENTANIL 08-26-16 81 FR 58834 8/26/2016 II
THIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
THIOFURANYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3- 11-04-13 07-02-14 79 FR 37623 8/18/2014 IV
METHOXYPHENYL)CYCLOHEXANOL)
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
ZIPEPROL (1-METHOXY-3-[4-(2-METHOXY-2- 05-14-20 11-21-22 87 FR 70717 12/21/2022 I
PHENYLETHYL)PIPERAZIN-1-YL]-1-PHENYLPROPAN-2-OL)
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV

Scheduling Actions - Alphabetical Order


07-Jul-23 Page 17 of 17
Scheduling Actions
Chronological Order
Scheduling Actions
- Chronological Order -
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE

METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II


AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I

Scheduling Actions - Chronological Order


Page 1 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted
RX
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted
RX
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV

Scheduling Actions - Chronological Order


Page 2 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V
3-METHYLFENTANYL * 03-25-85 50 FR 11690 4/25/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) * 05-31-85 50 FR 23118 7/1/1985 I
MPPP * 07-10-85 50 FR 28098 8/12/1985 I
PEPAP * 07-10-85 50 FR 28098 8/12/1985 I
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
ACETYL-ALPHA-METHYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
3-METHYLTHIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I

Scheduling Actions - Chronological Order


Page 3 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
THENYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I Expired
11/29/86
BETA-HYDROXYFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXY-3-METHYLFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired
11/29/86
ALPHA-METHYLTHIOFENTANYL * 10-29-85 50 FR 43698 11/29/1985 I
PARA-FLUOROFENTANYL * 02-07-86 51 FR 4722 3/10/1986 I
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
3-METHYLFENTANYL ** 04-24-86 51 FR 15474 4/25/1986 I
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) ** 06-17-86 51 FR 21911 7/1/1986 I
MPPP ** 08-11-86 51 FR 28695 8/12/1986 I
PEPAP ** 08-11-86 51 FR 28695 8/12/1986 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
ALPHA-METHYLTHIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXYFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
ACETYL-ALPHA-METHYLFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
THIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
3-METHYLTHIOFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXY-3-METHYLFENTANYL ** 11-26-86 51 FR 42834 11/29/1986 I Expired
5/29/87
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
PARA-FLUOROFENTANYL ** 03-10-87 52 FR 7270 3/10/1987 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I
4-METHYLAMINOREX * 10-15-87 52 FR 38225 10/15/1987 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE * 10-15-87 52 FR 38225 10/15/1987 I

Scheduling Actions - Chronological Order


Page 4 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-15-87 52 FR 38225 10/15/1987 I
MDEA) *
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
N,N-DIMETHYLAMPHETAMINE * 08-03-88 53 FR 29232 8/3/1988 I
4-METHYLAMINOREX ** 10-13-88 53 FR 40061 10/13/1988 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE ** 10-13-88 53 FR 40061 10/13/1988 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-13-88 53 FR 40061 10/13/1988 I
MDEA) **
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE; 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
MDEA)
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
N,N-DIMETHYLAMPHETAMINE ** 08-02-89 54 FR 31815 8/2/1989 I
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
METHCATHINONE * 05-01-92 57 FR 18824 5/1/1992 I
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0
Superseded
10/97
AMINOREX * 09-21-92 57 FR 43399 9/21/1992 I
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
ALPHA-ETHYLTRYPTAMINE * 03-12-93 58 FR 13533 3/12/1993 I
METHCATHINONE ** 04-29-93 58 FR 25934 5/1/1993 I
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II
AMINOREX ** 08-24-93 58 FR 44611 9/21/1993 I
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I

Scheduling Actions - Chronological Order


Page 5 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE * 01-06-94 59 FR 00671 1/6/1994 I
ALPHA-ETHYLTRYPTAMINE ** 03-07-94 59 FR 10720 3/12/1994 I
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE ** 12-21-94 59 FR 65710 1/6/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II
FENFLURAMINE 05-06-97 05-06-97 62 FR 24620 IV -> 0
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III
products
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification
of CII
control
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification
of CIV
control
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-20-02 67 FR 59163 9/20/2002 I
T-7) *
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
FENFLURAMINE 05-06-97 05-15-03 68 FR 26247 IV
Withdrew
97
proposed
rule
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-10-03 68 FR 53289 9/20/2003 I
T-7) **
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
T-7)
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0

Scheduling Actions - Chronological Order


Page 6 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 04-01-04 69 FR 17034 4/1/2004 I
**
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
3,17-dione)
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
en-17-ol, madol)
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE) * 10-21-11 76 FR 65371 10/21/2011 I
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I
(METHYLONE) *
3,4-METHYLENEDIOXYPYROVALERONE (MDPV) * 10-21-11 76 FR 65371 10/21/2011 I
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III
ANDROSTANO[3,2-C]PRYAZOLE)

Scheduling Actions - Chronological Order


Page 7 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
METHASTERONE (2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III
ANDROSTAN-17BETA-OL-3-ONE)
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 04-12-13 78 FR 21818 4/12/2013 I
(METHYLONE)
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144) *
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-
UR-144, XLR11) *
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-16-13 78 FR 28735 5/16/2013 I
CARBOXAMIDE (APINACA, AKB48) *
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I
METHOXYBENZYL)ETHANAMINE (25B-NBOMe) *
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) 11-15-13 78 FR 68716 11/15/2013 I
ETHANAMINE (25I-NBOMe) *
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I
METHOXYBENZYL)ETHANAMINE (25C-NBOMe) *
PERAMPANEL [2-(2-OXO-1-PHENYL-5-PYRIDIN-2-YL-l ,2- 10-22-13 12-02-13 78 FR 72013 1/2/2014 III
DIHYDROPYRIDIN-3-YL)BENZONITRILE]
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-10-14 79 FR 7577 2/10/2014 I
CARBOXYLATE (5-FLUORO-PB–22; 5F–PB–22) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 02-10-14 79 FR 7577 2/10/2014 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-10-14 79 FR 7577 2/10/2014 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA) *
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-10-14 79 FR 7577 2/10/2014 I
(PB–22; QUPIC) *
ALFAXALONE (5α-PREGNAN-3α-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) * 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE * 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE * 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE * 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) * 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) * 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-07-14 79 FR 12938 3/7/2014 I
MePPP) *
4-FLUORO-N-METHYLCATHINONE (4-FMC) * 03-07-14 79 FR 12938 3/7/2014 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) * 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE * 03-07-14 79 FR 12938 3/7/2014 I
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3- 11-04-13 07-02-14 79 FR 37623 8/18/2014 IV
METHOXYPHENYL)CYCLOHEXANOL)
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II

Scheduling Actions - Chronological Order


Page 8 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1- 01-30-15 80 FR 5042 1/30/2015 I
(CYCLOHEXYLMETHYL)1H-INDAZOLE-3-CARBOXAMIDE (AB-
CHMINACA) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H- 01-30-15 80 FR 5042 1/30/2015 I
INDAZOLE-3-CARBOXAMIDE (AB-PINACA) *
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1- 01-30-15 80 FR 5042 1/30/2015 I
YL)METHANONE (THJ-2201) *
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-15-15 80 FR 27854 5/15/2015 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144) **
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-15-15 80 FR 27854 5/15/2015 I
CARBOXAMIDE (APINACA, AKB48) **
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-15-15 80 FR 27854 5/5/2015 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-
UR-144, XLR11) **
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-17-15 80 FR 42381 7/17/2015 I
PHENYLACETAMIDE) *
ELUXADOLINE 08-11-15 11-12-15 80 FR 69861 12/17/2015 IV
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 02-05-16 81 FR 6171 2/5/2016 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-05-16 81 FR 6175 2/5/2016 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA) **
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-05-16 81 FR 6175 2/5/2016 I
(PB–22; QUPIC) **
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-05-16 81 FR 6175 2/5/2016 I
CARBOXYLATE (5-FLUORO-PB–22; 5F–PB–22) **
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 02-05-16 81 FR 6175 2/5/2016 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA) **
PENTYLONE ** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) ** 03-04-16 81 FR 11429 3/4/2016 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) ** 03-04-16 81 FR 11429 3/4/2016 I
PENTEDRONE ** 03-04-16 81 FR 11429 3/4/2016 I
4-FLUORO-N-METHYLCATHINONE (4-FMC) ** 03-04-16 81 FR 11429 3/4/2016 I
BUTYLONE ** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) ** 03-04-16 81 FR 11429 3/4/2016 I
NAPHYRONE ** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 81 FR 11429 3/4/2016 I
MePPP) **
4-METHYL-N-ETHYLCATHINONE (4-MEC) ** 03-04-16 81 FR 11429 3/4/2016 I
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-11-16 81 FR 29142 5/11/2016 I
TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLUORO-
UR-144, XLR11)
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-11-16 81 FR 29142 5/11/2016 I
CARBOXAMIDE (APINACA, AKB48)

Scheduling Actions - Chronological Order


Page 9 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-11-16 81 FR 29142 5/11/2016 I
TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)
BRIVARACETAM (BRV; UCB-34714; BRIVIACT) 05-12-16 81 FR 29487 5/12/2016 V
BUTYRYL FENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
BETA-HYDROXYTHIOFENTANYL * 05-12-16 81 FR 29492 5/12/2016 I
3,4-DICHLORO-N-[(1- 04-14-16 81 FR 22023 5/15/2016 I
DIMETHYLAMINO)CYCLOHEXYLMETHYL]BENZAMIDE)
(AH-7921)
THIAFENTANIL 08-26-16 81 FR 58834 8/26/2016 II
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 09-06-16 81 FR 61130 9/6/2016 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-
FUBINACA)
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB- 09-06-16 81 FR 61130 9/6/2016 I
22; QUPIC)
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 09-06-16 81 FR 61130 9/6/2016 I
1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 09-06-16 81 FR 61130 9/6/2016 I
CARBOXYLATE (5-FLUORO-PB-22; 5F-PB-22)
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N- 11-14-16 81 FR 79389 11/14/2016 I
METHYLBENZAMIDE (U-47700) *
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2- 11-29-16 81 FR 85873 11/29/2016 I
CARBOXAMIDE (FURANYL FENTANYL) *
NAPHYRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
3-FLUORO-N-METHYLCATHINONE (3-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-FLUORO-N-METHYLCATHINONE (4-FMC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
MePPP)
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
BUTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTEDRONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
PENTYLONE 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
4-METHYL-N-ETHYLCATHINONE (4-MEC) 03-04-16 03-01-17 82 FR 12171 3/1/2017 I
DRONABINOL IN ORAL SOLUTION IN DRUG PRODUCT 03-23-17 82 FR 14815 3/23/2017 II
APPROVED FOR MARKETING BY U.S. FOOD AND DRUG
ADMIN.
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA) *
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB) *
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 04-10-17 82 FR 17119 4/10/2017 I
3-CARBOXAMIDE (5F–APINACA, 5F–AKB48) *
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 04-10-17 82 FR 17119 4/10/2017 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE
(ADB–FUBINACA) *

Scheduling Actions - Chronological Order


Page 10 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA) *
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 04-10-17 82 FR 17119 4/10/2017 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE
(MDMB–FUBINACA) *
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 05-03-17 82 FR 20544 5/3/2017 I
YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL) *
ACETYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 06-07-17 82 FR 26349 6/7/2017 I
PHENYLACETAMIDE)
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-14-17 82 FR 32453 7/14/2017 I
PHENYLACRYLAMIDE) *
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1- 10-16-17 82 FR 47971 10/16/2017 I
(CYCLOHEXYLMETHYL)1H-INDAZOLE-3-CARBOXAMIDE (AB-
CHMINACA)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H- 10-16-17 82 FR 47971 10/16/2017 I
INDAZOLE-3-CARBOXAMIDE (AB-PINACA)
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1- 10-16-17 82 FR 47971 10/16/2017 I
YL)METHANONE (THJ-2201)
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2- 10-26-17 82 FR 49504 10/26/2017 I
FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL)) *
METHOXYACETYL FENTANYL (2-METHOXY-N-(1- 10-26-17 82 FR 49504 10/26/2017 I
PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE) *
TETRAHYDROFURANYL FENTANYL (N-(1- 10-26-17 82 FR 49504 10/26/2017 I
PHENETHYLPIPERIDIN-4-YL)-N-
PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE) *
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 11-03-17 82 FR 51154 11/3/2017 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE *
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4- 01-04-18 83 FR 469 1/4/2018 I
YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE) *
MT-45 (1-CYCLOHEXYL-4-(1,2- 12-13-17 82 FR 58557 1/12/2018 I
DIPHENYLETHYL)PIPERAZINE))
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 01-30-18 83 FR 4411 1/30/2018 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 02-01-18 83 FR 4580 2/1/2018 I
(VALERYL FENTANYL) *
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL) *
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL) *
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 02-01-18 83 FR 4580 2/1/2018 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)*
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 02-01-18 83 FR 4580 2/1/2018 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL) *
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 02-01-18 83 FR 4580 2/1/2018 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL) *

Scheduling Actions - Chronological Order


Page 11 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1- 02-01-18 83 FR 4580 2/1/2018 I
PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL) *
FENTANYL-RELATED SUBSTANCES, AS DEFINED IN 21 02-06-18 83 FR 5188 2/6/2018 I
CFR 1308.11(h)*
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLBUTANAMIDE 04-20-18 83 FR 17486 4/20/2018 I
(BUTYRYL FENTANYL)
3,4-DICHLORO-N-[2-(DIMETHYLAMINO)CYCLOHEXYL]-N- 04-20-18 83 FR 17486 4/20/2018 I
METHYLBENZAMIDE (U-47700)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 07-10-18 83 FR 31877 7/10/2018 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA) *
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-10-18 83 FR 31877 7/10/2018 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA) *
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 07-10-18 83 FR 31877 7/10/2018 I
CARBOXYLATE (NM2201; CBL2201) *
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 07-10-18 83 FR 31877 7/10/2018 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA) *
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-10-18 83 FR 31877 7/10/2018 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA) *
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 08-31-18 83 FR 44474 8/31/2018 I
ONE (N-ETHYLPENTYLONE, EPHYLONE) *
APPROVED CANNABIDIOL DRUGS , AS DEFINED IN 21 CFR 09-28-18 83 FR 48953 9/28/2018 V
1308.15(f)
TETRAHYDROFURANYL FENTANYL (N-(1- 11-29-18 83 FR 61320 11/29/2018 I
PHENETHYLPIPERIDIN-4-YL)-N-
PHENYLTETRAHYDROFURAN-2-CARBOXAMIDE)
ACRYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-29-18 83 FR 61320 11/29/2018 I
PHENYLACRYLAMIDE)
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-29-18 83 FR 61320 11/29/2018 I
YL)ISOBUTYRAMIDE (4-FLUOROISOBUTYRYL FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLFURAN-2- 11-29-18 83 FR 61320 11/29/2018 I
CARBOXAMIDE (FURANYL FENTANYL)
N-(2-FLUOROPHENYL)-2-METHOXY-N-(1- 11-29-18 83 FR 61320 11/29/2018 I
PHENETHYLPIPERIDIN-4-YL)ACETAMIDE (OCFENTANIL)
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1- 01-29-19 84 FR 444 1/29/2019 I
(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3-CARBOXAMIDE
(MAB-CHMINACA)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA) **
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA) **
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 04-08-19 84 FR 13796 4/8/2019 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE
(ADB–FUBINACA) **
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB) **

Scheduling Actions - Chronological Order


Page 12 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 04-08-19 84 FR 13796 4/8/2019 I
3-CARBOXAMIDE (5F-APINACA, 5F-AKB48) **
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 04-08-19 84 FR 13796 4/8/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
FUBINACA) **
(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 04-16-19 84 FR 15505 4/16/2019 I
TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144) *
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 04-16-19 84 FR 15505 4/16/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA) *
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 04-16-19 84 FR 15505 4/16/2019 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA) *
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 04-16-19 84 FR 15505 4/16/2019 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25) *
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-16-19 84 FR 15505 4/16/2019 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA) *
BETA-HYDROXYTHIOFENTANYL 05-08-19 84 FR 20023 5/8/2019 I
BREXANOLONE (3Α-HYDROXY-5Α-PREGNAN-20-ONE), 06-17-19 84 FR 27938 6/17/2019 IV
ALLOPREGNANOLONE
SOLRIAMFETOL (2-AMINO-3-PHENYLPROPYL CAR- 06-17-19 84 FR 27943 6/17/2019 IV
BAMATE; BENZENEPROPANOL,BETA-AMINO-, CARBAMATE
(ESTER))
N-ETHYLHEXEDRONE * 07-18-19 84 FR 34291 7/18/2019 I
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) * 07-18-19 84 FR 34291 7/18/2019 I
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) * 07-18-19 84 FR 34291 7/18/2019 I
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4- 07-18-19 84 FR 34291 7/18/2019 I
MEAP) *
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) * 07-18-19 84 FR 34291 7/18/2019 I
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 07-18-19 84 FR 34291 7/18/2019 I
CHLORO-A-PVP) *
N-(4-FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 10-25-19 84 FR 57323 10/25/2019 I
YL)BUTYRAMIDE (PARA-FLUOROBUTYRYL FENTANYL)
CYCLOPROPYL FENTANYL (N-(1-PHENETHYLPIPERIDIN-4- 10-25-19 84 FR 57323 10/25/2019 I
YL)-N-PHENYLCYCLOPROPANECARBOXAMIDE)
METHOXYACETYL FENTANYL (2-METHOXY-N-(1- 10-25-19 84 FR 57323 10/25/2019 I
PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)
ORTHO-FLUOROFENTANYL OR 2-FLUOROFENTANYL (N-(2- 10-25-19 84 FR 57323 10/25/2019 I
FLUOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4-YL))
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 10-30-19 84 FR 58045 11/3/2019 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE **
N-(ADAMANTAN-1-YL)-1-(5-FLUOROPENTYL)-1H-INDAZOLE- 01-24-20 85 FR 4211 1/24/2020 I
3-CARBOXAMIDE (5F-APINACA, 5F-AKB48)
METHYL 2-(1-(4-FLUOROBENZYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
FUBINACA)

Scheduling Actions - Chronological Order


Page 13 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-(4- 01-24-20 85 FR 4211 1/24/2020 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (ADB-
FUBINACA)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3-METHYLBUTANOATE (5F-AMB)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-ADB, 5F-
MDMB-PINACA)
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 01-24-20 85 FR 4211 1/24/2020 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (MDMB-
CHMICA)
6β-NALTREXOL ((5a,6β)-17-(CYCLOPROPYLMETHYL)-4,5- 01-24-20 85 FR 4215 1/24/2020 II -> 0
EPOXYMORPHINAN-3,6,14-TRIOL)
LASMIDITAN [2,4,6-TRIFLUORO-N-(6-(1-METHYLPIPERIDINE- 01-31-20 85 FR 5557 1/31/2020 V
4-CARBONYL)PYRIDINE-2-YL-BENZAMIDE]
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 01-30-20 85 FR 5321 2/1/2020 I
(VALERYL FENTANYL) **
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 01-30-20 85 FR 5321 2/1/2020 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 01-30-20 85 FR 5321 2/1/2020 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL) **
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 01-30-20 85 FR 5321 2/1/2020 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL) **
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 01-30-20 85 FR 5321 2/1/2020 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)**
CENOBAMATE [(1R)-1-(2-CHLOROPHENYL)-2-(TETRAZOL-2- 03-10-20 85 FR 13741 3/10/2020 V
YL)ETHYL]CARBAMATE
FUB-AMB, MMB-FUBINACA (METHYL 2-(1-(4- 03-30-20 85 FR 17494 3/30/2020 I
FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDO)-3-
METHYLBUTANOATE
LEMBOREXANT 04-07-20 85 FR 19387 4/7/2020 IV
NORFENTANYL (N-PHENYL-N-(PIPERIDIN-4- 09-17-19 04-17-20 85 FR 21320 5/18/2020 II
YL)PROPIONAMIDE)
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-13-20 85 FR 42296 7/10/2020 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA) **
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 07-13-20 85 FR 42296 7/10/2020 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA) **
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 07-13-20 85 FR 42296 7/10/2020 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA) **
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 07-13-20 85 FR 42296 7/10/2020 I
CARBOXYLATE (NM2201; CBL2201) **
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 07-13-20 85 FR 42296 7/10/2020 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA) **
ISOTONITAZENE (N,N-DIETHYL-2-(2-(4 08-20-20 85 FR 51342 8/20/2020 I
ISOPROPOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-
YL)ETHAN-1-AMINE) *

Scheduling Actions - Chronological Order


Page 14 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 08-27-20 85 FR 52915 8/31/2020 I
ONE (N-ETHYLPENTYLONE, EPHYLONE) **
CROTONYL FENTANYL ((E)-N-(1-PHENETHYLPIPERIDIN-4- 10-02-20 85 FR 62215 10/2/2020 I
YL)-N-PHENYLBUT-2-ENAMIDE)
REMIMAZOLAM (4H-IMIDAZOL[1,2-A][1,4]BENZODIAZEPINE- 10-06-20 85 FR 63014 10/6/2020 IV
4-PROPIONIC ACID)
OLICERIDINE 10-30-20 85 FR 68749 10/30/2020 II
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-25-20 85 FR 75231 11/25/2020 I
PHENYLCYCLOPENTANECARBOXAMIDE (CYCLOPENTYL
FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 11-25-20 85 FR 75231 11/25/2020 I
PHENYLISOBUTYRAMIDE (ISOBUTYRYL FENTANYL)
N-(4-CHLOROPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-25-20 85 FR 75231 11/25/2020 I
YL)ISOBUTYRAMIDE (PARA-CHLOROISOBUTYRYL
FENTANYL)
N-(4-METHOXYPHENYL)-N-(1-PHENETHYLPIPERIDIN-4- 11-25-20 85 FR 75231 11/25/2020 I
YL)BUTYRAMIDE (PARA-METHOXYBUTYRYL FENTANYL)
N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLPENTANAMIDE 11-25-20 85 FR 75231 11/25/2020 I
(VALERYL FENTANYL)
1-(1-(1-(4-BROMOPHENYL)ETHYL)PIPERIDIN-4-YL)-1,3- 03-01-21 86 FR 11862 3/1/2021 I
DIHYDRO-2H-BENZO[D]IMIDAZOL-2-ONE (BRORPHINE) *
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 03-31-21 86 FR 16669 4/16/2021 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA) **
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 03-31-21 86 FR 16669 4/16/2021 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA) **
(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 03-31-21 86 FR 16669 4/16/2021 I
TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144) **
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 03-31-21 86 FR 16669 4/16/2021 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25) **
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 03-31-21 86 FR 16669 4/16/2021 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA) **
SAMIDORPHAN 04-19-21 86 FR 20284 4/19/2021 II -> 0
THIOFURANYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
PARA-METHYLFENTANYL 04-27-21 86 FR 22113 4/27/2021 I
ORTHO-METHYL METHOXYACETYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
ORTHO-FLUOROBUTYRYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
4'-METHYL ACETYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
2'-FLUORO ORTHO-FLUOROFENTANYL 04-27-21 86 FR 22113 4/27/2021 I
BETA'-PHENYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
BETA-METHYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
ORTHO-METHYL ACETYLFENTANYL 04-27-21 86 FR 22113 4/27/2021 I
PHENYL FENTANYL 04-27-21 86 FR 22113 4/27/2021 I
FENTANYL CARBAMATE 05-04-21 86 FR 23602 5/4/2021 I
PARA-FLUORO FURANYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I

Scheduling Actions - Chronological Order


Page 15 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ORTHO-FLUOROACRYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I
ORTHO-FLUOROISOBUTYRYL FENTANYL 05-04-21 86 FR 23602 5/4/2021 I
SERDEXMETHYLPHENIDATE 05-07-21 86 FR 24487 5/7/2021 IV
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 06-10-21 86 FR 30775 6/10/2021 I
PYRROLO[2,3-B]PYRIDINE-3-CARBOXAMIDE (5F-CUMYL-
P7AICA)
NAPHTHALEN-1-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 06-10-21 86 FR 30775 6/10/2021 I
CARBOXYLATE (NM2201; CBL2201)
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(5- 06-10-21 86 FR 30775 6/10/2021 I
FLUOROPENTYL)-1H-INDAZOLE-3-CARBOXAMIDE (5F-AB-
PINACA)
1-(4-CYANOBUTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 06-10-21 86 FR 30775 6/10/2021 I
INDAZOLE-3-CARBOXAMIDE (4-CN-CUMYL-BUTINACA)
METHYL 2-(1-(CYCLOHEXYLMETHYL)-1H-INDOLE-3- 06-10-21 86 FR 30775 6/10/2021 I
CARBOXAMIDO)-3-METHYLBUTANOATE (MMB-CHMICA,
AMB-CHMICA)
1-(1,3-BENZODIOXOL-5-YL)-2-(ETHYLAMINO)-PENTAN-1- 06-14-21 86 FR 31427 6/14/2021 I
ONE (N-ETHYLPENTYLONE, EPHYLONE)
N-ETHYLHEXEDRONE ** 07-18-21 86 FR 37672 7/18/2021 I
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) ** 07-18-21 86 FR 37672 7/18/2021 I
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) 07-18-21 86 FR 37672 7/18/2021 I
**
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4- 07-18-21 86 FR 37672 7/18/2021 I
MEAP) **
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) ** 07-18-21 86 FR 37672 7/18/2021 I
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 07-18-21 86 FR 37672 7/18/2021 I
CHLORO-A-PVP) **
PARA-METHOXYMETHAMPHETAMINE (PMMA), 1-(4- 05-15-20 06-25-21 86 FR 33508 7/26/2021 I
METHOXYPHENYL)-N-METHYLPROPAN-2-AMINE
4,4′-DIMETHYLAMINOREX (4,4′-DMAR; 4,5-DIHYDRO-4- 04-07-20 08-12-21 86 FR 44270 9/13/2021 I
METHYL-5-(4-METHYLPHENYL)-2-OXAZOLAMINE)
ISOTONITAZENE (N,N-DIETHYL-2-(2-(4 11-04-21 86 FR 60761 12/6/2021 I
ISOPROPOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-
YL)ETHAN-1-AMINE)
4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE (4-OH-DiPT) 01-14-22 01-14-22 87 FR 2376 I
N,N-DIISOPROPYLTRYPTAMINE (DiPT) 01-14-22 01-14-22 87 FR 2376 I
5-METHOXY-N,N-DIETHYLTRYPTAMINE (MeO-DET) 01-14-22 01-14-22 87 FR 2376 I
5-METHOXY-N-METHYL-N-ISOPROPYLTRYPTAMINE (5-MeO- 01-14-22 01-14-22 87 FR 2376 I
MiPT)
5-METHOXY-ALPHA-METHYLTRYPTAMINE (5-MeO-AMT) 01-14-22 01-14-22 87 FR 2376 I
DARIDOREXANT (QUVIVIQ) 04-07-22 87 FR 20313 4/7/2022 IV
N-(ADAMANTAN-1-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE- 04-07-22 87 FR 20318 4/7/2022 I
3-CARBOXAMIDE (FUB-AKB48; FUB-APINACA)
(1-(4-FLUOROBENZYL)-1H-INDOL-3-YL)(2,2,3,3- 04-07-22 87 FR 20318 4/7/2022 I
TETRAMETHYLCYCLOPROPYL)METHANONE (FUB-144)

Scheduling Actions - Chronological Order


Page 16 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ETHYL 2-(1-(5-FLUOROPENTYL)-1H-INDAZOLE-3- 04-07-22 87 FR 20318 4/7/2022 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-EDMB-
PINACA)
METHYL 2-(1-(5-FLUOROPENTYL)-1H-INDOLE-3- 04-07-22 87 FR 20318 4/7/2022 I
CARBOXAMIDO)-3,3-DIMETHYLBUTANOATE (5F-MDMB-
PICA)
1-(5-FLUOROPENTYL)-N-(2-PHENYLPROPAN-2-YL)-1H- 04-07-22 87 FR 20318 4/7/2022 I
INDAZOLE-3-CARBOXAMIDE (5F-CUMYL-PINACA; SGT-25)
2,5-DIMETHOXY-4-IODOAMPHETAMINE (DOI) 04-11-22 04-11-22 87 FR 21069 I
2,5-DIMETHOXY-4-CHLOROAMPHETAMINE (DOC) 04-11-22 04-11-22 87 FR 21069 I
2-(2-(4-BUTOXYBENZYL)-5-NITRO-1H-BENZIMIDAZOL-1-YL)- 04-12-22 87 FR 21556 4/12/2022 I
N,N-DIETHYLETHAN-1-AMINE (BUTONITAZENE) *
2-(4-ETHOXYBENZYL)-5-NITRO-1-(2-(PYRROLIDIN-1- 04-12-22 87 FR 21556 4/12/2022 I
YL)ETHYL)-1H-BENZIMIDAZOLE (N-PYRROLIDINO
ETONITAZENE) *
N,N-DIETHYL-2-(5-NITRO-2-(4-PROPOXYBENZYL)-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (PROTONITAZENE) *
N,N-DIETHYL-2-(2-(4-METHOXYBENZYL)-1H-BENZIMIDAZOL- 04-12-22 87 FR 21556 4/12/2022 I
1-YL)ETHAN-1-AMINE (METODESNITAZENE) *
N,N-DIETHYL-2-(2-(4-FLUOROBENZYL)-5-NITRO-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (FLUNITAZENE) *
N,N-DIETHYL-2-(2-(4- METHOXYBENZYL)-5-NITRO-1H- 04-12-22 87 FR 21556 4/12/2022 I
BENZIMIDAZOL-1-YL)ETHAN-1-AMINE (METONITAZENE) *
2-(2-(4-ETHOXYBENZYL)-1H-BENZIMIDAZOL-1-YL)-N,N- 04-12-22 87 FR 21556 4/12/2022 I
DIETHYLETHAN-1-AMINE (ETODESNITAZENE; ETAZENE) *
3-ALPHA-HYDROXY-3-BETA-METHYL-5-ALPHA-PREGNAN- 06-01-22 87 FR 32991 6/1/2022 V
20-ONE (GANAXOLONE)
ALPHA-PYRROLIDINOHEXANOPHENONE (A-PHP) 06-01-22 87 FR 32996 6/1/2022 I
N-ETHYLHEXEDRONE 06-01-22 87 FR 32996 6/1/2022 I
4'-CHLORO-ALPHA-PYRROLIDINOVALEROPHENONE (4- 06-01-22 87 FR 32996 6/1/2022 I
CHLORO-A-PVP)
4´-METHYL-ALPHA-PYRROLIDINOHEXIOPHENONE (MPHP) 06-01-22 87 FR 32996 6/1/2022 I
4-METHYL-ALPHA-ETHYLAMINOPENTIOPHENONE (4- 06-01-22 87 FR 32996 6/1/2022 I
MEAP)
ALPHA-PYRROLIDINOHEPTAPHENONE (PV8) 06-01-22 87 FR 32996 6/1/2022 I
METHOXETAMINE 12-07-21 06-07-22 87 FR 34166 7/6/2022 I
5-METHOXY-ALPHA-METHYLTRYPTAMINE (5-MeO-AMT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
N,N-DIISOPROPYLTRYPTAMINE (DiPT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
5-METHOXY-N-METHYL-N-ISOPROPYLTRYPTAMINE (5-MeO- 01-14-22 07-27-22 87 FR 45076 I Withdrew
MiPT) 2022
proposed
rule

Scheduling Actions - Chronological Order


Page 17 of 18
07-Jul-23
FINAL ORDER

SUBSTANCE PROPOSAL FEDERAL


*Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA
**Extension of temporary control DATE DATE CITATION DATE SCHEDULE
4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE (4-OH-DiPT) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
5-METHOXY-N,N-DIETHYLTRYPTAMINE (MeO-DET) 01-14-22 07-27-22 87 FR 45076 I Withdrew
2022
proposed
rule
2,5-DIMETHOXY-4-CHLOROAMPHETAMINE (DOC) 04-11-22 08-29-22 87 FR 52712 I Withdrew
2022
proposed
rule
2,5-DIMETHOXY-4-IODOAMPHETAMINE (DOI) 04-11-22 08-29-22 87 FR 52712 I Withdrew
2022
proposed
rule
AMINEPTINE (7-[(10,11-DIHYDRO-5H- 07-22-22 11-17-22 87 FR 68895 12/19/2022 I
DIBENZO[A,D]CYCLOHEPTEN-5-YL)AMINO]HEPTANOIC
ACID)
ZIPEPROL (1-METHOXY-3-[4-(2-METHOXY-2- 05-14-20 11-21-22 87 FR 70717 12/21/2022 I
PHENYLETHYL)PIPERAZIN-1-YL]-1-PHENYLPROPAN-2-OL)
MESOCARB (N-PHENYL-N'-(3-(1-PHENYLPROPAN-2-YL)- 08-11-21 11-22-22 87 FR 71247 12/22/2022 I
1,2,3-OXADIAZOL-3-IUM-5-YL)CARBAMIMIDATE)
FENFLURAMINE 07-19-22 12-23-22 87 FR 78857 12/23/2022 IV -> 0
METHIOPROPAMINE (N-METHYL-1-(THIOPHEN-2- 09-02-21 12-09-22 87 FR 75470 1/9/2023 I
YL)PROPANE-2-AMINE
1-(1-(1-(4-BROMOPHENYL)ETHYL)PIPERIDIN-4-YL)-1,3- 03-06-23 88 FR 13692 4/5/2023 I
DIHYDRO-2H-BENZO[D]IMIDAZOL-2-ONE (BRORPHINE)
EUTYLONE (1-(1,3-BENZODIOXOL-5-YL)-2- 04-10-23 88 FR 21101 4/10/2023 I
(ETHYLAMINO)BUTAN-1-ONE)

Scheduling Actions - Chronological Order


Page 18 of 18
07-Jul-23
Controlled Substances
Alphabetical Order
Controlled Substances
- Alphabetical Order -

CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

(1-(4-Fluorobenzyl)-1H-indol-3-yl)(2,2,3,3- 7014 I N FUB-144


tetramethylcyclopropyl)methanone
[3,2-c]-furazan-5α-androstan-17β-ol 4000 III N

[3,2-c]pyrazole-androst-4-en-17β-ol 4000 III N

1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine


1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
1-(5-Fluoropentyl)-N-(2-phenylpropan-2-yl)-1H-indazole- 7083 I N 5F-CUMYL-PINACA; SGT-25
3-carboxamide
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N

17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N


androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N

17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N


4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone
hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
17α-Methyl-5α-androstan-17β-ol 4000 III N

17α-methyl-androst-2-ene-3,17β-diol 4000 III N

17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N

17α-Methyl-androstan-3-hydroxyimine-17β-ol 4000 III N

17β-Hydroxy-androstano[2,3-d]isoxazole 4000 III N

17β-Hydroxy-androstano[3,2-c]isoxazole 4000 III N

18a-Homo-3-hydroxy-estra-2,5(10)-dien-17-one 4000 III N

19-Nor-4,9(10)-androstadienedione 4000 III N

19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N


ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N

19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N


ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N

1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N


androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-
androst-1-ene)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 1 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N

1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin


1-Phenylcyclohexylamine 7460 II N PCP precursor
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P
P)
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E) 7509 I N 2C-E

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36
ethanamine (25B-NBOMe)
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82
ethanamine (25C-NBOMe)
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C-T- 7385 I N 2C-T-2
2)
2-(4-iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5
ethanamine (25I-NBOMe)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4
(2C-T-4)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
2-(ethylamino)-2-(3-methoxyphenyl)cyclohexan-1-one 7286 I N MXE, methoxetamine
(methoxetamine)
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7
7)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET

(Positional Isomer: 1-(2,5-dimethoxy-4-


methylphenyl)butan-2-amine)
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
2'-Fluoro ortho-fluorofentanyl (N-(1-(2- 9855 I Y
fluorophenethyl)piperidin-4-yl)-N-(2-
fluorophenyl)propionamide; also known as 2'-fluoro 2-
fluorofentanyl)
2-methoxy-N-(1-phenethylpiperidin-4-yl)-N- 9825 I Y Methoxyacetyl fentanyl
phenylacetamide
2α,17α-dimethyl-17β-hydroxy-5β-androstan-3-one 4000 III N

2α,3α-epithio-17α-methyl-5α-androstan-17β-ol 4000 III N

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 2 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

3,4,5-Trimethoxyamphetamine 7390 I N TMA

(Positional Isomers: 2,4,5-Trimethoxy-amphetamine


(TMA-5), 2,4,6-Trimethoxy-amphetamine (TMA-6),
Escaline)
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA

(Positional Isomer: MDMB)


3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N

3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N

3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one)

(Positional Isomer: 2-FMC)


3-Methylfentanyl 9813 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
3β-hydroxy-estra-4,9,11-trien-17-one 4000 III N

4,4′-Dimethylaminorex (4,4′-DMAR; 4,5-dihydro-4- 1595 I N


methyl-5-(4-methylphenyl)-2-oxazolamine; 4-methyl-5-
(4-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine)
4´-methyl-alpha-pyrrolidinohexiophenone (MPHP) 7446 I N MPHP; 4'-methyl-alpha-pyrrolidinohexanophenone; 1-
(4-methylphenyl)-2-(pyrrolidin-1-yl)hexan-1-one)
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD
ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N

4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP, Despropionyl fentanyl


4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-chloro-17α-methyl-17β-hydroxy-androst-4-en-3-one 4000 III N

4-chloro-17α-methyl-17β-hydroxy-androst-4-ene-3,11- 4000 III N


dione
4-chloro-17α-methyl-androst-4-ene-3β,17β-diol 4000 III N

4-chloro-17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N

4'-chloro-alpha-pyrrolidinovalerophenone (4-chloro-α- 7443 I N 4-chloro-α-PVP; 4'-chloro-α-


PVP) pyrrolidinopentiophenone; 1-(4-chlorophenyl)-2-
(pyrrolidin-1-yl)pentan-1-one)
4-CN-CUMYL-BUTINACA (1-(4-cyanobutyl)-N-(2- 7089 I N 4-cyano-CUMYL-BUTINACA; 4-CN-CUMYL
phenylpropan-2-yl)-1 H-indazole-3-carboxamide) BINACA; CUMYL-4CN-BINACA; SGT-78
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone
one)
4-Fluoroisobutyryl fentanyl (N-(4-fluorophenyl)-N-(1- 9824 I Y Para-fluoroisobutyryl fentanyl
phenethylpiperidin-4-yl)isobutyramide)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 3 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-


(methylamino)propan-1-one)

(Positional Isomer: 2-FMC)


4F-MDMB-BINACA (4F-MDMB-BUTINACA or methyl 2- 7043 I N
(1-(4-fluorobutyl)-1H-indazole-3-carboxamido)-3,3-
dimethylbutanoate)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N
4-en-3-one)
4-Hydroxy-androst-4-ene-3,17-dione 4000 III N Listed as 4-Hydroxy-androst-4-ene-3,17-dione[3,2-
c]pyrazole-5α-androstan-17β-ol
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N
en-3-one)
4-Methoxyamphetamine 7411 I N PMA
4'-Methyl acetyl fentanyl (N-(1-(4- 9819 I Y
methylphenethyl)piperidin-4-yl)-N-phenylacetamide)
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
4-methyl-alpha-ethylaminopentiophenone (4-MEAP) 7245 I N 4-MEAP; 2-(ethylamino)-1-(4-methylphenyl)pentan-1-
one)
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-
methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC),


4-ethylmethcathinone (4-EMC), 4-methylbuphedrone
(4-MeMABP;4-MeBP), 3,4-
dimethylmethcathinone(3,4-DMMC),N-
ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N
ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N

5F-AB-PINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7025 I N


1-(5-fluoropentyl)-1 H-indazole-3-carboxamide)
5F–ADB; 5F–MDMB–PINACA (Methyl 2-(1-(5- 7034 I N 5F-ADB, 5F-MDMB-PINACA, 5F-AEB, 5F-EMB-
fluoropentyl)-1H-indazole-3-carboxamido)-3,3- PINACA
dimethylbutanoate)
5F–AMB (Methyl 2-(1-(5-fluoropentyl)-1H-indazole-3- 7033 I N 5F-AMB
carboxamido)-3-methylbutanoate)
5F–APINACA, 5F–AKB48 (N-(adamantan-1-yl)-1-(5- 7049 I N 5F-APINACA, 5F-AKB48
fluoropentyl)-1H-indazole-3-carboxamide)
5F-CUMYL-P7AICA (1-(5-fluoropentyl)-N-(2- 7085 I N
phenylpropan-2-yl)-1 H-pyrrolo[2,3-b]pyridine-3-
carboxamide)
5-Fluoro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Fluoro-UR-144, XLR-11 and XLR11
indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 4 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22


carboxylate)
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT

(Positional Isomer: 5-Methoxy-N,N-


dipropyltryptamine (5-MeO-DPT))
5-Methoxy-N,N-dimethyltryptamine 7431 I N 5-MeO-DMT

(Positional Isomer: 4-Methoxy-N,N-


dimethyltryptamine (4-MeO-DMT))
5α-Androstan-3,6,17-trione 4000 III N

6-bromo-androsta-1,4-diene-3,17-dione 4000 III N

6-bromo-androstan-3,17-dione 4000 III N

6α-Methyl-androst-4-ene-3,17-dione 4000 III N

AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA


oxobutan-2-yl)-1-(cyclohexylmethyl)-
1H-indazole-3-carboxamide
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA
1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA
1-oxobutan-2-yl)-1-pentyl-1H-indazole-
3-carboxamide)
Acetorphine 9319 I Y

Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y


phenylacetamide)
Acetyl-alpha-methylfentanyl 9815 I Y

Acetyldihydrocodeine 9051 I Y Acetylcodone


Acetylmethadol 9601 I Y Methadyl acetate
Acryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9811 I Y Acryloylfentanyl
phenylacrylamide)
ADB–FUBINACA (N-(1-amino-3,3-dimethyl-1-oxobutan- 7010 I N ADB-FUBINACA
2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA
yl)-1-pentyl-1H-indazole-3-carboxamide)
AH-7921 (3,4-dichloro-N-[(1- 9551 I Y AH-7921
dimethylamino)cyclohexylmethyl]benzamide))
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Alfentanil 9737 II Y Alfenta
Allylprodine 9602 I Y

Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y

Alpha-ethyltryptamine 7249 I N ET, Trip


Alphameprodine 9604 I Y

Alphamethadol 9605 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 5 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Alpha-methylfentanyl 9814 I Y China White, fentanyl


Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
Alpha-methyltryptamine 7432 I N AMT

(Positional Isomer: N-Methyltryptamine)


Alphaprodine 9010 II Y Nisentil
alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
alpha-pyrrolidinoheptaphenone (PV8) 7548 I N PV8; 1-phenyl-2-(pyrrolidin-1-yl)heptan-1-one)
alpha-pyrrolidinohexanophenone (α-PHP) 7544 I N α-PHP; α-pyrrolidinohexanophenone; 1-phenyl-2-
(pyrrolidin-1-yl)hexan-1-one)
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-
yl)pentan-1-one)

(Positional Isomers: 4-methyl-α-


pyrrolidinobutiophenone (4-MePBP), 1-phenyl-2-
(piperidin-1-yl)butan-1-one)
Alprazolam 2882 IV N Xanax
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Amineptine (7-[(10,11-dihydro-5H- 1219 I N
dibenzo[a,d]cyclohepten-5-yl)amino]heptanoic acid)
Aminorex 1585 I N has been sold as methamphetamine
Amobarbital 2125 II N Amytal, Tuinal
Amobarbital & noncontrolled active ingred. 2126 III N

Amobarbital suppository dosage form 2126 III N

Amphetamine 1100 II N Dexedrine, Adderall, Obetrol


Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N

Anileridine 9020 II Y Leritine


APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48
indazole-3-carboxamide
Aprobarbital 2100 III N Alurate
Barbital 2145 IV N Veronal, Plexonal, barbitone
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Benzethidine 9606 I Y

Benzphetamine 1228 III N Didrex, Inapetyl


Benzylmorphine 9052 I Y

Betacetylmethadol 9607 I Y

Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl


Beta-hydroxyfentanyl 9830 I Y China White, fentanyl

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 6 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-


N-phenylpropionamide, N-[1-[2-hydroxy-2-(2-
thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide
Betameprodine 9608 I Y

Betamethadol 9609 I Y

beta-Methyl fentanyl (N-phenyl-N-(1-(2- 9856 I Y


phenylpropyl)piperidin-4-yl)propionamide; also known
as β-methyl fentanyl)
beta'-Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N,3- 9842 I Y
diphenylpropanamide; also known as β'-phenyl
fentanyl; 3-phenylpropanoyl fentanyl)
Betaprodine 9611 I Y

Bezitramide 9800 II Y Burgodin


Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N
hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N

Brexanolone (3α-hydroxy-5α-pregnan-20-one) 2400 IV N Allopregnanolone


Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-
propylpyrrolidin-1-yl] butanamide)
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Brorphine (1-(1-(1-(4-bromophenyl)ethyl)piperidin-4-yl)- 9098 I Y 1-[1-[1-(4-bromophenyl)ethyl]-4-piperidinyl]-1,3-
1,3-dihydro-2H-benzo[d]imidazol-2-one) dihydro-2H-benzimidazol-2-one)
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Butonitazene (2-(2-(4-butoxybenzyl)-5-nitro-1H- 9751 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-
(methylamino)butan-1-one)

(Positional Isomers: dimethylone (bk-MDDMA;


MDDMC), N,N-dimethyl-3,4-
methylenedioxycathinone)
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-
(1-phenethylpiperidin-4-yl)-N-phenylbutanamide
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb
hydroxyandrost-4-en-3-one)
Camazepam 2749 IV N Albego, Limpidon, Paxor
Carfentanil 9743 II Y Wildnil
Carisoprodol 8192 IV N Soma

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 7 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine


Cathinone 1235 I N Constituent of "Khat" plant
Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2- 2720 V N 2H-tetrazole-2-ethanol, alpha-(2-chlorophenyl)-,
yl)ethyl]carbamate carbamate (ester), (alphaR)-; carbamic acid (R)-(+)-1-
(2-chlorophenyl)-2-(2H-tetrazol-2-yl)ethyl ester)
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clobazam 2751 IV N Urbadan, Urbanyl
Clonazepam 2737 IV N Klonopin, Clonopin
Clonitazene 9612 I Y

Clorazepate 2768 IV N Tranxene


Clortermine 1647 III N Voranil
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Coca Leaves 9040 II Y

Cocaine 9041 II Y Methyl benzoylecgonine, Crack


Codeine 9050 II Y Morphine methyl ester, methyl morphine
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Codeine methylbromide 9070 I Y

Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof


Codeine-N-oxide 9053 I Y

CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497


hydroxycyclohexy]-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue
[(1R,3S)3-hydroxycyclohexyl]-phenol)
Crotonyl fentanyl ((E)-N-(1-phenethylpiperidin-4-yl)-N- 9844 I Y
phenylbut-2-enamide)
Cyclopentyl fentanyl 9847 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopentanecarboxamide
Cyclopropyl Fentanyl 9845 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopropanecarboxamide
Cyprenorphine 9054 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 8 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Daridorexant [(S)-2-(5-chloro-4-methyl- 2410 IV N QUVIVIQ


1H benzo[d]imidazol-2-yl)-2-
methylpyrrolidin-1-yl](5-methoxy-2-
(2H-1,2,3-triazol-2-
yl)phenyl)methanone
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol
hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Delorazepam 2754 IV N

Delta1-dihydrotestosterone (17beta-hydroxy-5alpha- 4000 III N 1-Testosterone


androst-1-en-3-one)
Desomorphine 9055 I Y

Desoxymethyltestosterone 4000 III N

Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo


Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Diampromide 9615 I Y

Diazepam 2765 IV N Valium, Diastat


Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Diethylpropion 1610 IV N Tenuate, Tepanil
Diethylthiambutene 9616 I Y

Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine

(Positional Isomer: N-Methyl-N-isopropyltryptamine


(MiPT))
Difenoxin 9168 I Y Lyspafen
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine 9120 II Y Didrate, Parzone
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others
gm)
Dihydroetorphine 9334 II Y DHE
Dihydromorphine 9145 I Y

Dimenoxadol 9617 I Y

Dimepheptanol 9618 I Y

Dimethylthiambutene 9619 I Y

Dimethyltryptamine 7435 I N DMT


Dioxaphetyl butyrate 9621 I Y

Diphenoxylate 9170 II Y

Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen


Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 9 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as
capsule as approved by FDA approved by FDA
Dronabinol in an oral solution in a drug product 7365 II N Syndros
approved for marketing by the U.S. Food and Drug
Administration
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril
androstan-3-one)
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Eluxadoline 9725 IV N VIBERZI
Embutramide 2020 III N Tributane
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Estra-4,9,11-triene-3,17-dione 4000 III N

Ethchlorvynol 2540 IV N Placidyl


Ethinamate 2545 IV N Valmid, Valamin
Ethyl 2-(1-(5-fluoropentyl)-1H-indazole-3-carboxamido)- 7036 I N 5F-EDMB-PINACA
3,3-dimethylbutanoate
Ethyl loflazepate 2758 IV N

Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral


Ethylmethylthiambutene 9623 I Y

Ethylmorphine 9190 II Y Dionin


Ethylmorphine combination product 15 mg/du 9808 III Y

Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y

Ethylone 7547 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)propan-1-one;


3,4-methylenedioxy-N-ethylcathinone; bk-MDEA;
MDEC
Etodesnitazene; etazene (2-(2-(4-ethoxybenzyl)-1H- 9765 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Etonitazene 9624 I Y

Etorphine (except HCl) 9056 I Y

Etorphine HCl 9059 II Y M 99


Etoxeridine 9625 I Y

Eutylone 7549 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)butan-1-one,


bk-EBDB
Ezogabine 2779 V N Potiga
Fencamfamin 1760 IV N Reactivan
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Fenproporex 1575 IV N Gacilin, Solvolip
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Fentanyl carbamate (ethyl (1-phenethylpiperidin-4- 9851 I Y
yl)(phenyl)carbamate)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 10 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Fentanyl related-substances as defined in 21 CFR 9850 I Y


1308.11(h)
Fludiazepam 2759 IV N

Flunitazene (N,N-diethyl-2-(2-(4-fluorobenzyl)-5- nitro- 9756 I Y


1H-benzimidazol-1-yl)ethan-1-amine)
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl
11beta,17beta-dihydroxyandrost-4-en-3-one)
Flurazepam 2767 IV N Dalmane
Formebolone (2-formyl-17alpha-methyl-11alpha,17beta- 4000 III N Esiclene, Hubernol
dihydroxyandrost-1,4-dien-3-one)
Fospropofol 2138 IV N Lusedra
Furanyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9834 I Y
phenylfuran-2-carboxamide)
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu
hydroxyandrostano[2,3-c]-furazan)
Furethidine 9626 I Y

Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate


Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Ganaxolone (3α-hydroxy-3β-methyl-5α-pregnan-20-one) 2401 V N

Glutethimide 2550 II N Doriden, Dorimide


Halazepam 2762 IV N Paxipam
Haloxazolam 2771 IV N

Heroin 9200 I Y Diacetylmorphine, diamorphine


Hydrocodone 9193 II Y dihydrocodeinone
Hydromorphinol 9301 I Y

Hydromorphone 9150 II Y Dilaudid, dihydromorphinone


Hydroxypethidine 9627 I Y

Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant


Isobutyryl fentanyl 9827 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylisobutyramide
Isomethadone 9226 II Y Isoamidone
Isotonitazene (N,N-diethyl-2-(2-(4 isopropoxybenzyl)-5- 9614 I Y N,N-diethyl-2-[[4-(1-methylethoxy)phenyl]methyl]-5-
nitro-1H-benzimidazol-1-yl)ethan-1-amine) nitro-1H-benzimidazole-1-ethanamine
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678
naphthoyl)indole)
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl)indole) 7081 I N JWH-081
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl)indole) 7122 I N JWH-122
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200
naphthoyl)indole)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 11 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl)indole) 7203 I N JWH-203


JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl)indole) 6250 I N JWH-250
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl)indole) 7398 I N JWH-398
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Ketobemidone 9628 I Y Cliradon
Lacosamide 2746 V N Vimpat
Lasmiditan [2,4,6-trifluoro-N-(6-(1-methylpiperidine-4- 2790 V N Reyvow
carbonyl)pyridine-2-yl-benzamide]
Lemborexant 2245 IV N (1R,2S)-2-[(2,4-dimethylpyrimidin-5-yl)oxymethyl]-2-
(3-fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropane-
1-carboxamide
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Levomethorphan 9210 II Y

Levomoramide 9629 I Y

Levophenacylmorphan 9631 I Y

Levorphanol 9220 II Y Levo-Dromoran


Lisdexamfetamine 1205 II N Vyvanse
Loprazolam 2773 IV N

Lorazepam 2885 IV N Ativan


Lorcaserin 1625 IV N Belviq
Lormetazepam 2774 IV N Noctamid
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Lysergic acid diethylamide 7315 I N LSD, lysergide
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1-oxobutan- 7032 I N MAB-CHMINACA and ADB-CHMINACA
2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
Marihuana 7360 I N Cannabis, marijuana
Marihuana Extract 7350 I N

Mazindol 1605 IV N Sanorex, Mazanor


MDMB–CHMICA, MMB–CHMINACA (Methyl 2-(1- 7042 I N MDMB-CHMICA, MMB-CHMINACA
(cyclohexylmethyl)-1H-indole-3-carboxamido)-3,3-
dimethylbutanoate)
MDMB–FUBINACA (Methyl 2-(1-(4-fluorobenzyl)-1H- 7020 I N MDMB-FUBINACA
indazole-3-carboxamido)-3,3-dimethylbutanoate)
(Positional Isomer: EMB-FUBINACA)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 12 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV

(Positional Isomers: 1-(1,3-benzodioxol-5-yl)-2-


(cyclohexylamino)propan-1-one(n-cyclohexyl
methylone or 3,4-methylenedioxy-α-
cyclohexylaminopropiophenone) ; 1-(1,3-benzodioxol-
4-yl)-2-(pyrrolidin-1-yl)pentan-1-one (2,3-
methylenedioxy pyrovalerone)
Mebutamate 2800 IV N Capla
Mecloqualone 2572 I N Nubarene
Medazepam 2836 IV N Nobrium
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N 4-MMC

(Positional Isomers: 3-Methyl-methcathinone,


Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Mescaline 7381 I N Constituent of "Peyote" cacti
Mesocarb (N-phenyl-N'-(3-(1-phenylpropan-2-yl)-1,2,3- 1227 I N
oxadiazol-3-ium-5-yl)carbamimidate)
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Assimil, Ermalone, Methybol, Tantarone
androstan-3-one)
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Androviron, Proviron, Testiwop
androstan-3-one)
Metazocine 9240 II Y

Methadone 9250 II Y Dolophine, Methadose, Amidone


Methadone intermediate 9254 II Y Methadone precursor
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Methandienone (17alpha-methyl-17beta- 4000 III N Dianabol, Metabolina, Nerobol, Perbolin
hydroxyandrost-1,4-dien-3-one)
Methandriol (17alpha-methyl-3beta,17beta- 4000 III N Sinesex, Stenediol, Troformone
dihydroxyandrost-5-ene)
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Methasterone (2alpha,17alpha-dimethyl-5alpha- 4000 III N Methasterone; 2α,17α-dimethyl-17β-hydroxy-5α-
androstan-17beta-ol-3-one) androstan-3-one
Methcathinone 1237 I N N-Methylcathinone, "cat"
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst- 4000 III N Primobolan, Primobolan Depot, Primobolan S
1-en-3-one)
Methiopropamine (N-methyl-1-(thiophen-2-yl)propan-2- 1478 I N
amine)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 13 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Methohexital 2264 IV N Brevital


Methyl 2-(1-(4-fluorobenzyl)-1H-indazole-3- 7021 I N FUB–AMB, MMB– FUBINACA, AMB–FUBINACA
carboxamido)-3-methylbutanoate
Methyl 2-(1-(5-fluoropentyl)-1H-indole-3-carboxamido)- 7041 I N 5F-MDMB-PICA
3,3-dimethylbutanoate
(Positional Isomer: 5F-EMB-PICA or 5-fluoro-EMB-
PICA)
Methyldesorphine 9302 I Y

Methyldienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N


4,9(10)-dien-3-one)
Methyldihydromorphine 9304 I Y

Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N


(Positional Isomer: 2,3-
methylenedioxymethcathinone (2,3-MDMC, 1-
(benzo[d][1,3]dioxol-4-yl)-2-(methylamino)propan-1-
one))
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Methyltestosterone (17alpha-methyl-17beta- 4000 III N Android, Oreton, Testred, Virilon
hydroxyandrost-4-en-3-one)
Methyltrienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N Metribolone
4,9,11-trien-3-one)
Methyprylon 2575 III N Noludar
Metodesnitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)- 9764 I Y
1H-benzimidazol-1- yl)ethan-1-amine)
Metonitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)-5- 9757 I Y
nitro-1H-benzimidazol-1-yl)ethan-1-amine)
Metopon 9260 II Y

Mibolerone (7alpha,17alpha-dimethyl-17beta- 4000 III N Cheque, Matenon


hydroxyestr-4-en-3-one)
Midazolam 2884 IV N Versed
MMB-CHMICA, AMB-CHMICA (methyl 2-(1- 7044 I N
(cyclohexylmethyl)-1 H-indole-3-carboxamido)-3-
methylbutanoate)
Modafinil 1680 IV N Provigil
Moramide-intermediate 9802 II Y

Morpheridine 9632 I Y

Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR


Morphine combination product/50 mg/(100 ml or 100 9810 III Y
gm)
Morphine methylbromide 9305 I Y

Morphine methylsulfonate 9306 I Y

Morphine-N-oxide 9307 I Y

MT-45 (1-cyclohexyl-4-(1,2-diphenylethyl)piperazine)) 9560 I Y MT-45

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 14 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Myrophine 9308 I Y

N-(1-phenethylpiperidin-4-yl)-N-phenyltetrahydrofuran- 9843 I Y Tetrahydrofuranyl fentanyl


2-carboxamide
N-(2-fluorophenyl)-N-(1-phenethylpiperidin-4- 9816 I Y Ortho-fluorofentanyl or 2-fluorofentanyl
yl)propionamide
N-(Adamantan-1-yl)-1-(4-fluorobenzyl)-1H-indazole-3- 7047 I N FUB-AKB48; FUB-APINACA; AKB48 N-(4-
carboxamide FLUOROBENZYL)
N,N-Dimethylamphetamine 1480 I N

Nabilone 7379 II N Cesamet


Nalorphine 9400 III Y Nalline
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-
(pyrrolidin-1-yl)pentan-1-one)

(Positional Isomer: α-naphyrone)


N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Ethylamphetamine 1475 I N NEA
N-ethylhexedrone 7246 I N α-ethylaminohexanophenone; 2-(ethylamino)-1-
phenylhexan-1-one)
N-Ethylpentylone (1-(1,3-benzodioxol-5-yl)-2- 7543 I N Ephylone
(ethylamino)-pentan-1-one)
(Positional Isomers: 3,4-methylenedioxy-α-
propylaminobutiophenone; N,N-dimethylpentylone)
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
Nicocodeine 9309 I Y

Nicomorphine 9312 I Y Vilan


Nimetazepam 2837 IV N Erimin
Nitrazepam 2834 IV N Mogadon
NM2201; CBL2201 (Naphthalen-1-yl 1-(5-fluoropentyl)- 7221 I N
1 H-indole-3-carboxylate)
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
Noracymethadol 9633 I Y

Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol


hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar
en-3-one)
Norfentanyl (N-phenyl-N-(piperidin-4-yl)propionamide) 8366 II Y

Norlevorphanol 9634 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 15 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Normethadone 9635 I Y Phenyldimazone


Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron
hydroxyestr-4-en-3-one)
Normorphine 9313 I Y

Noroxymorphone 9668 II Y

Norpipanone 9636 I Y

N-pyrrolidino etonitazene; etonitazepyne 9758 I Y 2-(4-ethoxybenzyl)-5-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-


(2-(4-ethoxybenzyl)-5-nitro-1-(2- (pyrrolidin-1-yl)ethyl)- 1H-benzimidazole
1H-benzimidazole)
Ocfentanil 9838 I Y N-(2-fluorophenyl)-2-methoxy-N-(1-
phenethylpiperidin-4-yl)acetamide
Oliceridine (N-[(3-methoxythiophen-2-yl)methyl] ({2- 9245 II Y
[(9R)-9-(pyridin-2-yl)-6-oxaspiro [4.5]decan-9-
yl]ethyl{time} )amine fumarate)
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Opium extracts 9610 II Y

Opium fluid extract 9620 II Y

Opium poppy 9650 II Y Papaver somniferum


Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Opium tincture 9630 II Y Laudanum
Opium, granulated 9640 II Y Granulated opium
Opium, powdered 9639 II Y Powdered opium
Opium, raw 9600 II Y Raw opium, gum opium
Oripavine 9330 II Y

ortho-Fluoroacryl fentanyl (N-(2-fluorophenyl)-N-(1- 9852 I Y


phenethylpiperidin-4-yl)acrylamide)
ortho-Fluorobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9846 I Y
phenethylpiperidin-4-yl)butyramide; also known as 2-
fluorobutyryl fentanyl)
ortho-Fluoroisobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9853 I Y
phenethylpiperidin-4-yl)isobutyramide)
ortho-Methyl acetylfentanyl (N-(2-methylphenyl)-N-(1- 9848 I Y
phenethylpiperidin-4-yl)acetamide; also known as 2-
methyl acetylfentanyl)
ortho-Methyl methoxyacetyl fentanyl (2-methoxy-N-(2- 9820 I Y 2-methyl methoxyacetyl fentanyl
methylphenyl)-N-(1-phenethylpiperidin-4-yl)acetamide)
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome
5alpha-androstan-3-one)
Oxazepam 2835 IV N Serax, Serenid-D
Oxazolam 2839 IV N Serenal, Convertal
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10
dihydroxyandrost-4-en-3-one)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 16 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Oxymetholone (17alpha-methyl-2-hydroxymethylene- 4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd


17beta-hydroxy-5alpha-androstan-3-one)
Oxymorphone 9652 II Y Numorphan
Para-chloroisobutyryl fentanyl 9826 I Y N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-
yl)isobutyramide
Para-Fluoro furanyl fentanyl (N-(4-fluorophenyl)-N-(1- 9854 I Y
phenethylpiperidin-4-yl)furan-2-carboxamide)
Para-fluorobutyryl fentanyl 9823 I Y N-(4-fluorophenyl)-N-(1-phenethylpiperidin-4-
yl)butyramide
Para-Fluorofentanyl 9812 I Y China White, fentanyl
Parahexyl 7374 I N Synhexyl
Paraldehyde 2585 IV N Paral
Para-methoxybutyryl fentanyl 9837 I Y N-(4-methoxyphenyl)-N-(1-phenethylpiperidin-4-
yl)butyramide
Para-Methoxymethamphetamine (PMMA), 1-(4- 1245 I N
methoxyphenyl)-N-methylpropan-2-amine
Para-Methylfentanyl (N-(4-methylphenyl)-N-(1- 9817 I Y
phenethylpiperidin-4-yl)propionamide; also known as 4-
methylfentanyl)
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
Pemoline 1530 IV N Cylert
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC),


4-ethylmethcathinone (4-EMC), 4-methylbuphedrone
(4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone
(3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
Pentobarbital 2270 II N Nembutal
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-
(methylamino)pentan-1-one)

(Positional Isomers: dibutylone (bk-DMBDB) and


propylone (3',4'-methylenedioxy-N-
propylaminocathinone, 1-(benzo[d][1,3]dioxol-5-yl)-2-
(propylamino)propan-1-one))
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-
5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Peyote 7415 I N Cactus which contains mescaline
Phenadoxone 9637 I Y

Phenampromide 9638 I Y

Phenazocine 9715 II Y Narphen, Prinadol

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 17 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Phencyclidine 7471 II N PCP, Sernylan


Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Phenmetrazine 1631 II N Preludin
Phenobarbital 2285 IV N Luminal, Bellergal-S
Phenomorphan 9647 I Y

Phenoperidine 9641 I Y Operidine, Lealgin


Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9841 I Y
phenylbenzamide; also known as benzoyl fentanyl)
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Piminodine 9730 II Y

Pinazepam 2883 IV N Domar


Pipradrol 1750 IV N Detaril, Stimolag Fortis
Piritramide 9642 I Y Piridolan
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS
Prazepam 2764 IV N Centrax
Pregabalin 2782 V N Lyrica
Proheptazine 9643 I Y

Properidine 9644 I Y

Propiram 9649 I Y Algeril


Prostanozol (17beta-hydroxy-5alpha-androstano[3,2- 4000 III N Prostanozol; [3,2-c]pyrazole-5α-androstan-17β-ol
c]pyrazole)
Protonitazene (N,N-diethyl-2-(5-nitro-2-(4- 9759 I Y
propoxybenzyl)-1H-benzimidazol-1- yl)ethan-1-amine)
Psilocybin 7437 I N Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"

(Positional Isomers: 6-hydroxy DMT; 7-hydroxy DMT)


Pyrovalerone 1485 V N Centroton, Thymergix
Quazepam 2881 IV N Doral
Racemethorphan 9732 II Y

Racemoramide 9645 I Y

Racemorphan 9733 II Y Dromoran


Remifentanil 9739 II Y Ultiva
Remimazolam (4H-imidazol[1,2-a][1,4]benzodiazepine- 2846 IV N 8-bromo-1-methyl-6-(2-pyridinyl)-(4S)-methyl ester,
4-propionic acid) benzenesulfonate (1:1) and also, methyl 3-[(4S)-8-
bromo-1-methyl-6-pyridin-2-yl-4H-imidazo[1,2-
a][1,4]benzodiazepin-
4yl]propanoate benzenesulfonic acid

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 18 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Secobarbital 2315 II N Seconal, Tuinal


Secobarbital & noncontrolled active ingred 2316 III N

Secobarbital suppository dosage form 2316 III N

Serdexmethylphenidate 1729 IV N

Sibutramine 1675 IV N Meridia


Solriamfetol (2-amino-3-phenylpropyl car-bamate; 1650 IV N
benzenepropanol, beta-amino-, carbamate (ester))
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
SR-18 (1-Cyclohexylethyl-3-(2-methoxyphenylacetyl) 7008 I N SR-18 and RCS-8
indole)
SR-19 (1-Pentyl-3-[(4-methoxy)-benzoyl] indole 7104 I N SR-19 and RCS-4
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Winstrol, Winstrol-V
androst-2-eno[3,2-c]-pyrazole)
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst- 4000 III N
1-en-3-one)
Stimulant compounds previously excepted 1405 III N Mediatric
Sufentanil 9740 II Y Sufenta
Sulfondiethylmethane 2600 III N

Sulfonethylmethane 2605 III N

Sulfonmethane 2610 III N

Suvorexant 2223 IV N MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-


methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-
triazol-2-yl)phenyl]methanone
Talbutal 2100 III N Lotusate
Tapentadol 9780 II Y

Temazepam 2925 IV N Restoril


Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta- 4000 III N Teolit, Teslac
1,4-dien-17-oic acid lactone)
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and
others
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta- 4000 III N THG
hydroxygon-4,9,11-trien-3-one)
Tetrazepam 2886 IV N Myolastan, Musaril
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Thebaine 9333 II Y Precursor of many narcotics
Thiafentanil 9729 II Y Thianil
Thiamylal 2100 III N Surital
Thiofentanyl 9835 I Y Chine white, fentanyl
Thiofuranyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9839 I Y
phenylthiophene-2-carboxamide; also known as 2-
thiofuranyl fentanyl; thiophene fentanyl)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 19 of 20
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES

Thiopental 2100 III N Pentothal


THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3- 7024 I N THJ-2201
yl](naphthalen-1-yl)methanone
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol
methoxyphenyl)cyclohexanol)
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
Triazolam 2887 IV N Halcion
Trimeperidine 9646 I Y Promedolum
U-47700 (3,4-dichloro-N-[2-(dimethylamino)cyclohexyl]- 9547 I Y U-47700
N-methylbenzamide)
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- 7144 I N UR-144
tetramethylcyclopropyl)metanone
Valeryl fentanyl 9840 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylpentanamide
Vinbarbital 2100 III N Delvinal, vinbarbitone
Zaleplon 2781 IV N Sonata
Zipeprol (1-methoxy-3[-4-(2-methoxy-2- 9873 I Y
phenylethyl)piperazin-1-yl]-1-phenylpropan-2-ol)
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - Alphabetical Order


07-Jul-23 Page 20 of 20
Controlled Substances
DEA Drug Code Number
Controlled Substances
- by Controlled Substance Code Number -

CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others
gm)
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Lisdexamfetamine 1205 II N Vyvanse
Amineptine (7-[(10,11-dihydro-5H- 1219 I N
dibenzo[a,d]cyclohepten-5-yl)amino]heptanoic acid)
Mesocarb (N-phenyl-N'-(3-(1-phenylpropan-2-yl)-1,2,3- 1227 I N
oxadiazol-3-ium-5-yl)carbamimidate)
Benzphetamine 1228 III N Didrex, Inapetyl
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine
3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one)

(Positional Isomer: 2-FMC)


Cathinone 1235 I N Constituent of "Khat" plant
Methcathinone 1237 I N N-Methylcathinone, "cat"
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-
one)

(Positional Isomer: 2-FMC)


Para-Methoxymethamphetamine (PMMA), 1-(4- 1245 I N
methoxyphenyl)-N-methylpropan-2-amine
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC), 4-


ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-
MeMABP;4-MeBP), 3,4-dimethylmethcathinone (3,4-
DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N 4-MMC

(Positional Isomers: 3-Methyl-methcathinone,


Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 1 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC), 4-


ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-
MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-
DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-(pyrrolidin-1-
yl)pentan-1-one)

(Positional Isomer: α-naphyrone)


Stimulant compounds previously excepted 1405 III N Mediatric
N-Ethylamphetamine 1475 I N NEA
Methiopropamine (N-methyl-1-(thiophen-2-yl)propan-2- 1478 I N
amine)
N,N-Dimethylamphetamine 1480 I N
Pyrovalerone 1485 V N Centroton, Thymergix
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Pemoline 1530 IV N Cylert
Fenproporex 1575 IV N Gacilin, Solvolip
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Aminorex 1585 I N has been sold as methamphetamine
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4,4′-Dimethylaminorex (4,4′-DMAR; 4,5-dihydro-4- 1595 I N
methyl-5-(4-methylphenyl)-2-oxazolamine; 4-methyl-5-
(4-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine)
Mazindol 1605 IV N Sanorex, Mazanor
Diethylpropion 1610 IV N Tenuate, Tepanil
Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Lorcaserin 1625 IV N Belviq
Phenmetrazine 1631 II N Preludin
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clortermine 1647 III N Voranil
Solriamfetol (2-amino-3-phenylpropyl car-bamate; 1650 IV N
benzenepropanol, beta-amino-, carbamate (ester))
Sibutramine 1675 IV N Meridia
Modafinil 1680 IV N Provigil
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Serdexmethylphenidate 1729 IV N
Pipradrol 1750 IV N Detaril, Stimolag Fortis
Fencamfamin 1760 IV N Reactivan

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 2 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Embutramide 2020 III N Tributane
Aprobarbital 2100 III N Alurate
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Talbutal 2100 III N Lotusate
Thiamylal 2100 III N Surital
Thiopental 2100 III N Pentothal
Vinbarbital 2100 III N Delvinal, vinbarbitone
Amobarbital 2125 II N Amytal, Tuinal
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Fospropofol 2138 IV N Lusedra
Barbital 2145 IV N Veronal, Plexonal, barbitone
Suvorexant 2223 IV N MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-
1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-
yl)phenyl]methanone
Lemborexant 2245 IV N (1R,2S)-2-[(2,4-dimethylpyrimidin-5-yl)oxymethyl]-2-(3-
fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropane-1-
carboxamide
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-
5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Methohexital 2264 IV N Brevital
Pentobarbital 2270 II N Nembutal
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Phenobarbital 2285 IV N Luminal, Bellergal-S
Secobarbital 2315 II N Seconal, Tuinal
Secobarbital & noncontrolled active ingred 2316 III N
Secobarbital suppository dosage form 2316 III N
Brexanolone (3α-hydroxy-5α-pregnan-20-one) 2400 IV N Allopregnanolone
Ganaxolone (3α-hydroxy-3β-methyl-5α-pregnan-20-one) 2401 V N
Daridorexant [(S)-2-(5-chloro-4-methyl- 2410 IV N QUVIVIQ
1H benzo[d]imidazol-2-yl)-2-
methylpyrrolidin-1-yl](5-methoxy-2-
(2H-1,2,3-triazol-2-
yl)phenyl)methanone

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 3 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Glutethimide 2550 II N Doriden, Dorimide
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Mecloqualone 2572 I N Nubarene
Methyprylon 2575 III N Noludar
Paraldehyde 2585 IV N Paral
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Sulfondiethylmethane 2600 III N
Sulfonethylmethane 2605 III N
Sulfonmethane 2610 III N
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-
propylpyrrolidin-1-yl] butanamide)
Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2- 2720 V N 2H-tetrazole-2-ethanol, alpha-(2-chlorophenyl)-,
yl)ethyl]carbamate carbamate (ester), (alphaR)-; carbamic acid (R)-(+)-1-(2-
chlorophenyl)-2-(2H-tetrazol-2-yl)ethyl ester)
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Clonazepam 2737 IV N Klonopin, Clonopin
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Lacosamide 2746 V N Vimpat
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Camazepam 2749 IV N Albego, Limpidon, Paxor
Clobazam 2751 IV N Urbadan, Urbanyl
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Delorazepam 2754 IV N
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Ethyl loflazepate 2758 IV N
Fludiazepam 2759 IV N
Halazepam 2762 IV N Paxipam
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Prazepam 2764 IV N Centrax
Diazepam 2765 IV N Valium, Diastat
Flurazepam 2767 IV N Dalmane

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 4 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Clorazepate 2768 IV N Tranxene
Haloxazolam 2771 IV N
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Loprazolam 2773 IV N
Lormetazepam 2774 IV N Noctamid
Ezogabine 2779 V N Potiga
Zaleplon 2781 IV N Sonata
Pregabalin 2782 V N Lyrica
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta
Lasmiditan [2,4,6-trifluoro-N-(6-(1-methylpiperidine-4- 2790 V N Reyvow
carbonyl)pyridine-2-yl-benzamide]
Mebutamate 2800 IV N Capla
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Nitrazepam 2834 IV N Mogadon
Oxazepam 2835 IV N Serax, Serenid-D
Medazepam 2836 IV N Nobrium
Nimetazepam 2837 IV N Erimin
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Oxazolam 2839 IV N Serenal, Convertal
Remimazolam (4H-imidazol[1,2-a][1,4]benzodiazepine- 2846 IV N 8-bromo-1-methyl-6-(2-pyridinyl)-(4S)-methyl ester,
4-propionic acid) benzenesulfonate (1:1) and also, methyl 3-[(4S)-8-bromo-
1-methyl-6-pyridin-2-yl-4H-imidazo[1,2-
a][1,4]benzodiazepin-
4yl]propanoate benzenesulfonic acid
Quazepam 2881 IV N Doral
Alprazolam 2882 IV N Xanax
Pinazepam 2883 IV N Domar
Midazolam 2884 IV N Versed
Lorazepam 2885 IV N Ativan
Tetrazepam 2886 IV N Myolastan, Musaril
Triazolam 2887 IV N Halcion
Temazepam 2925 IV N Restoril
[3,2-c]-furazan-5α-androstan-17β-ol 4000 III N
[3,2-c]pyrazole-androst-4-en-17β-ol 4000 III N
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N
androstane

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 5 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N
4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone
hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
17α-Methyl-5α-androstan-17β-ol 4000 III N
17α-methyl-androst-2-ene-3,17β-diol 4000 III N
17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N
17α-Methyl-androstan-3-hydroxyimine-17β-ol 4000 III N
17β-Hydroxy-androstano[2,3-d]isoxazole 4000 III N
17β-Hydroxy-androstano[3,2-c]isoxazole 4000 III N
18a-Homo-3-hydroxy-estra-2,5(10)-dien-17-one 4000 III N
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N
androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-
androst-1-ene)
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
2α,17α-dimethyl-17β-hydroxy-5β-androstan-3-one 4000 III N
2α,3α-epithio-17α-methyl-5α-androstan-17β-ol 4000 III N
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
3β-hydroxy-estra-4,9,11-trien-17-one 4000 III N
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD
ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-chloro-17α-methyl-17β-hydroxy-androst-4-en-3-one 4000 III N
4-chloro-17α-methyl-17β-hydroxy-androst-4-ene-3,11- 4000 III N
dione
4-chloro-17α-methyl-androst-4-ene-3β,17β-diol 4000 III N
4-chloro-17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone
one)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N
4-en-3-one)
4-Hydroxy-androst-4-ene-3,17-dione 4000 III N Listed as 4-Hydroxy-androst-4-ene-3,17-dione[3,2-
c]pyrazole-5α-androstan-17β-ol

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 6 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N
en-3-one)
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N
ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
5α-Androstan-3,6,17-trione 4000 III N
6-bromo-androsta-1,4-diene-3,17-dione 4000 III N
6-bromo-androstan-3,17-dione 4000 III N
6α-Methyl-androst-4-ene-3,17-dione 4000 III N
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N
hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb
hydroxyandrost-4-en-3-one)
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol
hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha- 4000 III N 1-Testosterone
androst-1-en-3-one)
Desoxymethyltestosterone 4000 III N
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril
androstan-3-one)
Estra-4,9,11-triene-3,17-dione 4000 III N
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl
11beta,17beta-dihydroxyandrost-4-en-3-one)
Formebolone (2-formyl-17alpha-methyl-11alpha,17beta- 4000 III N Esiclene, Hubernol
dihydroxyandrost-1,4-dien-3-one)
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu
hydroxyandrostano[2,3-c]-furazan)
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Assimil, Ermalone, Methybol, Tantarone
androstan-3-one)
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Androviron, Proviron, Testiwop
androstan-3-one)
Methandienone (17alpha-methyl-17beta- 4000 III N Dianabol, Metabolina, Nerobol, Perbolin
hydroxyandrost-1,4-dien-3-one)
Methandriol (17alpha-methyl-3beta,17beta- 4000 III N Sinesex, Stenediol, Troformone
dihydroxyandrost-5-ene)
Methasterone (2alpha,17alpha-dimethyl-5alpha- 4000 III N Methasterone; 2α,17α-dimethyl-17β-hydroxy-5α-
androstan-17beta-ol-3-one) androstan-3-one
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst- 4000 III N Primobolan, Primobolan Depot, Primobolan S
1-en-3-one)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 7 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Methyldienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N
4,9(10)-dien-3-one)
Methyltestosterone (17alpha-methyl-17beta- 4000 III N Android, Oreton, Testred, Virilon
hydroxyandrost-4-en-3-one)
Methyltrienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N Metribolone
4,9,11-trien-3-one)
Mibolerone (7alpha,17alpha-dimethyl-17beta- 4000 III N Cheque, Matenon
hydroxyestr-4-en-3-one)
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol
hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar
en-3-one)
Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron
hydroxyestr-4-en-3-one)
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome
5alpha-androstan-3-one)
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10
dihydroxyandrost-4-en-3-one)
Oxymetholone (17alpha-methyl-2-hydroxymethylene- 4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd
17beta-hydroxy-5alpha-androstan-3-one)
Prostanozol (17beta-hydroxy-5alpha-androstano[3,2- 4000 III N Prostanozol; [3,2-c]pyrazole-5α-androstan-17β-ol
c]pyrazole)
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Winstrol, Winstrol-V
androst-2-eno[3,2-c]-pyrazole)
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst- 4000 III N
1-en-3-one)
Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta- 4000 III N Teolit, Teslac
1,4-dien-17-oic acid lactone)
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta- 4000 III N THG
hydroxygon-4,9,11-trien-3-one)
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl)indole) 6250 I N JWH-250
SR-18 (1-Cyclohexylethyl-3-(2-methoxyphenylacetyl) 7008 I N SR-18 and RCS-8
indole)
ADB–FUBINACA (N-(1-amino-3,3-dimethyl-1-oxobutan- 7010 I N ADB-FUBINACA
2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
5-Fluoro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Fluoro-UR-144, XLR-11 and XLR11
indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA
1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
(1-(4-Fluorobenzyl)-1H-indol-3-yl)(2,2,3,3- 7014 I N FUB-144
tetramethylcyclopropyl)methanone
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
MDMB–FUBINACA (Methyl 2-(1-(4-fluorobenzyl)-1H- 7020 I N MDMB-FUBINACA
indazole-3-carboxamido)-3,3-dimethylbutanoate)
(Positional Isomer: EMB-FUBINACA)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 8 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Methyl 2-(1-(4-fluorobenzyl)-1H-indazole-3- 7021 I N FUB–AMB, MMB– FUBINACA, AMB–FUBINACA
carboxamido)-3-methylbutanoate
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA
1-oxobutan-2-yl)-1-pentyl-1H-indazole-
3-carboxamide)
THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3- 7024 I N THJ-2201
yl](naphthalen-1-yl)methanone
5F-AB-PINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7025 I N
1-(5-fluoropentyl)-1 H-indazole-3-carboxamide)
AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA
oxobutan-2-yl)-1-(cyclohexylmethyl)-
1H-indazole-3-carboxamide
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1-oxobutan- 7032 I N MAB-CHMINACA and ADB-CHMINACA
2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
5F–AMB (Methyl 2-(1-(5-fluoropentyl)-1H-indazole-3- 7033 I N 5F-AMB
carboxamido)-3-methylbutanoate)
5F–ADB; 5F–MDMB–PINACA (Methyl 2-(1-(5- 7034 I N 5F-ADB, 5F-MDMB-PINACA, 5F-AEB, 5F-EMB-PINACA
fluoropentyl)-1H-indazole-3-carboxamido)-3,3-
dimethylbutanoate)
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA
yl)-1-pentyl-1H-indazole-3-carboxamide)
Ethyl 2-(1-(5-fluoropentyl)-1H-indazole-3-carboxamido)- 7036 I N 5F-EDMB-PINACA
3,3-dimethylbutanoate
Methyl 2-(1-(5-fluoropentyl)-1H-indole-3-carboxamido)- 7041 I N 5F-MDMB-PICA
3,3-dimethylbutanoate
(Positional Isomer: 5F-EMB-PICA or 5-fluoro-EMB-PICA)
MDMB–CHMICA, MMB–CHMINACA (Methyl 2-(1- 7042 I N MDMB-CHMICA, MMB-CHMINACA
(cyclohexylmethyl)-1H-indole-3-carboxamido)-3,3-
dimethylbutanoate)
4F-MDMB-BINACA (4F-MDMB-BUTINACA or methyl 2- 7043 I N
(1-(4-fluorobutyl)-1H-indazole-3-carboxamido)-3,3-
dimethylbutanoate)
MMB-CHMICA, AMB-CHMICA (methyl 2-(1- 7044 I N
(cyclohexylmethyl)-1 H-indole-3-carboxamido)-3-
methylbutanoate)
N-(Adamantan-1-yl)-1-(4-fluorobenzyl)-1H-indazole-3- 7047 I N FUB-AKB48; FUB-APINACA; AKB48 N-(4-
carboxamide FLUOROBENZYL)
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48
indazole-3-carboxamide
5F–APINACA, 5F–AKB48 (N-(adamantan-1-yl)-1-(5- 7049 I N 5F-APINACA, 5F-AKB48
fluoropentyl)-1H-indazole-3-carboxamide)
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl)indole) 7081 I N JWH-081
1-(5-Fluoropentyl)-N-(2-phenylpropan-2-yl)-1H-indazole- 7083 I N 5F-CUMYL-PINACA; SGT-25
3-carboxamide
5F-CUMYL-P7AICA (1-(5-fluoropentyl)-N-(2- 7085 I N
phenylpropan-2-yl)-1 H-pyrrolo[2,3-b]pyridine-3-
carboxamide)
4-CN-CUMYL-BUTINACA (1-(4-cyanobutyl)-N-(2- 7089 I N 4-cyano-CUMYL-BUTINACA; 4-CN-CUMYL BINACA;
phenylpropan-2-yl)-1 H-indazole-3-carboxamide) CUMYL-4CN-BINACA; SGT-78
SR-19 (1-Pentyl-3-[(4-methoxy)-benzoyl] indole 7104 I N SR-19 and RCS-4
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678
naphthoyl)indole)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 9 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl)indole) 7122 I N JWH-122
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- 7144 I N UR-144
tetramethylcyclopropyl)metanone
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200
naphthoyl)indole)
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl)indole) 7203 I N JWH-203
NM2201; CBL2201 (Naphthalen-1-yl 1-(5-fluoropentyl)- 7221 I N
1 H-indole-3-carboxylate)
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22
carboxylate)
4-methyl-alpha-ethylaminopentiophenone (4-MEAP) 7245 I N 4-MEAP; 2-(ethylamino)-1-(4-methylphenyl)pentan-1-one)
N-ethylhexedrone 7246 I N α-ethylaminohexanophenone; 2-(ethylamino)-1-
phenylhexan-1-one)
Alpha-ethyltryptamine 7249 I N ET, Trip
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
2-(ethylamino)-2-(3-methoxyphenyl)cyclohexan-1-one 7286 I N MXE, methoxetamine
(methoxetamine)
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497
hydroxycyclohexy]-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue
[(1R,3S)3-hydroxycyclohexyl]-phenol)
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Lysergic acid diethylamide 7315 I N LSD, lysergide
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7
7)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
Marihuana Extract 7350 I N
Marihuana 7360 I N Cannabis, marijuana
Dronabinol in an oral solution in a drug product 7365 II N Syndros
approved for marketing by the U.S. Food and Drug
Administration
Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as
capsule as approved by FDA approved by FDA
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and others
Parahexyl 7374 I N Synhexyl
Nabilone 7379 II N Cesamet
Mescaline 7381 I N Constituent of "Peyote" cacti

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 10 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C-T- 7385 I N 2C-T-2
2)
3,4,5-Trimethoxyamphetamine 7390 I N TMA

(Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-


5), 2,4,6-Trimethoxy-amphetamine (TMA-6), Escaline)
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl)indole) 7398 I N JWH-398
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET

(Positional Isomer: 1-(2,5-dimethoxy-4-


methylphenyl)butan-2-amine)
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA

(Positional Isomer: MDMB)


3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
4-Methoxyamphetamine 7411 I N PMA
Peyote 7415 I N Cactus which contains mescaline
5-Methoxy-N,N-dimethyltryptamine 7431 I N 5-MeO-DMT

(Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-


MeO-DMT))
Alpha-methyltryptamine 7432 I N AMT

(Positional Isomer: N-Methyltryptamine)


Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine

(Positional Isomer: N-Methyl-N-isopropyltryptamine


(MiPT))
Dimethyltryptamine 7435 I N DMT
Psilocybin 7437 I N Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"

(Positional Isomers: 6-hydroxy DMT; 7-hydroxy DMT)


5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT

(Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-


MeO-DPT))

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 11 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
4'-chloro-alpha-pyrrolidinovalerophenone (4-chloro-α- 7443 I N 4-chloro-α-PVP; 4'-chloro-α-pyrrolidinopentiophenone; 1-
PVP) (4-chlorophenyl)-2-(pyrrolidin-1-yl)pentan-1-one)
4´-methyl-alpha-pyrrolidinohexiophenone (MPHP) 7446 I N MPHP; 4'-methyl-alpha-pyrrolidinohexanophenone; 1-(4-
methylphenyl)-2-(pyrrolidin-1-yl)hexan-1-one)
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
Phencyclidine 7471 II N PCP, Sernylan
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-
methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E) 7509 I N 2C-E

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P
P)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4
(2C-T-4)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV

(Positional Isomers: 1-(1,3-benzodioxol-5-yl)-2-


(cyclohexylamino)propan-1-one(n-cyclohexyl methylone or
3,4-methylenedioxy-α-cyclohexylaminopropiophenone) ; 1-
(1,3-benzodioxol-4-yl)-2-(pyrrolidin-1-yl)pentan-1-one (2,3-
methylenedioxy pyrovalerone)
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36
ethanamine (25B-NBOMe)
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82
ethanamine (25C-NBOMe)
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5
ethanamine (25I-NBOMe)
Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N
(Positional Isomer: 2,3-methylenedioxymethcathinone
(2,3-MDMC, 1-(benzo[d][1,3]dioxol-4-yl)-2-
(methylamino)propan-1-one))

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 12 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-
1-one)

(Positional Isomers: dimethylone (bk-MDDMA; MDDMC),


N,N-dimethyl-3,4-methylenedioxycathinone)
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-
(methylamino)pentan-1-one)

(Positional Isomers: dibutylone (bk-DMBDB) and


propylone (3',4'-methylenedioxy-N-propylaminocathinone,
1-(benzo[d][1,3]dioxol-5-yl)-2-(propylamino)propan-1-one))
N-Ethylpentylone (1-(1,3-benzodioxol-5-yl)-2- 7543 I N Ephylone
(ethylamino)-pentan-1-one)
(Positional Isomers: 3,4-methylenedioxy-α-
propylaminobutiophenone; N,N-dimethylpentylone)
alpha-pyrrolidinohexanophenone (α-PHP) 7544 I N α-PHP; α-pyrrolidinohexanophenone; 1-phenyl-2-
(pyrrolidin-1-yl)hexan-1-one)
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-
yl)pentan-1-one)

(Positional Isomers: 4-methyl-α-pyrrolidinobutiophenone


(4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
Ethylone 7547 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)propan-1-one; 3,4-
methylenedioxy-N-ethylcathinone; bk-MDEA; MDEC
alpha-pyrrolidinoheptaphenone (PV8) 7548 I N PV8; 1-phenyl-2-(pyrrolidin-1-yl)heptan-1-one)
Eutylone 7549 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)butan-1-one, bk-
EBDB
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Carisoprodol 8192 IV N Soma
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP, Despropionyl fentanyl
Norfentanyl (N-phenyl-N-(piperidin-4-yl)propionamide) 8366 II Y
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
Alphaprodine 9010 II Y Nisentil
Anileridine 9020 II Y Leritine
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Acetyldihydrocodeine 9051 I Y Acetylcodone
Benzylmorphine 9052 I Y
Codeine-N-oxide 9053 I Y
Cyprenorphine 9054 I Y
Desomorphine 9055 I Y
Etorphine (except HCl) 9056 I Y
Etorphine HCl 9059 II Y M 99

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 13 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Codeine methylbromide 9070 I Y
Brorphine (1-(1-(1-(4-bromophenyl)ethyl)piperidin-4-yl)- 9098 I Y 1-[1-[1-(4-bromophenyl)ethyl]-4-piperidinyl]-1,3-dihydro-2H-
1,3-dihydro-2H-benzo[d]imidazol-2-one) benzimidazol-2-one)
Dihydrocodeine 9120 II Y Didrate, Parzone
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Dihydromorphine 9145 I Y
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Difenoxin 9168 I Y Lyspafen
Diphenoxylate 9170 II Y
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Ethylmorphine 9190 II Y Dionin
Hydrocodone 9193 II Y dihydrocodeinone
Heroin 9200 I Y Diacetylmorphine, diamorphine
Levomethorphan 9210 II Y
Levorphanol 9220 II Y Levo-Dromoran
Isomethadone 9226 II Y Isoamidone
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Metazocine 9240 II Y
Oliceridine (N-[(3-methoxythiophen-2-yl)methyl] ({2- 9245 II Y
[(9R)-9-(pyridin-2-yl)-6-oxaspiro [4.5]decan-9-
yl]ethyl{time} )amine fumarate)
Methadone 9250 II Y Dolophine, Methadose, Amidone
Methadone intermediate 9254 II Y Methadone precursor
Metopon 9260 II Y
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR
Hydromorphinol 9301 I Y
Methyldesorphine 9302 I Y
Methyldihydromorphine 9304 I Y
Morphine methylbromide 9305 I Y
Morphine methylsulfonate 9306 I Y
Morphine-N-oxide 9307 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 14 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Myrophine 9308 I Y
Nicocodeine 9309 I Y
Nicomorphine 9312 I Y Vilan
Normorphine 9313 I Y
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Acetorphine 9319 I Y
Oripavine 9330 II Y
Thebaine 9333 II Y Precursor of many narcotics
Dihydroetorphine 9334 II Y DHE
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Nalorphine 9400 III Y Nalline
U-47700 (3,4-dichloro-N-[2-(dimethylamino)cyclohexyl]- 9547 I Y U-47700
N-methylbenzamide)
AH-7921 (3,4-dichloro-N-[(1- 9551 I Y AH-7921
dimethylamino)cyclohexylmethyl]benzamide))
MT-45 (1-cyclohexyl-4-(1,2-diphenylethyl)piperazine)) 9560 I Y MT-45
Opium, raw 9600 II Y Raw opium, gum opium
Acetylmethadol 9601 I Y Methadyl acetate
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Benzethidine 9606 I Y
Betacetylmethadol 9607 I Y
Betameprodine 9608 I Y
Betamethadol 9609 I Y
Opium extracts 9610 II Y
Betaprodine 9611 I Y
Clonitazene 9612 I Y
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Isotonitazene (N,N-diethyl-2-(2-(4 isopropoxybenzyl)-5- 9614 I Y N,N-diethyl-2-[[4-(1-methylethoxy)phenyl]methyl]-5-nitro-
nitro-1H-benzimidazol-1-yl)ethan-1-amine) 1H-benzimidazole-1-ethanamine
Diampromide 9615 I Y
Diethylthiambutene 9616 I Y
Dimenoxadol 9617 I Y
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 15 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Opium fluid extract 9620 II Y
Dioxaphetyl butyrate 9621 I Y
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Ethylmethylthiambutene 9623 I Y
Etonitazene 9624 I Y
Etoxeridine 9625 I Y
Furethidine 9626 I Y
Hydroxypethidine 9627 I Y
Ketobemidone 9628 I Y Cliradon
Levomoramide 9629 I Y
Opium tincture 9630 II Y Laudanum
Levophenacylmorphan 9631 I Y
Morpheridine 9632 I Y
Noracymethadol 9633 I Y
Norlevorphanol 9634 I Y
Normethadone 9635 I Y Phenyldimazone
Norpipanone 9636 I Y
Phenadoxone 9637 I Y
Phenampromide 9638 I Y
Opium, powdered 9639 II Y Powdered opium
Opium, granulated 9640 II Y Granulated opium
Phenoperidine 9641 I Y Operidine, Lealgin
Piritramide 9642 I Y Piridolan
Proheptazine 9643 I Y
Properidine 9644 I Y
Racemoramide 9645 I Y
Trimeperidine 9646 I Y Promedolum
Phenomorphan 9647 I Y
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Propiram 9649 I Y Algeril
Opium poppy 9650 II Y Papaver somniferum
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Oxymorphone 9652 II Y Numorphan
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
Noroxymorphone 9668 II Y
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

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07-Jul-23 Page 16 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Phenazocine 9715 II Y Narphen, Prinadol
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Eluxadoline 9725 IV N VIBERZI
Thiafentanil 9729 II Y Thianil
Piminodine 9730 II Y
Racemethorphan 9732 II Y
Racemorphan 9733 II Y Dromoran
Alfentanil 9737 II Y Alfenta
Remifentanil 9739 II Y Ultiva
Sufentanil 9740 II Y Sufenta
Carfentanil 9743 II Y Wildnil
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Butonitazene (2-(2-(4-butoxybenzyl)-5-nitro-1H- 9751 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol
methoxyphenyl)cyclohexanol)
Flunitazene (N,N-diethyl-2-(2-(4-fluorobenzyl)-5- nitro- 9756 I Y
1H-benzimidazol-1-yl)ethan-1-amine)
Metonitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)-5- 9757 I Y
nitro-1H-benzimidazol-1-yl)ethan-1-amine)
N-pyrrolidino etonitazene; etonitazepyne 9758 I Y 2-(4-ethoxybenzyl)-5-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-
(2-(4-ethoxybenzyl)-5-nitro-1-(2- (pyrrolidin-1-yl)ethyl)- benzimidazole
1H-benzimidazole)
Protonitazene (N,N-diethyl-2-(5-nitro-2-(4- 9759 I Y
propoxybenzyl)-1H-benzimidazol-1- yl)ethan-1-amine)
Metodesnitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)- 9764 I Y
1H-benzimidazol-1- yl)ethan-1-amine)
Etodesnitazene; etazene (2-(2-(4-ethoxybenzyl)-1H- 9765 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Tapentadol 9780 II Y
Bezitramide 9800 II Y Burgodin
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Moramide-intermediate 9802 II Y
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Ethylmorphine combination product 15 mg/du 9808 III Y
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Morphine combination product/50 mg/(100 ml or 100 9810 III Y
gm)
Acryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9811 I Y Acryloylfentanyl
phenylacrylamide)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

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07-Jul-23 Page 17 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Para-Fluorofentanyl 9812 I Y China White, fentanyl
3-Methylfentanyl 9813 I Y China White, fentanyl
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Acetyl-alpha-methylfentanyl 9815 I Y
N-(2-fluorophenyl)-N-(1-phenethylpiperidin-4- 9816 I Y Ortho-fluorofentanyl or 2-fluorofentanyl
yl)propionamide
Para-Methylfentanyl (N-(4-methylphenyl)-N-(1- 9817 I Y
phenethylpiperidin-4-yl)propionamide; also known as 4-
methylfentanyl)
4'-Methyl acetyl fentanyl (N-(1-(4- 9819 I Y
methylphenethyl)piperidin-4-yl)-N-phenylacetamide)
ortho-Methyl methoxyacetyl fentanyl (2-methoxy-N-(2- 9820 I Y 2-methyl methoxyacetyl fentanyl
methylphenyl)-N-(1-phenethylpiperidin-4-yl)acetamide)
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y
phenylacetamide)
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-
phenethylpiperidin-4-yl)-N-phenylbutanamide
Para-fluorobutyryl fentanyl 9823 I Y N-(4-fluorophenyl)-N-(1-phenethylpiperidin-4-yl)butyramide
4-Fluoroisobutyryl fentanyl (N-(4-fluorophenyl)-N-(1- 9824 I Y Para-fluoroisobutyryl fentanyl
phenethylpiperidin-4-yl)isobutyramide)
2-methoxy-N-(1-phenethylpiperidin-4-yl)-N- 9825 I Y Methoxyacetyl fentanyl
phenylacetamide
Para-chloroisobutyryl fentanyl 9826 I Y N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-
yl)isobutyramide
Isobutyryl fentanyl 9827 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylisobutyramide
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
Furanyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9834 I Y
phenylfuran-2-carboxamide)
Thiofentanyl 9835 I Y Chine white, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-
phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-
piperidinyl]-N-phenylpropanamide
Para-methoxybutyryl fentanyl 9837 I Y N-(4-methoxyphenyl)-N-(1-phenethylpiperidin-4-
yl)butyramide
Ocfentanil 9838 I Y N-(2-fluorophenyl)-2-methoxy-N-(1-phenethylpiperidin-4-
yl)acetamide
Thiofuranyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9839 I Y
phenylthiophene-2-carboxamide; also known as 2-
thiofuranyl fentanyl; thiophene fentanyl)
Valeryl fentanyl 9840 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylpentanamide
Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9841 I Y
phenylbenzamide; also known as benzoyl fentanyl)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

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07-Jul-23 Page 18 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
beta'-Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N,3- 9842 I Y
diphenylpropanamide; also known as β'-phenyl
fentanyl; 3-phenylpropanoyl fentanyl)
N-(1-phenethylpiperidin-4-yl)-N-phenyltetrahydrofuran- 9843 I Y Tetrahydrofuranyl fentanyl
2-carboxamide
Crotonyl fentanyl ((E)-N-(1-phenethylpiperidin-4-yl)-N- 9844 I Y
phenylbut-2-enamide)
Cyclopropyl Fentanyl 9845 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopropanecarboxamide
ortho-Fluorobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9846 I Y
phenethylpiperidin-4-yl)butyramide; also known as 2-
fluorobutyryl fentanyl)
Cyclopentyl fentanyl 9847 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopentanecarboxamide
ortho-Methyl acetylfentanyl (N-(2-methylphenyl)-N-(1- 9848 I Y
phenethylpiperidin-4-yl)acetamide; also known as 2-
methyl acetylfentanyl)
Fentanyl related-substances as defined in 21 CFR 9850 I Y
1308.11(h)
Fentanyl carbamate (ethyl (1-phenethylpiperidin-4- 9851 I Y
yl)(phenyl)carbamate)
ortho-Fluoroacryl fentanyl (N-(2-fluorophenyl)-N-(1- 9852 I Y
phenethylpiperidin-4-yl)acrylamide)
ortho-Fluoroisobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9853 I Y
phenethylpiperidin-4-yl)isobutyramide)
Para-Fluoro furanyl fentanyl (N-(4-fluorophenyl)-N-(1- 9854 I Y
phenethylpiperidin-4-yl)furan-2-carboxamide)
2'-Fluoro ortho-fluorofentanyl (N-(1-(2- 9855 I Y
fluorophenethyl)piperidin-4-yl)-N-(2-
fluorophenyl)propionamide; also known as 2'-fluoro 2-
fluorofentanyl)
beta-Methyl fentanyl (N-phenyl-N-(1-(2- 9856 I Y
phenylpropyl)piperidin-4-yl)propionamide; also known
as β-methyl fentanyl)
Zipeprol (1-methoxy-3[-4-(2-methoxy-2- 9873 I Y
phenylethyl)piperazin-1-yl]-1-phenylpropan-2-ol)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by Controlled Substance Code Number


07-Jul-23 Page 19 of 19
Controlled Substances
CSA Schedule
Controlled Substances
- by CSA Schedule -

CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
(1-(4-Fluorobenzyl)-1H-indol-3-yl)(2,2,3,3- 7014 I N FUB-144
tetramethylcyclopropyl)methanone
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
1-(5-Fluoropentyl)-N-(2-phenylpropan-2-yl)-1H-indazole- 7083 I N 5F-CUMYL-PINACA; SGT-25
3-carboxamide
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P
P)
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E) 7509 I N 2C-E

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36
ethanamine (25B-NBOMe)
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82
ethanamine (25C-NBOMe)
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C-T- 7385 I N 2C-T-2
2)
2-(4-iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5
ethanamine (25I-NBOMe)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4
(2C-T-4)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
2-(ethylamino)-2-(3-methoxyphenyl)cyclohexan-1-one 7286 I N MXE, methoxetamine
(methoxetamine)
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7
7)
(Positional Isomer: 2,5-Dimethoxy-4-
ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET

(Positional Isomer: 1-(2,5-dimethoxy-4-


methylphenyl)butan-2-amine)
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 1 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
2'-Fluoro ortho-fluorofentanyl (N-(1-(2- 9855 I Y
fluorophenethyl)piperidin-4-yl)-N-(2-
fluorophenyl)propionamide; also known as 2'-fluoro 2-
fluorofentanyl)
2-methoxy-N-(1-phenethylpiperidin-4-yl)-N- 9825 I Y Methoxyacetyl fentanyl
phenylacetamide
3,4,5-Trimethoxyamphetamine 7390 I N TMA

(Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-


5), 2,4,6-Trimethoxy-amphetamine (TMA-6), Escaline)
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA

(Positional Isomer: MDMB)


3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one)

(Positional Isomer: 2-FMC)


3-Methylfentanyl 9813 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
4,4′-Dimethylaminorex (4,4′-DMAR; 4,5-dihydro-4- 1595 I N
methyl-5-(4-methylphenyl)-2-oxazolamine; 4-methyl-5-
(4-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine)
4´-methyl-alpha-pyrrolidinohexiophenone (MPHP) 7446 I N MPHP; 4'-methyl-alpha-pyrrolidinohexanophenone; 1-(4-
methylphenyl)-2-(pyrrolidin-1-yl)hexan-1-one)
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4'-chloro-alpha-pyrrolidinovalerophenone (4-chloro-α- 7443 I N 4-chloro-α-PVP; 4'-chloro-α-pyrrolidinopentiophenone; 1-
PVP) (4-chlorophenyl)-2-(pyrrolidin-1-yl)pentan-1-one)
4-CN-CUMYL-BUTINACA (1-(4-cyanobutyl)-N-(2- 7089 I N 4-cyano-CUMYL-BUTINACA; 4-CN-CUMYL BINACA;
phenylpropan-2-yl)-1 H-indazole-3-carboxamide) CUMYL-4CN-BINACA; SGT-78
4-Fluoroisobutyryl fentanyl (N-(4-fluorophenyl)-N-(1- 9824 I Y Para-fluoroisobutyryl fentanyl
phenethylpiperidin-4-yl)isobutyramide)
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-
one)

(Positional Isomer: 2-FMC)


4F-MDMB-BINACA (4F-MDMB-BUTINACA or methyl 2- 7043 I N
(1-(4-fluorobutyl)-1H-indazole-3-carboxamido)-3,3-
dimethylbutanoate)
4-Methoxyamphetamine 7411 I N PMA
4'-Methyl acetyl fentanyl (N-(1-(4- 9819 I Y
methylphenethyl)piperidin-4-yl)-N-phenylacetamide)
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP

(Positional Isomer: 2,5-Dimethoxy-3,4-


dimethylphenethylamine (2C-G))
4-methyl-alpha-ethylaminopentiophenone (4-MEAP) 7245 I N 4-MEAP; 2-(ethylamino)-1-(4-methylphenyl)pentan-1-one)
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-
methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

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07-Jul-23 Page 2 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC), 4-


ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-
MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-
DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
5F-AB-PINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7025 I N
1-(5-fluoropentyl)-1 H-indazole-3-carboxamide)
5F–ADB; 5F–MDMB–PINACA (Methyl 2-(1-(5- 7034 I N 5F-ADB, 5F-MDMB-PINACA, 5F-AEB, 5F-EMB-PINACA
fluoropentyl)-1H-indazole-3-carboxamido)-3,3-
dimethylbutanoate)
5F–AMB (Methyl 2-(1-(5-fluoropentyl)-1H-indazole-3- 7033 I N 5F-AMB
carboxamido)-3-methylbutanoate)
5F–APINACA, 5F–AKB48 (N-(adamantan-1-yl)-1-(5- 7049 I N 5F-APINACA, 5F-AKB48
fluoropentyl)-1H-indazole-3-carboxamide)
5F-CUMYL-P7AICA (1-(5-fluoropentyl)-N-(2- 7085 I N
phenylpropan-2-yl)-1 H-pyrrolo[2,3-b]pyridine-3-
carboxamide)
5-Fluoro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Fluoro-UR-144, XLR-11 and XLR11
indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22
carboxylate)
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT

(Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-


MeO-DPT))
5-Methoxy-N,N-dimethyltryptamine 7431 I N 5-MeO-DMT

(Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-


MeO-DMT))
AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA
oxobutan-2-yl)-1-(cyclohexylmethyl)-
1H-indazole-3-carboxamide
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA
1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA
1-oxobutan-2-yl)-1-pentyl-1H-indazole-
3-carboxamide)
Acetorphine 9319 I Y
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y
phenylacetamide)
Acetyl-alpha-methylfentanyl 9815 I Y
Acetyldihydrocodeine 9051 I Y Acetylcodone
Acetylmethadol 9601 I Y Methadyl acetate
Acryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9811 I Y Acryloylfentanyl
phenylacrylamide)
ADB–FUBINACA (N-(1-amino-3,3-dimethyl-1-oxobutan- 7010 I N ADB-FUBINACA
2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 3 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA
yl)-1-pentyl-1H-indazole-3-carboxamide)
AH-7921 (3,4-dichloro-N-[(1- 9551 I Y AH-7921
dimethylamino)cyclohexylmethyl]benzamide))
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Alpha-ethyltryptamine 7249 I N ET, Trip
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
Alpha-methyltryptamine 7432 I N AMT

(Positional Isomer: N-Methyltryptamine)


alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
alpha-pyrrolidinoheptaphenone (PV8) 7548 I N PV8; 1-phenyl-2-(pyrrolidin-1-yl)heptan-1-one)
alpha-pyrrolidinohexanophenone (α-PHP) 7544 I N α-PHP; α-pyrrolidinohexanophenone; 1-phenyl-2-
(pyrrolidin-1-yl)hexan-1-one)
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-
yl)pentan-1-one)

(Positional Isomers: 4-methyl-α-pyrrolidinobutiophenone


(4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Amineptine (7-[(10,11-dihydro-5H- 1219 I N
dibenzo[a,d]cyclohepten-5-yl)amino]heptanoic acid)
Aminorex 1585 I N has been sold as methamphetamine
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48
indazole-3-carboxamide
Benzethidine 9606 I Y
Benzylmorphine 9052 I Y
Betacetylmethadol 9607 I Y
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-
phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-
piperidinyl]-N-phenylpropanamide
Betameprodine 9608 I Y
Betamethadol 9609 I Y
beta-Methyl fentanyl (N-phenyl-N-(1-(2- 9856 I Y
phenylpropyl)piperidin-4-yl)propionamide; also known
as β-methyl fentanyl)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 4 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
beta'-Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N,3- 9842 I Y
diphenylpropanamide; also known as β'-phenyl
fentanyl; 3-phenylpropanoyl fentanyl)
Betaprodine 9611 I Y
Brorphine (1-(1-(1-(4-bromophenyl)ethyl)piperidin-4-yl)- 9098 I Y 1-[1-[1-(4-bromophenyl)ethyl]-4-piperidinyl]-1,3-dihydro-2H-
1,3-dihydro-2H-benzo[d]imidazol-2-one) benzimidazol-2-one)
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Butonitazene (2-(2-(4-butoxybenzyl)-5-nitro-1H- 9751 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-
1-one)

(Positional Isomers: dimethylone (bk-MDDMA; MDDMC),


N,N-dimethyl-3,4-methylenedioxycathinone)
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-
phenethylpiperidin-4-yl)-N-phenylbutanamide
Cathinone 1235 I N Constituent of "Khat" plant
Clonitazene 9612 I Y
Codeine methylbromide 9070 I Y
Codeine-N-oxide 9053 I Y
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497
hydroxycyclohexy]-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue
[(1R,3S)3-hydroxycyclohexyl]-phenol)
Crotonyl fentanyl ((E)-N-(1-phenethylpiperidin-4-yl)-N- 9844 I Y
phenylbut-2-enamide)
Cyclopentyl fentanyl 9847 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopentanecarboxamide
Cyclopropyl Fentanyl 9845 I Y N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopropanecarboxamide
Cyprenorphine 9054 I Y
Desomorphine 9055 I Y
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Diampromide 9615 I Y
Diethylthiambutene 9616 I Y
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine

(Positional Isomer: N-Methyl-N-isopropyltryptamine


(MiPT))
Difenoxin 9168 I Y Lyspafen
Dihydromorphine 9145 I Y
Dimenoxadol 9617 I Y
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y
Dimethyltryptamine 7435 I N DMT

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 5 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Dioxaphetyl butyrate 9621 I Y
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Ethyl 2-(1-(5-fluoropentyl)-1H-indazole-3-carboxamido)- 7036 I N 5F-EDMB-PINACA
3,3-dimethylbutanoate
Ethylmethylthiambutene 9623 I Y
Ethylone 7547 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)propan-1-one; 3,4-
methylenedioxy-N-ethylcathinone; bk-MDEA; MDEC
Etodesnitazene; etazene (2-(2-(4-ethoxybenzyl)-1H- 9765 I Y
benzimidazol-1-yl)-N,N-diethylethan-1-amine)
Etonitazene 9624 I Y
Etorphine (except HCl) 9056 I Y
Etoxeridine 9625 I Y
Eutylone 7549 I N 1-(1,3-benzodioxol-5-yl)-2-(ethylamino)butan-1-one, bk-
EBDB
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Fentanyl carbamate (ethyl (1-phenethylpiperidin-4- 9851 I Y
yl)(phenyl)carbamate)
Fentanyl related-substances as defined in 21 CFR 9850 I Y
1308.11(h)
Flunitazene (N,N-diethyl-2-(2-(4-fluorobenzyl)-5- nitro- 9756 I Y
1H-benzimidazol-1-yl)ethan-1-amine)
Furanyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9834 I Y
phenylfuran-2-carboxamide)
Furethidine 9626 I Y
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Heroin 9200 I Y Diacetylmorphine, diamorphine
Hydromorphinol 9301 I Y
Hydroxypethidine 9627 I Y
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
Isobutyryl fentanyl 9827 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylisobutyramide
Isotonitazene (N,N-diethyl-2-(2-(4 isopropoxybenzyl)-5- 9614 I Y N,N-diethyl-2-[[4-(1-methylethoxy)phenyl]methyl]-5-nitro-
nitro-1H-benzimidazol-1-yl)ethan-1-amine) 1H-benzimidazole-1-ethanamine
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678
naphthoyl)indole)
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl)indole) 7081 I N JWH-081
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl)indole) 7122 I N JWH-122
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200
naphthoyl)indole)
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl)indole) 7203 I N JWH-203
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl)indole) 6250 I N JWH-250

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 6 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl)indole) 7398 I N JWH-398
Ketobemidone 9628 I Y Cliradon
Levomoramide 9629 I Y
Levophenacylmorphan 9631 I Y
Lysergic acid diethylamide 7315 I N LSD, lysergide
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1-oxobutan- 7032 I N MAB-CHMINACA and ADB-CHMINACA
2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
Marihuana 7360 I N Cannabis, marijuana
Marihuana Extract 7350 I N
MDMB–CHMICA, MMB–CHMINACA (Methyl 2-(1- 7042 I N MDMB-CHMICA, MMB-CHMINACA
(cyclohexylmethyl)-1H-indole-3-carboxamido)-3,3-
dimethylbutanoate)
MDMB–FUBINACA (Methyl 2-(1-(4-fluorobenzyl)-1H- 7020 I N MDMB-FUBINACA
indazole-3-carboxamido)-3,3-dimethylbutanoate)
(Positional Isomer: EMB-FUBINACA)
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV

(Positional Isomers: 1-(1,3-benzodioxol-5-yl)-2-


(cyclohexylamino)propan-1-one(n-cyclohexyl methylone or
3,4-methylenedioxy-α-cyclohexylaminopropiophenone) ; 1-
(1,3-benzodioxol-4-yl)-2-(pyrrolidin-1-yl)pentan-1-one (2,3-
methylenedioxy pyrovalerone)
Mecloqualone 2572 I N Nubarene
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N 4-MMC

(Positional Isomers: 3-Methyl-methcathinone,


Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)
Mescaline 7381 I N Constituent of "Peyote" cacti
Mesocarb (N-phenyl-N'-(3-(1-phenylpropan-2-yl)-1,2,3- 1227 I N
oxadiazol-3-ium-5-yl)carbamimidate)
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Methcathinone 1237 I N N-Methylcathinone, "cat"
Methiopropamine (N-methyl-1-(thiophen-2-yl)propan-2- 1478 I N
amine)
Methyl 2-(1-(4-fluorobenzyl)-1H-indazole-3- 7021 I N FUB–AMB, MMB– FUBINACA, AMB–FUBINACA
carboxamido)-3-methylbutanoate
Methyl 2-(1-(5-fluoropentyl)-1H-indole-3-carboxamido)- 7041 I N 5F-MDMB-PICA
3,3-dimethylbutanoate
(Positional Isomer: 5F-EMB-PICA or 5-fluoro-EMB-PICA)
Methyldesorphine 9302 I Y
Methyldihydromorphine 9304 I Y
Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N
(Positional Isomer: 2,3-methylenedioxymethcathinone
(2,3-MDMC, 1-(benzo[d][1,3]dioxol-4-yl)-2-
(methylamino)propan-1-one))
Metodesnitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)- 9764 I Y
1H-benzimidazol-1- yl)ethan-1-amine)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 7 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Metonitazene (N,N-diethyl-2-(2-(4- methoxybenzyl)-5- 9757 I Y
nitro-1H-benzimidazol-1-yl)ethan-1-amine)
MMB-CHMICA, AMB-CHMICA (methyl 2-(1- 7044 I N
(cyclohexylmethyl)-1 H-indole-3-carboxamido)-3-
methylbutanoate)
Morpheridine 9632 I Y
Morphine methylbromide 9305 I Y
Morphine methylsulfonate 9306 I Y
Morphine-N-oxide 9307 I Y
MT-45 (1-cyclohexyl-4-(1,2-diphenylethyl)piperazine)) 9560 I Y MT-45
Myrophine 9308 I Y
N-(1-phenethylpiperidin-4-yl)-N-phenyltetrahydrofuran- 9843 I Y Tetrahydrofuranyl fentanyl
2-carboxamide
N-(2-fluorophenyl)-N-(1-phenethylpiperidin-4- 9816 I Y Ortho-fluorofentanyl or 2-fluorofentanyl
yl)propionamide
N-(Adamantan-1-yl)-1-(4-fluorobenzyl)-1H-indazole-3- 7047 I N FUB-AKB48; FUB-APINACA; AKB48 N-(4-
carboxamide FLUOROBENZYL)
N,N-Dimethylamphetamine 1480 I N
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-(pyrrolidin-1-
yl)pentan-1-one)

(Positional Isomer: α-naphyrone)


N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Ethylamphetamine 1475 I N NEA
N-ethylhexedrone 7246 I N α-ethylaminohexanophenone; 2-(ethylamino)-1-
phenylhexan-1-one)
N-Ethylpentylone (1-(1,3-benzodioxol-5-yl)-2- 7543 I N Ephylone
(ethylamino)-pentan-1-one)
(Positional Isomers: 3,4-methylenedioxy-α-
propylaminobutiophenone; N,N-dimethylpentylone)
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
Nicocodeine 9309 I Y
Nicomorphine 9312 I Y Vilan
NM2201; CBL2201 (Naphthalen-1-yl 1-(5-fluoropentyl)- 7221 I N
1 H-indole-3-carboxylate)
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
Noracymethadol 9633 I Y
Norlevorphanol 9634 I Y
Normethadone 9635 I Y Phenyldimazone
Normorphine 9313 I Y
Norpipanone 9636 I Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 8 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
N-pyrrolidino etonitazene; etonitazepyne 9758 I Y 2-(4-ethoxybenzyl)-5-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-
(2-(4-ethoxybenzyl)-5-nitro-1-(2- (pyrrolidin-1-yl)ethyl)- benzimidazole
1H-benzimidazole)
Ocfentanil 9838 I Y N-(2-fluorophenyl)-2-methoxy-N-(1-phenethylpiperidin-4-
yl)acetamide
ortho-Fluoroacryl fentanyl (N-(2-fluorophenyl)-N-(1- 9852 I Y
phenethylpiperidin-4-yl)acrylamide)
ortho-Fluorobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9846 I Y
phenethylpiperidin-4-yl)butyramide; also known as 2-
fluorobutyryl fentanyl)
ortho-Fluoroisobutyryl fentanyl (N-(2-fluorophenyl)-N-(1- 9853 I Y
phenethylpiperidin-4-yl)isobutyramide)
ortho-Methyl acetylfentanyl (N-(2-methylphenyl)-N-(1- 9848 I Y
phenethylpiperidin-4-yl)acetamide; also known as 2-
methyl acetylfentanyl)
ortho-Methyl methoxyacetyl fentanyl (2-methoxy-N-(2- 9820 I Y 2-methyl methoxyacetyl fentanyl
methylphenyl)-N-(1-phenethylpiperidin-4-yl)acetamide)
Para-chloroisobutyryl fentanyl 9826 I Y N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-
yl)isobutyramide
Para-Fluoro furanyl fentanyl (N-(4-fluorophenyl)-N-(1- 9854 I Y
phenethylpiperidin-4-yl)furan-2-carboxamide)
Para-fluorobutyryl fentanyl 9823 I Y N-(4-fluorophenyl)-N-(1-phenethylpiperidin-4-yl)butyramide
Para-Fluorofentanyl 9812 I Y China White, fentanyl
Parahexyl 7374 I N Synhexyl
Para-methoxybutyryl fentanyl 9837 I Y N-(4-methoxyphenyl)-N-(1-phenethylpiperidin-4-
yl)butyramide
Para-Methoxymethamphetamine (PMMA), 1-(4- 1245 I N
methoxyphenyl)-N-methylpropan-2-amine
Para-Methylfentanyl (N-(4-methylphenyl)-N-(1- 9817 I Y
phenethylpiperidin-4-yl)propionamide; also known as 4-
methylfentanyl)
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)

(Positional Isomers: 3-methylethcathinone (3-MEC), 4-


ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-
MeMABP;4-MeBP), 3,4-dimethylmethcathinone (3,4-
DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-
methylcathinone(EMC))
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-
(methylamino)pentan-1-one)

(Positional Isomers: dibutylone (bk-DMBDB) and


propylone (3',4'-methylenedioxy-N-propylaminocathinone,
1-(benzo[d][1,3]dioxol-5-yl)-2-(propylamino)propan-1-one))
Peyote 7415 I N Cactus which contains mescaline
Phenadoxone 9637 I Y
Phenampromide 9638 I Y
Phenomorphan 9647 I Y
Phenoperidine 9641 I Y Operidine, Lealgin

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 9 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Phenyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9841 I Y
phenylbenzamide; also known as benzoyl fentanyl)
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Piritramide 9642 I Y Piridolan
Proheptazine 9643 I Y
Properidine 9644 I Y
Propiram 9649 I Y Algeril
Protonitazene (N,N-diethyl-2-(5-nitro-2-(4- 9759 I Y
propoxybenzyl)-1H-benzimidazol-1- yl)ethan-1-amine)
Psilocybin 7437 I N Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"

(Positional Isomers: 6-hydroxy DMT; 7-hydroxy DMT)


Racemoramide 9645 I Y
SR-18 (1-Cyclohexylethyl-3-(2-methoxyphenylacetyl) 7008 I N SR-18 and RCS-8
indole)
SR-19 (1-Pentyl-3-[(4-methoxy)-benzoyl] indole 7104 I N SR-19 and RCS-4
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and others
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Thiofentanyl 9835 I Y Chine white, fentanyl
Thiofuranyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9839 I Y
phenylthiophene-2-carboxamide; also known as 2-
thiofuranyl fentanyl; thiophene fentanyl)
THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3- 7024 I N THJ-2201
yl](naphthalen-1-yl)methanone
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Trimeperidine 9646 I Y Promedolum
U-47700 (3,4-dichloro-N-[2-(dimethylamino)cyclohexyl]- 9547 I Y U-47700
N-methylbenzamide)
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- 7144 I N UR-144
tetramethylcyclopropyl)metanone
Valeryl fentanyl 9840 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylpentanamide
Zipeprol (1-methoxy-3[-4-(2-methoxy-2- 9873 I Y
phenylethyl)piperazin-1-yl]-1-phenylpropan-2-ol)
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP, Despropionyl fentanyl
Alfentanil 9737 II Y Alfenta
Alphaprodine 9010 II Y Nisentil
Amobarbital 2125 II N Amytal, Tuinal
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Anileridine 9020 II Y Leritine
Bezitramide 9800 II Y Burgodin

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 10 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Carfentanil 9743 II Y Wildnil
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Dihydrocodeine 9120 II Y Didrate, Parzone
Dihydroetorphine 9334 II Y DHE
Diphenoxylate 9170 II Y
Dronabinol in an oral solution in a drug product 7365 II N Syndros
approved for marketing by the U.S. Food and Drug
Administration
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Ethylmorphine 9190 II Y Dionin
Etorphine HCl 9059 II Y M 99
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Glutethimide 2550 II N Doriden, Dorimide
Hydrocodone 9193 II Y dihydrocodeinone
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Isomethadone 9226 II Y Isoamidone
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Levomethorphan 9210 II Y
Levorphanol 9220 II Y Levo-Dromoran
Lisdexamfetamine 1205 II N Vyvanse
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Metazocine 9240 II Y
Methadone 9250 II Y Dolophine, Methadose, Amidone
Methadone intermediate 9254 II Y Methadone precursor
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Metopon 9260 II Y
Moramide-intermediate 9802 II Y
Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR
Nabilone 7379 II N Cesamet
Norfentanyl (N-phenyl-N-(piperidin-4-yl)propionamide) 8366 II Y
Noroxymorphone 9668 II Y

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 11 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Oliceridine (N-[(3-methoxythiophen-2-yl)methyl] ({2- 9245 II Y
[(9R)-9-(pyridin-2-yl)-6-oxaspiro [4.5]decan-9-
yl]ethyl{time} )amine fumarate)
Opium extracts 9610 II Y
Opium fluid extract 9620 II Y
Opium poppy 9650 II Y Papaver somniferum
Opium tincture 9630 II Y Laudanum
Opium, granulated 9640 II Y Granulated opium
Opium, powdered 9639 II Y Powdered opium
Opium, raw 9600 II Y Raw opium, gum opium
Oripavine 9330 II Y
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Oxymorphone 9652 II Y Numorphan
Pentobarbital 2270 II N Nembutal
Phenazocine 9715 II Y Narphen, Prinadol
Phencyclidine 7471 II N PCP, Sernylan
Phenmetrazine 1631 II N Preludin
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
Piminodine 9730 II Y
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS
Racemethorphan 9732 II Y
Racemorphan 9733 II Y Dromoran
Remifentanil 9739 II Y Ultiva
Secobarbital 2315 II N Seconal, Tuinal
Sufentanil 9740 II Y Sufenta
Tapentadol 9780 II Y
Thebaine 9333 II Y Precursor of many narcotics
Thiafentanil 9729 II Y Thianil
[3,2-c]-furazan-5α-androstan-17β-ol 4000 III N
[3,2-c]pyrazole-androst-4-en-17β-ol 4000 III N
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N
4-hydroxy-17beta-hydroxyestr-4-en-3-one)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 12 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone
hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
17α-Methyl-5α-androstan-17β-ol 4000 III N
17α-methyl-androst-2-ene-3,17β-diol 4000 III N
17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N
17α-Methyl-androstan-3-hydroxyimine-17β-ol 4000 III N
17β-Hydroxy-androstano[2,3-d]isoxazole 4000 III N
17β-Hydroxy-androstano[3,2-c]isoxazole 4000 III N
18a-Homo-3-hydroxy-estra-2,5(10)-dien-17-one 4000 III N
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N
androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-
androst-1-ene)
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
2α,17α-dimethyl-17β-hydroxy-5β-androstan-3-one 4000 III N
2α,3α-epithio-17α-methyl-5α-androstan-17β-ol 4000 III N
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
3β-hydroxy-estra-4,9,11-trien-17-one 4000 III N
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD
ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-chloro-17α-methyl-17β-hydroxy-androst-4-en-3-one 4000 III N
4-chloro-17α-methyl-17β-hydroxy-androst-4-ene-3,11- 4000 III N
dione
4-chloro-17α-methyl-androst-4-ene-3β,17β-diol 4000 III N
4-chloro-17α-methyl-androsta-1,4-diene-3,17β-diol 4000 III N
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone
one)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N
4-en-3-one)
4-Hydroxy-androst-4-ene-3,17-dione 4000 III N Listed as 4-Hydroxy-androst-4-ene-3,17-dione[3,2-
c]pyrazole-5α-androstan-17β-ol
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N
en-3-one)
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N
ene)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 13 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
5α-Androstan-3,6,17-trione 4000 III N
6-bromo-androsta-1,4-diene-3,17-dione 4000 III N
6-bromo-androstan-3,17-dione 4000 III N
6α-Methyl-androst-4-ene-3,17-dione 4000 III N
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Aprobarbital 2100 III N Alurate
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Benzphetamine 1228 III N Didrex, Inapetyl
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N
hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb
hydroxyandrost-4-en-3-one)
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clortermine 1647 III N Voranil
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol
hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha- 4000 III N 1-Testosterone
androst-1-en-3-one)
Desoxymethyltestosterone 4000 III N
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as
capsule as approved by FDA approved by FDA
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril
androstan-3-one)
Embutramide 2020 III N Tributane
Estra-4,9,11-triene-3,17-dione 4000 III N

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 14 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Ethylmorphine combination product 15 mg/du 9808 III Y
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl
11beta,17beta-dihydroxyandrost-4-en-3-one)
Formebolone (2-formyl-17alpha-methyl-11alpha,17beta- 4000 III N Esiclene, Hubernol
dihydroxyandrost-1,4-dien-3-one)
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu
hydroxyandrostano[2,3-c]-furazan)
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Assimil, Ermalone, Methybol, Tantarone
androstan-3-one)
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Androviron, Proviron, Testiwop
androstan-3-one)
Methandienone (17alpha-methyl-17beta- 4000 III N Dianabol, Metabolina, Nerobol, Perbolin
hydroxyandrost-1,4-dien-3-one)
Methandriol (17alpha-methyl-3beta,17beta- 4000 III N Sinesex, Stenediol, Troformone
dihydroxyandrost-5-ene)
Methasterone (2alpha,17alpha-dimethyl-5alpha- 4000 III N Methasterone; 2α,17α-dimethyl-17β-hydroxy-5α-
androstan-17beta-ol-3-one) androstan-3-one
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst- 4000 III N Primobolan, Primobolan Depot, Primobolan S
1-en-3-one)
Methyldienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N
4,9(10)-dien-3-one)
Methyltestosterone (17alpha-methyl-17beta- 4000 III N Android, Oreton, Testred, Virilon
hydroxyandrost-4-en-3-one)
Methyltrienolone (17alpha-methyl-17beta-hydroxyestra- 4000 III N Metribolone
4,9,11-trien-3-one)
Methyprylon 2575 III N Noludar
Mibolerone (7alpha,17alpha-dimethyl-17beta- 4000 III N Cheque, Matenon
hydroxyestr-4-en-3-one)
Morphine combination product/50 mg/(100 ml or 100 9810 III Y
gm)
Nalorphine 9400 III Y Nalline
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol
hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar
en-3-one)
Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron
hydroxyestr-4-en-3-one)
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome
5alpha-androstan-3-one)

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 15 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10
dihydroxyandrost-4-en-3-one)
Oxymetholone (17alpha-methyl-2-hydroxymethylene- 4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd
17beta-hydroxy-5alpha-androstan-3-one)
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-
5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Prostanozol (17beta-hydroxy-5alpha-androstano[3,2- 4000 III N Prostanozol; [3,2-c]pyrazole-5α-androstan-17β-ol
c]pyrazole)
Secobarbital & noncontrolled active ingred 2316 III N
Secobarbital suppository dosage form 2316 III N
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Winstrol, Winstrol-V
androst-2-eno[3,2-c]-pyrazole)
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst- 4000 III N
1-en-3-one)
Stimulant compounds previously excepted 1405 III N Mediatric
Sulfondiethylmethane 2600 III N
Sulfonethylmethane 2605 III N
Sulfonmethane 2610 III N
Talbutal 2100 III N Lotusate
Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta- 4000 III N Teolit, Teslac
1,4-dien-17-oic acid lactone)
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta- 4000 III N THG
hydroxygon-4,9,11-trien-3-one)
Thiamylal 2100 III N Surital
Thiopental 2100 III N Pentothal
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
Vinbarbital 2100 III N Delvinal, vinbarbitone
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Alprazolam 2882 IV N Xanax
Barbital 2145 IV N Veronal, Plexonal, barbitone
Brexanolone (3α-hydroxy-5α-pregnan-20-one) 2400 IV N Allopregnanolone
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Camazepam 2749 IV N Albego, Limpidon, Paxor
Carisoprodol 8192 IV N Soma
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 16 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Clobazam 2751 IV N Urbadan, Urbanyl
Clonazepam 2737 IV N Klonopin, Clonopin
Clorazepate 2768 IV N Tranxene
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Daridorexant [(S)-2-(5-chloro-4-methyl- 2410 IV N QUVIVIQ
1H benzo[d]imidazol-2-yl)-2-
methylpyrrolidin-1-yl](5-methoxy-2-
(2H-1,2,3-triazol-2-
yl)phenyl)methanone
Delorazepam 2754 IV N
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Diazepam 2765 IV N Valium, Diastat
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Diethylpropion 1610 IV N Tenuate, Tepanil
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Eluxadoline 9725 IV N VIBERZI
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Ethyl loflazepate 2758 IV N
Fencamfamin 1760 IV N Reactivan
Fenproporex 1575 IV N Gacilin, Solvolip
Fludiazepam 2759 IV N
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Flurazepam 2767 IV N Dalmane
Fospropofol 2138 IV N Lusedra
Halazepam 2762 IV N Paxipam
Haloxazolam 2771 IV N
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Lemborexant 2245 IV N (1R,2S)-2-[(2,4-dimethylpyrimidin-5-yl)oxymethyl]-2-(3-
fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropane-1-
carboxamide
Loprazolam 2773 IV N
Lorazepam 2885 IV N Ativan
Lorcaserin 1625 IV N Belviq

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 17 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Lormetazepam 2774 IV N Noctamid
Mazindol 1605 IV N Sanorex, Mazanor
Mebutamate 2800 IV N Capla
Medazepam 2836 IV N Nobrium
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Methohexital 2264 IV N Brevital
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Midazolam 2884 IV N Versed
Modafinil 1680 IV N Provigil
Nimetazepam 2837 IV N Erimin
Nitrazepam 2834 IV N Mogadon
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Oxazepam 2835 IV N Serax, Serenid-D
Oxazolam 2839 IV N Serenal, Convertal
Paraldehyde 2585 IV N Paral
Pemoline 1530 IV N Cylert
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Phenobarbital 2285 IV N Luminal, Bellergal-S
Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Pinazepam 2883 IV N Domar
Pipradrol 1750 IV N Detaril, Stimolag Fortis
Prazepam 2764 IV N Centrax
Quazepam 2881 IV N Doral
Remimazolam (4H-imidazol[1,2-a][1,4]benzodiazepine- 2846 IV N 8-bromo-1-methyl-6-(2-pyridinyl)-(4S)-methyl ester,
4-propionic acid) benzenesulfonate (1:1) and also, methyl 3-[(4S)-8-bromo-
1-methyl-6-pyridin-2-yl-4H-imidazo[1,2-
a][1,4]benzodiazepin-
4yl]propanoate benzenesulfonic acid
Serdexmethylphenidate 1729 IV N
Sibutramine 1675 IV N Meridia
Solriamfetol (2-amino-3-phenylpropyl car-bamate; 1650 IV N
benzenepropanol, beta-amino-, carbamate (ester))
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
Suvorexant 2223 IV N MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-
1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-
yl)phenyl]methanone
Temazepam 2925 IV N Restoril
Tetrazepam 2886 IV N Myolastan, Musaril

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 18 of 19
CSA
SUBSTANCE CSCN SCH NARC OTHER NAMES
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol
methoxyphenyl)cyclohexanol)
Triazolam 2887 IV N Halcion
Zaleplon 2781 IV N Sonata
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-
propylpyrrolidin-1-yl] butanamide)
Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2- 2720 V N 2H-tetrazole-2-ethanol, alpha-(2-chlorophenyl)-,
yl)ethyl]carbamate carbamate (ester), (alphaR)-; carbamic acid (R)-(+)-1-(2-
chlorophenyl)-2-(2H-tetrazol-2-yl)ethyl ester)
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others
gm)
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Ezogabine 2779 V N Potiga
Ganaxolone (3α-hydroxy-3β-methyl-5α-pregnan-20-one) 2401 V N
Lacosamide 2746 V N Vimpat
Lasmiditan [2,4,6-trifluoro-N-(6-(1-methylpiperidine-4- 2790 V N Reyvow
carbonyl)pyridine-2-yl-benzamide]
Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Pregabalin 2782 V N Lyrica
Pyrovalerone 1485 V N Centroton, Thymergix

Abbreviations: "NARC" = Narcotic, "CSA SCH" = CSA Schedule, "CSCN" = Controlled Substance Code Number

Controlled Substances - by CSA Schedule


07-Jul-23 Page 19 of 19
List I and List II Regulated Chemicals
1. Alphabetical Order
2. DEA Number
3. List Number
4. Illicit Uses and Threshold Quantities
List I and II Regulated Chemicals
- Alphabetical Order -

DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE

1-BOC-4-AP (tert-butyl 4-(phenylamino)piperidine-1-carboxylate) and its salts I 8336 87 FR 67550 11/9/2022


4-ANILINOPIPERIDINE (N-phenylpiperidin-4-amine; N phenyl-4- I 8335 85 FR 20822 5/15/2020
piperidinamine; 4–AP) including its amides,its carbamates, and its salts
4-PIPERIDONE (piperidin-4-one) including its acetals, its amides, its I 8330 88 FR 21902 5/12/2023
carbamates, its salts, and salts of its acetals, its amides, and its carbamates,
and any combination thereof, whenever the existence of such is possible
ACETIC ANHYDRIDE II 8519 Pub. L. 100-690 3/18/1989
ACETONE II 6532 Pub. L. 100-690 3/18/1989
N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690 3/18/1989
ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690 3/18/1989
APAA (Alpha-phenylacetoacetamide) and its optical isomers (Effective I 8515 86 FR 24703 6/9/2021
06/09/2021)
APAAN (Alpha-phenylacetoacetoniltrile), salts, optical isomers, salts of I 8512 82 FR 32457 8/14/2017
optical isomers
BENZALDEHYDE I 8256 Pub. L. 103-200 4/17/1994
BENZYL CHLORIDE II 8570 Pub. L. 100-690 3/18/1989
BENZYL CYANIDE I 8735 Pub. L. 100-690 3/18/1989
BENZYLFENTANYL (N-(1-benzylpiperidin-4-yl)-N-phenylpropionamide), I 8334 85 FR 20822 5/15/2020
including its salts.
gamma-BUTYROLACTONE I 2011 Pub. L. 106-172 2/18/2000
EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690 3/18/1989
EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200 4/17/1994
EPHEDRINE-remove exemption for OTC combination products and establish I 8113 Pub. L. 104-237 10/3/1996
a 24 g retail threshold. Threshold remains zero for single entity products.
Mail order report requirements imposed. For more info, see 21 CFR Parts
1309, 1310, 1313
ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690 3/18/1989
ERGOCRISTINE I 8612 76 FR 17778 5/2/2011
ERGOTAMINE & salts I 8676 Pub. L. 100-690 3/18/1989
ETHYLAMINE & salts I 8678 Pub. L. 101-647 2/27/1991
N-ETHYLEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991
N-ETHYLEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
ETHYL ETHER II 6584 Pub. L. 100-690 3/18/1989
N-ETHYLPSEUDOEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991
N-ETHYLPSEUDOEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992
HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237 10/3/1996

* Remain in Schedule III


List I and II Regulated Chemicals - Alphabetical Order
07-Jul-23 Page 1 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690 3/18/1989
HYDRIODIC ACID I 6695 Pub. L. 101-647 2/27/1991
HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, I 6797 66 FR 52670 11/16/2001
calcium hypophosphite, iron hypophosphite, potassium hypophosphite,
manganese hypophosphite, magnesium hypophosphite, and sodium
hypophosphite)
IODINE - superseded by 2007 action II 6699 Pub. L. 104-237 10/3/1996
IODINE I 6699 72 FR 35920 8/1/2007
ISOSAFROLE I 8704 Pub. L. 101-647 2/27/1991
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers- I 7300 Pub. L. 101-647 2/27/1991
superseded
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers* REMOVED 7300 Pub. L. 103-200 4/17/1994
METHYLAMINE and salts I 8520 Pub. L. 101-647 2/27/1991
METHYL ALPHA-PHENYLACETOACETATE (MAPA) I 8795 86 FR 64362 12/20/2021
3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690 3/18/1989
N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647 2/27/1991
METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690 3/18/1989
METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995
N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical I 8119 Pub. L. 101-647 2/27/1991
isomers
NITROETHANE I 6724 Pub. L. 103-200 4/17/1994
NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690 3/18/1989
N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007
PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE-remove exemption for certain OTC I 1225 Pub. L. 104-237 10/3/1997
transactions. Retail threshold of 24 g established for products not distributed
in blister packs. Mail order report requirements imposed. For more info, see
21 CFR Parts 1309, 1310, and 1313.
PIPERIDINE and salts I 2704 Pub. L. 100-690 3/18/1989
PIPERONAL I 8750 Pub. L. 101-647 2/27/1991
PMK GLYCIDATE (3,4-MDP-2-P METHYL GLYCIDATE) and its optical and I 8535 86 FR 24703 6/9/2021
geometric isomers (Effective 06/09/2021)
PMK GLYCIDIC ACID (3,4-MDP-2-P METHYL GLYCIDIC ACID) and its I 8525 86 FR 24703 6/9/2021
salts, optical and geometric isomers, and salts of isomers (Effective
06/09/2021)
POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690 3/18/1989
PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647 2/27/1991
PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100-690 3/18/1989
PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. I 8112 Pub. L. 104-237 10/3/1997
Retail threshold of 24 g established for products not distributed in blister
packs. Mail order report requirements imposed. For more info, see 21 CFR
Parts 1309, 1310, and 1313.
RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001
SAFROLE (includes sassafras oil) I 8323 Pub. L. 101-647 2/27/1991

* Remain in Schedule III


List I and II Regulated Chemicals - Alphabetical Order
07-Jul-23 Page 2 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006
SULFURIC ACID II 6552 57 FR 43614 10/22/1992
TOLUENE II 6594 Pub. L. 100-690 3/18/1989
WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001

* Remain in Schedule III


List I and II Regulated Chemicals - Alphabetical Order
07-Jul-23 Page 3 of 3
List I and II Regulated Chemicals
- by DEA Chemical Code Number -
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE

N-ETHYLEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991


N-ETHYLEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
N-ETHYLPSEUDOEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991
N-ETHYLPSEUDOEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE-remove exemption for certain OTC transactions. I 1225 Pub. L. 104-237 10/3/1997
Retail threshold of 24 g established for products not distributed in blister
packs. Mail order report requirements imposed. For more info, see 21 CFR
Parts 1309, 1310, and 1313.
gamma-BUTYROLACTONE I 2011 Pub. L. 106-172 2/18/2000
PIPERIDINE and salts I 2704 Pub. L. 100-690 3/18/1989
ACETONE II 6532 Pub. L. 100-690 3/18/1989
HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992
HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237 10/3/1996
SULFURIC ACID II 6552 57 FR 43614 10/22/1992
POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690 3/18/1989
ETHYL ETHER II 6584 Pub. L. 100-690 3/18/1989
SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006
TOLUENE II 6594 Pub. L. 100-690 3/18/1989
HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690 3/18/1989
HYDRIODIC ACID I 6695 Pub. L. 101-647 2/27/1991
IODINE - superseded by 2007 action II 6699 Pub. L. 104-237 10/3/1996
IODINE I 6699 72 FR 35920 8/1/2007
METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690 3/18/1989
METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995
NITROETHANE I 6724 Pub. L. 103-200 4/17/1994
RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001
WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001
HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, I 6797 66 FR 52670 11/16/2001
calcium hypophosphite, iron hypophosphite, potassium hypophosphite,
manganese hypophosphite, magnesium hypophosphite, and sodium
hypophosphite)
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers- I 7300 Pub. L. 101-647 2/27/1991
superseded
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers* REMOVED 7300 Pub. L. 103-200 4/17/1994
PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100-690 3/18/1989

* Remain in Schedule III


List I and II Regulated Chemicals - by DEA Chemical Code Number
07-Jul-23 Page 1 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. I 8112 Pub. L. 104-237 10/3/1997
Retail threshold of 24 g established for products not distributed in blister
packs. Mail order report requirements imposed. For more info, see 21 CFR
Parts 1309, 1310, and 1313.
EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690 3/18/1989
EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200 4/17/1994
EPHEDRINE-remove exemption for OTC combination products and establish I 8113 Pub. L. 104-237 10/3/1996
a 24 g retail threshold. Threshold remains zero for single entity products. Mail
order report requirements imposed. For more info, see 21 CFR Parts 1309,
1310, 1313
N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647 2/27/1991
N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical I 8119 Pub. L. 101-647 2/27/1991
isomers
BENZALDEHYDE I 8256 Pub. L. 103-200 4/17/1994
NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690 3/18/1989
SAFROLE (includes sassafras oil) I 8323 Pub. L. 101-647 2/27/1991
PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647 2/27/1991
4-PIPERIDONE (piperidin-4-one) including its acetals, its amides, its I 8330 88 FR 21902 5/12/2023
carbamates, its salts, and salts of its acetals, its amides, and its carbamates,
and any combination thereof, whenever the existence of such is possible
N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007
BENZYLFENTANYL (N-(1-benzylpiperidin-4-yl)-N-phenylpropionamide), I 8334 85 FR 20822 5/15/2020
including its salts.
4-ANILINOPIPERIDINE (N-phenylpiperidin-4-amine; N phenyl-4- I 8335 85 FR 20822 5/15/2020
piperidinamine; 4–AP) including its amides,its carbamates, and its salts
1-BOC-4-AP (tert-butyl 4-(phenylamino)piperidine-1-carboxylate) and its salts I 8336 87 FR 67550 11/9/2022
3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690 3/18/1989
APAAN (Alpha-phenylacetoacetoniltrile), salts, optical isomers, salts of I 8512 82 FR 32457 8/14/2017
optical isomers
APAA (Alpha-phenylacetoacetamide) and its optical isomers (Effective I 8515 86 FR 24703 6/9/2021
06/09/2021)
ACETIC ANHYDRIDE II 8519 Pub. L. 100-690 3/18/1989
METHYLAMINE and salts I 8520 Pub. L. 101-647 2/27/1991
N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690 3/18/1989
PMK GLYCIDIC ACID (3,4-MDP-2-P METHYL GLYCIDIC ACID) and its salts, I 8525 86 FR 24703 6/9/2021
optical and geometric isomers, and salts of isomers (Effective 06/09/2021)
ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690 3/18/1989
PMK GLYCIDATE (3,4-MDP-2-P METHYL GLYCIDATE) and its optical and I 8535 86 FR 24703 6/9/2021
geometric isomers (Effective 06/09/2021)
BENZYL CHLORIDE II 8570 Pub. L. 100-690 3/18/1989
ERGOCRISTINE I 8612 76 FR 17778 5/2/2011
ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690 3/18/1989
ERGOTAMINE & salts I 8676 Pub. L. 100-690 3/18/1989
ETHYLAMINE & salts I 8678 Pub. L. 101-647 2/27/1991
ISOSAFROLE I 8704 Pub. L. 101-647 2/27/1991

* Remain in Schedule III


List I and II Regulated Chemicals - by DEA Chemical Code Number
07-Jul-23 Page 2 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
BENZYL CYANIDE I 8735 Pub. L. 100-690 3/18/1989
PIPERONAL I 8750 Pub. L. 101-647 2/27/1991
PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690 3/18/1989
METHYL ALPHA-PHENYLACETOACETATE (MAPA) I 8795 86 FR 64362 12/20/2021

* Remain in Schedule III


List I and II Regulated Chemicals - by DEA Chemical Code Number
07-Jul-23 Page 3 of 3
List I and II Regulated Chemicals
- by List Number -
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE

1-BOC-4-AP (tert-butyl 4-(phenylamino)piperidine-1-carboxylate) and its salts I 8336 87 FR 67550 5/15/2020

4-ANILINOPIPERIDINE (N-phenylpiperidin-4-amine; N phenyl-4- I 8335 85 FR 20822 5/15/2020


piperidinamine; 4–AP) including its amides,its carbamates, and its salts

4-PIPERIDONE (piperidin-4-one) including its acetals, its amides, its I 8330 88 FR 21902 5/12/2023
carbamates, its salts, and salts of its acetals, its amides, and its carbamates,
and any combination thereof, whenever the existence of such is possible

N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690 3/18/1989

ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690 3/18/1989

APAA (Alpha-phenylacetoacetamide) and its optical isomers (Effective I 8515 86 FR 24703 6/9/2021
06/09/2021)

APAAN (Alpha-acetoacetonitrile), salts, optical isomers, & salts of optical I 8512 82 FR 32457 8/14/2017
isomer

BENZALDEHYDE I 8256 Pub. L. 103-200 4/17/1994

BENZYL CYANIDE I 8735 Pub. L. 100-690 3/18/1989

BENZYLFENTANYL (N-(1-benzylpiperidin-4-yl)-N-phenylpropionamide), I 8334 85 FR 20822 5/15/2020


including its salts.

gamma-BUTYROLACTONE I 2011 Pub. L. 106-172 2/18/2000

EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690 3/18/1989

EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200 4/17/1994

EPHEDRINE remove exemption for OTC ephedrine combination products I 8113 Pub. L. 104-237 10/3/1996
and establish a 24 g retail threshold. Threshold remains zero for single entity
products. Mail order report requirements imposed. For more info, see 21
CFR Parts 1309, 1310, 1313.

ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690 3/18/1989

ERGOCRISTINE and its salts I 8612 76 FR 17778 5/2/2011

ERGOTAMINE & salts I 8676 Pub. L. 100-690 3/18/1989

ETHYLAMINE & salts I 8678 Pub. L. 101-647 2/27/1991

HYDRIODIC ACID I 6695 Pub. L. 101-647 2/27/1991

HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, I 6797 66 FR 52670 11/16/2001


calcium hypophosphite, iron hypophosphite, potassium hypophosphite,
manganese hypophosphite, magnesium hypophosphite, and sodium
hypophosphite)

IODINE I 6699 72 FR 35920 8/1/2007

ISOSAFROLE I 8704 Pub. L. 101-647 2/27/1991

METHYLAMINE and salts I 8520 Pub. L. 101-647 2/27/1991

METHYL ALPHA-PHENYLACETOACETATE (MAPA) and its optical isomers I 8795 86 FR 64362 12/20/2021

List I and II Regulated Chemicals - by List Number


07-Jul-23 Page 1 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE

3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690 3/18/1989

N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647 2/27/1991

N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical I 8119 Pub. L. 101-647 2/27/1991
isomers

NITROETHANE I 6724 Pub. L. 103-200 4/17/1994

NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690 3/18/1989

N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007

PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690 3/18/1989

PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690 3/18/1989

PHENYLPROPANOLAMINE -remove exemption for certain OTC I 1225 Pub. L. 104-237 10/3/1997
transactions. Retail threshold of 24 g established for products not distributed
in blister packs. Mail order report requirements imposed. For more info, see
21 CFR Parts 1309, 1310, and 1313.

PIPERIDINE and salts I 2704 Pub. L. 100-690 3/18/1989

PIPERONAL I 8750 Pub. L. 101-647 2/27/1991

PMK GLYCIDATE (3,4-MDP-2-P METHYL GLYCIDATE) and its optical and I 8535 86 FR 24703 6/9/2021
geometric isomers (Effective 06/09/2021)

PMK GLYCIDIC ACID (3,4-MDP-2-P METHYL GLYCIDIC ACID) and its I 8525 86 FR 24703 6/9/2021
salts, optical and geometric isomers, and salts of isomers (Effective
06/09/2021)

PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647 2/27/1991

PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100-690 3/18/1989

PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. I 8112 Pub. L. 104-237 10/3/1997
Retail threshold of 24 g established for products not distributed in blister
packs. Mail order report requirements imposed. For more info, see 21 CFR
Parts 1309, 1310, and 1313.

RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001

SAFROLE (includes sassafras oil) I 8323 Pub. L. 101-647 2/27/1991

WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001

ACETIC ANHYDRIDE II 8519 Pub. L. 100-690 3/18/1989

ACETONE II 6532 Pub. L. 100-690 3/18/1989

BENZYL CHLORIDE II 8570 Pub. L. 100-690 3/18/1989

ETHYL ETHER II 6584 Pub. L. 100-690 3/18/1989

HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992

HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237 10/3/1996

HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690 3/18/1989

IODINE - superseded by 2007 action II 6699 Pub. L. 104-237 10/3/1996

METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690 3/18/1989

METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995

List I and II Regulated Chemicals - by List Number


07-Jul-23 Page 2 of 3
DEA
CHEMICAL
LIST CODE EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE

POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690 3/18/1989

SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006

SULFURIC ACID II 6552 57 FR 43614 10/22/1992

TOLUENE II 6594 Pub. L. 100-690 3/18/1989

List I and II Regulated Chemicals - by List Number


07-Jul-23 Page 3 of 3
Listed Chemicals Regulated Under the  CONTROLLED SUBSTANCE PRODUCED

N,N‐Dimethylamphetamine
Controlled Substances Act

Fentanyl & analogues

Phenyl‐2‐propanone
Phencyclidine (PCP)
Methamphetamine
Ethylamphetamine

4‐Methylaminorex
See 21 C.F.R. §§ 1309, 1310, 1313 and 1314 

Methcathinone
Methaqualone
Amphetamine
for details

THRESHOLDS
DEA
Reagent =  Chemical

Cocaine
Precursor  = 

MDMA
Heroin
Last Update: Jul 07, 2023  Code

MDA

MDE
GHB
Solvent = 

LSD
Number
1. 1‐Boc‐4‐AP
 1
8336  0 0
2. 4‐Anilinopiperidine 
8
8335  0 0
3. 4‐Piperidone
12
8330  0 0
4. N‐Acetylanthranilic acid 2 8522  0 0

5. Alpha‐Phenylacetoacetamide  (APAA) 8515     0 0

6. Alpha‐Phenylacetoacetonitrile  (APAAN) 8512     0 0
7. Anthranilic acid 
2
8530  30 30
8. Benzaldehyde 8256   4 4
9. Benzyl cyanide 8735  1 1
10. Benzylfentanyl
 1
8334  0 0
11. Ephedrine 
3&7
8113   0 0
12. Ergocristine 
1
8612  0 0
13. Ergonovine 
1
8675  0.010 0.010
14. Ergotamine 
1
8676  0.020 0.020
15. Ethylamine 
1
8678   1 1
16. gamma‐Butyrolactone (GBL) 2011  0 0
17. Hydriodic acid 6695  1.7 1.7
1
18. Hypophosphorous acid  6797   0 0
19. Iodine 6699   0 0
LIST I

20. Isosafrole 8704    4 4


21. Methyl alpha‐phenylacetoacetate (MAPA) 
9
8795    0 0
22. Methylamine 
1
8520   1 1
23. 3,4‐Methylenedioxyphenyl‐2‐propanone 8502    4 4
24. N‐Methylephedrine 
3
8115  1 1
25. N‐Methylpseudoephedrine 
3
8119  1 1
26. N‐phenethyl‐4‐piperidone (NPP) 8332  0 0
27. Nitroethane 6724    2.5 2.5
28. Norpseudoephedrine 
3
8317   2.5 2.5
29. Phenylacetic acid 
2
8791  1 1
30. Phenylpropanolamine  3&7 1225   0 0
31. Phosphorus (red) 6795   0 0
32. Phosphorus (white or yellow) 6796   0 0
33. Piperidine 
1
2704  0.500 0.500
34. Piperonal (heliotropin) 8750    4 4
35. PMK glycidate 
10
8535    0 0
36. PMK glycidic acid 
11
8525    0 0
37. Propionic anhydride 8328  0.001 0.001
38. Pseudoephedrine 
3&7
8112   0 0
39. Safrole 8323    4 4
40. Acetic anhydride 8519    1,023 1,023
41. Acetone 6532        150 1,500
42. Benzyl chloride 8570  1 4
43. Ethyl ether 6584              135.8 1,364
Hydrochloric acid 5&6 6545               N/C 222.3
44.
Hydrogen chloride gas 5&6
LIST II

6545               0 27
45. Methyl ethyl ketone (2‐Butanone) 6714      145 1,455
4
46. Methyl isobutyl ketone  6715      N/C 1,523
47. Potassium permanganate 6579  55 500
48. Sodium permanganate 6588  55 500
5&6
49. Sulfuric acid  6552        N/C 347
50. Toluene 6594      159 1,591
1 and its salts
2 and its salts and esters
IMPORTS &
DOMESTIC

3 and its salts, optical isomers, and salts of optical isomers
EXPORTS

4 Exports only, to all Western Hemisphere except Canada
5 Exports to all South American countries & Panama ‐ Domestic for HCI gas
6 Threshold for HCI acid and sulfuric acid is 50 gallons, the equivalent weight in kilograms is shown
7 For pseudoephedrine, phenylpropanolamine and ephedrine drug products, see 21 USC § 802(45)(A) and 21 C.F.R. Part 1314
8  Including its amides, its carbamates, and its salts
9 and its optical isomers
10 and its optical and geometric isomers
11 and its salts, optical and geometric iosmers and salts of optical and geometric isomers KILOGRAMS
12 and its acetals, amides, carbamates, salts, and salts of acetals, amides, carbamates, and any combinaton thereof, whenever that existence of such is possible

N/C = Not Controlled

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