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S e m e s t e r G a s a l T. A 2 0 1 9 / 2 0 2 0
N -Terminal chain
Membrane VII VI
Transmembrane
V IV III II I helix
G-Protein
binding region
HO2C
Variable
C -Terminal chain
intracellular loop Intracellular loops
Struktur Dasar
• 7 Transmembrane Domains (TMDs),
• 3 intracellular loops,
• 3 extracellular loops, Pharmacol Ther. 2004 Jul;103(1):21-80
• N- and C-teminals
Basic structure: GPCRs are lipoproteins
Diversity of GPRS Receptors