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ANTIHISTAMINICS
Dr.Vijay bhushanam
HISTAMINE (Introduction)
• Exocrine Glands
• Gastric glands
• Salivary glands
• Sweat glands Secretion
• Pancreas
• Bronchial glands
• Lacrimal glands
HISTAMINE (Pharmacological Effects)
• Vasodilation
• Arterioles,
• Increased
permeability(edema)
• Capillaries • Systemic
• Venules hypotension
HISTAMINE (Pharmacological Effects)
• Metabolism: In liver
• Excretion: In urine
Antihistaminics
(Pharmacological actions)
• Smooth Muscle: Inhibit most of the effects of histamine
on smooth muscles, especially the constriction of
respiratory smooth muscle
• H3 antihistaminics: Thioperamide
• No clinical utility.
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