Professional Documents
Culture Documents
Jimmy Posangi
Anti infeksi bakteri
Levofloxacin
Chloramphenicol
Dibecacin
Sulfacetamide
Fusidic acid
Ciprofloxacin
Gentamicin
Tobramycin
Tetracyclin
Oxytetracyclin
Gramicidin
Polymixin B
Ofloxacin
Neomycin
Framycetin
Five Basic Mechanisms of Antibiotic
Action against Bacterial Cells:
1. Inhibition of Cell Wall Synthesis
Beta-Lactams ---> Inhibition of
peptidoglycan synthesis (bactericidal)
2. Inhibition of Protein Synthesis
(Translation)
30S Ribosome site
Aminoglycosides ---> Irreversibly bind 30S
ribosomal proteins (bactericidal)
3. Alteration of Cell Membranes
Polymyxins (topical) ---> Cationic
detergent-like activity (topical use)
4. Inhibition of Nucleic Acid Synthesis
DNA Effects
Quinolones ---> Inhibit DNA gyrases or
topoisomerases required for supercoiling of
DNA; bind to alpha subunit
5. Antimetabolite Activity
Sulfonamides & Dapsone ---> Compete
with p-aminobenzoic acid (PABA)
preventing synthesis of folic acid
Antiseptic
Thimerosal
(pengawetan vaksin)
Antivirus
Iodoxuridine
Acyclovir
Corticosteroid
Betamethasone
Hydrocortisone
Prednisolone
Fluorometholone
Dexamethasone
Antihistamin
Chlorpheniramine maleate
Pemirolast
Lodoxamide
Na cromoglycate
Midriatikum
Tropicamide
Scopolamin
Atropine
Homatropine
Phenylephrine
Miotikum
Betaxolol
Pilocarpine
Acetylcholine
Tropicamide
Pilocarpine
Scopolamin Phenylephrine Betaxolol
Acetylcholine
Atropine
Homatropine
Glaucoma
Brinzolamide
Betaxolol
Pilocarpine
Timolol
Latanoprost
Diuretics
MANNITOL
Proximal THIAZIDES
Convulated Tubule
Early Distal
Convulated Tubule
65%
10%
Fluorecin