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2 o7 2010

AUTOCOInS

ets
Auotoid

Hovmone
ypes oell
many ddd Site o Produchom

Spetyic Endocvine Ctlands


Ac
Ac via Blood Distan
site nothing b
S
HORM DNES
LOCAL

ao
all
Peptiden tokihe

Amine Upids
Kinins
ete

HisBamine PG main tYPOD


-Apgiolengin
Seaokonin. -LT aR
(5-HT)

in
RA
UNIT

srat
Presaglandins
Let US

them
NSAID

Phospholipids
se Az
Phospholipa

Arachidonit asid
-oygenae
C cox)
cyclo
LK Lipo-omygenase NSAD
PGs Prostoqlandins
LT
C l e u o i e n o s

Z\leuton

mediobfs Tnlommm

HepafoToxicit
yochidonic aid Ejs
Let us Shit
o us to Housekepí
CoX-1 '- tonshnH h
mcmbane )
Hihpid
AA Tnduobu enzy»
-Cox-2
COX Atvi 1M1 lomnr,
Inlemediak

othes Tisa39e

inside dethe liumm


Platelets frostacyclin
Tsomease
sAthase
TXsynthae

TXA, Pqsak CPros ha tych)


b yaodila ion
PG PaEre2
Jvaotonshtho

platele AnhPlate ler


9egahon
39ea hon Tiyre (Aocim
House Kee?ing doio
S6 blood

is at
Balana Hemesram Injlammahon
Ce)
1 1 1 uveokgdelal
Forchons
(A HOUSE Keepng
v e e l

P e m e a b i i k y
wabeula
ennancen

olechon oGost
TOP D&eREASED vse Do e) n Angb e N Glautoma

Hemosraxs
AFERENT GF
Renal Dilate
SoNSAID dierehe achm

UTERUS
OCervica Ripening in favtum
Utevine Con ac hon

fet lahon
erolaion PG keep DUCTOS ARreRiosos
Cbypas Fea lo)
tmnec
Polm at 4 Aorto

BIRTH Fetus
G J P leel
dochus autuots
9s CLOSE
Somehme colled
Patent Ductos tHrteriosu iament 4}Yexiosui
tam Heaut i
Long

ndoethadh (n-fw
Touprohen
Someime child b01n Otme CHD
by 6URGERY

So1 the
e
to eep T)uctos open
Time o gey

PGEHIprostadl
anaog

(Bediohs PAINa InlamMn


by coxR
NSAIDS
COX inhibinm -by
6Tiea

AOSTA&UANDIN

PG E analogues

a MisoPROSTO L
bAlprostadt&
To Keep DUCTUS

Oper
Pephc ulcey

MTP Erech unchon

cevvical vipen
Posr auhu Ingenea

DTUgs for E
Inra-Caveynes al inj
Mobieus Syndrome qive
Oe can (inhb penis)
CYanjal Neu Alpro stadi O660LETE.

Phentolamint
devmitg
Papaviv

ORAL
Sildenaffl

moinl fov

PGER analogues
,CFRMCALijeni
Vlerine unradoon

DINOPYOSTonelabo induchon

cevica vipeni
'.Dinopro5t Avoid
ao UA
n

avo
pros PPH (Tm ini) Asthmahcs

Latanoprost 10P
inGlaucoma

BYoncho csnuichon

Produch

NSAID TnhibiH COX PG

Prachtal clanffeahion

CoX inhtbilov
N o n Selectve,

Irveverib Aeby baliyie Aid


Revev ba only oe drog
CASPIRIN)

COX-8
COX-& . selechve inhibinu
COXIB

COX-3 aibib
aracetarndlAcehaminepher
Non Selechve COX # vesible

Havmul Achon
Beneaal othion erosin
mutosal
) G a sic
P n i - Inlammaoy
Beeding9 Anh ploteek achon

Pnalge
Pnyreht
3 NethTopath
GFEleun
Kenal apilly Necw

(Analgesit nephvopathg

0 Indome thaci'n Hig Potenoy loru alh


PDA
DoC Acute qo0UT

= avoid in Driven
wo YeYs elc
Sedahon
Head ache

chîlden
IbuPYoen Safes NSAID in k KEYES Snd
Go LOwEST

COX2inhbi

Dicbfenac Prejevrenhai qasrhs

efe
fevea
ropulau Percsibe
L mild cai
mild ain

i
Banned Cevn
So
NimEsULIDE S e tlepabh
xic
childen
No 8ae i

JNSOD pYodn
PDDYTiONAL, al

an udlam J TNF ete


8'Yen Iv
Ketorolac
Pos OP pain
movpu
similan
Cejhica

ENTEROtHepahc ciruln.

PROX CAM vndeg

6ie

Longenhes
BaceungvgaH )
LveY

via
PORTAL
veth

So Longe achhg
Henu
OD is onou
n u da

CoX inhibio RREvERS18E

Non Non Sel


dependen

ASPIAIN dose

Modeiare High-dose
dose
Low
=
Ani Jlamn
o 45-300 holet qthm 93g-/ achion
abe 5tavenging
V wV V
Free Raditals
Analgecie
5 0 - a53 /a
DISPIRIN Antipyretic
does ave

vsed
CMedenale Karey
Tero OYder
Kinehic
Kineho

TSorlex kinehts

High dose
matjen

ty 4-5k a n o how m u c h m o n

ceviain (ah he
taken
UTic Aud Retenhonm URicD SOc Acid
Lot Dose
dete, 11 vicasid
excrehon
High in URINE

NT- PLATeLET JTXAa Pproan


G mOA IrveveYsib coinhbin
inhbion

Sina PlaBe lels


cox -Aspiin LaCk
nucle
COX
fovm New
CoX p r oe m

Can no

T Syn t h a

Plalelet

TXA2
enkre

i 4 naba to
Sqm TA2

C 1 0day)

LOW dose
but why Lo ose
in
PYodn
G Inhibt TXA
TXA22

Flae I n a c h e

plateleh

S Higd d6se
No
ASA deaeylahon NET e alyo inhii PGla
Edotheliur

Hgbdo

ASA In ve,
on
ddacetylah
to
du
P l a t e l e

Salicylak

fspirin Inach e

Plalelek
e HIGH do
all ASA,
ve can de ace tyla
PORTAL shsh|l som ASA
Hena ib achm
SIE veqnont
A8 CDG* rgnat
ASTHmA Canleod 4o pivin
ndoced, HSTHMA

In Sch Pt, giw NOT an allegit Rn


te
Karacetamdl
HSN Yn
Nemesvlde NOT an

AA
LOX

Ts So PG
mok

towaudy

LTS
Jead
ASthma

Blecdi disovde Hemophilio


Denguu
Pephc Ulcea disea

Viral diseax
re
CHILDKen yeuvevîng CFlo chicken fox)

Aspivh
Encephalepaty ReVE
Gs8 Hepaneoon Symdrau

rabeke Atpinincavk
Uh coupling
Oxidahue Hiyh 1h
Phesphovyloho

CoUT Normal
Hyper Uhiteie

LOW Birth, weigkt


n a
lhaw tloson
P r e m a t v r e

child
Pheg orny G d 4riesle voIal NSAID CTUS
5alicylate Tox1ciTy

Ontouplirg Ovidohiu thotphnybhe

produchn Hyperthernaa
leads 111 Heat
tYPeR- Vénhlai
111 Co2 rtdo
Prodh

Shmulale
YEspitahsS
(Tachyphes
mo
o a s h o b

So

KesProKAUDSIS

m pensabry Kidny
So excvehon
y
HCO3

lead to
enitolh)
etcbolic idotir l )

Salicylae ih dic woYSenn


aid
aids

+unu
mebabolic Acdons
Otypethumia

N/v
Tinohs

meral fvst*

Natt NaHCO03

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