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Drug Classes 2.0
Drug Classes 2.0
ACTING) ACTING)
Non-Selective – Selective Alpha-1 Agonists SABAs (Salbutamol/Albuterol)
NE, E, DA - Phenylephrine,
Phenylpropanolamine, LABAs (Salmeterol, Formoterol)
Non-Selective Beta Agonist – Pseudoephedrine, Methoxamine
Isoproterenol Tocolytics (Terbutaline, Isosuxpride,
Selective Alpha-2 Agonists Ritodrine)
Non-Selective Alpha Agonist - - Clonidine, Methyldopa,
Oxymetazoline Guanabenz, Guanfacine Selective Dopamine-1 Agonist
Fenoldopam
Selective Beta-1 Agonists
- Dobutamine
ADRENERGIC AGONISTS (INDIRECT- ADRENERGIC AGONISTS (MIXED- ADRENERGIC ANTAGONISTS
ACTING) ACTING)
Tyramine, Ephedrine, Phenylpropanolamine Non-Selective
Amphetamine, - Labetalol, Carvedilol
Methylphenidate,
Phentermine Non-Selective Alpha Blockers
- Phenoxybenzamine, Phentolamine
DRUGS FOR ALZHEIMER'S DISEASE CHOLINERGIC ANTAGONISTS: ANTI- CHOLINERGIC ANTAGONISTS: ANTI-
MUSCARINICS NICOTINICS
Donepezil, - Atropine, Scopolamine Ganglionic Blockers
Tacrine, - Homatropine, Cyclopentolate, - Hexamethonium, Mecamylamine,
Rivastigmine, Tropicamide Trimetaphan
Galantamine - Ipratropium, Tiotropium
- Benztropine, Trihexyphenidyl, Biperiden Neuromuscular Blocker
- Oxybutinin, Dicycloverine, Hyoscine, - Depolarizing: Succinylcholine
Glycopyrrolate - Non-Depo (Steroidal) - Pancuronium
- Non-Depo (Isoquinoline) - Tubocurarine,
Atracurium
DIURETICS VASODILATORS
Carbonic Anhydrase Inhibitors Thiazide Diuretics Hydralazine,
- Acetazolamide, Brinzolamide, - Benzothiadiazide: HCTZ, Chlorthiazide Diazoxide,
Dorzolamide, Metazolamide, - Sulfonamide Thiazide-like: Minoxidil,
Dichlorphenamide Chlorthalidone, Indapamide, Metalozone Fenoldepam,
Na nitroprusside
Osmotic Diuretic K-sparring Diuretics
- Mannitol - Aldosterone Blockers: Spironolactone,
Eplerenone
Loop Diuretics - Na channel Blockers: Amiloride,
- Sulfonamide: Furosemide, Bumetanide Triamterene
- Sulfonylurea: Torsemide
- Phenoxyacetatic: Ethacrynic acid
ACE Inhibitors (-prils) AR Blockers (-sartans) RENIN INHIBITOR
Captopril, Losartan, Aliskerin
Lisinopril Valsartan,
Irbesartan
CALCIUM CHANNEL BLOCKERS NITROVASODILATORS OTHER DRUGS FOR CAD
- Dihydropyridine: Nitroglycerin, pFOX inhibitor
Amlodipine, Nifedipinde, Nicardipine, Isosorbide mononitrate
Felodipine Isosorbide dinitrate Trimetazidine,
Ranolazine
- Non-Dihydropyridine:
Verapamil, Diltiazem
INOTROPICS UNLOADERS ANTI-ARRHYTHMIC AGENTS
Cardiac Glycoside: Digoxin Neprilysin Inhibitor + ARB: Sacubitril + Class IA
- PDE III Inhibitor: Milrinone Valsartan - Quinidine, Disopyramide, Procainamide
- Ca sensitizer: Levosimendan - BNP: Nesiritide
- Beta-1 Agonists - ACEIs/ARBs Class IB
- Diuretics - Lidocaine, Phenytoin, Tocainamide,
- Beta Blockers Mexiletine
Class IC
- Moricizine, Propafenone, Flecainide,
Encainide
Class II
- Cardioselective Beta Blockers
Class III
- Sotalol, Amiodarone, Bretylium,
Ibutilide, Dofetilide
Class IV
- Verapamil, Diltiazem
Others Anti-Arrhythmias
- Adenosine
- MgSO4
ANTI-PSYCHOTICS
1ST GENERATION/TYPICAL 2ND GENERATION/ATYPICAL TRICYCLIC ANTIDEPRESSANTS
- Phenothiazine Clozapine, - Amitriptyline, Nortriptyline, Imipramine,
> Alipathic - Chlorpromazine Olanzapine, Desipramine, Doxepin
> Piperazine - Fluphenazine Risperidone,
> Piperidine - Thioridazine Paliperidone, Anti-Mania
Aripiprazole, - Lithium carbonate
- Butyrophenone: Amisulpride,
Haloperidol, Quetiapine SSRIs
Droperidol - Fluoxetine, Sertraline, Citalopram,
Escitalopram
- Thioxanthene:
Thiothixene SSNRIs
- Venlafaxine, Desvenlafaxine, Duloxetine
MAO INHIBITORS ATYPICAL ANTIDEPRESSANTS BENZODIAZEPINES
- Non-Selective: Bupropion, - Midazolam,
Phenelzine, T Mirtazapine, Lorazepam,
ranylcypromine, Nefazodone, Diazepam,
Isocarboxacid Trazodone Flunitrazepam,
Alprazolam
- MAO-a:
Moclobemide Non-Benzodiazepine
- Zolpidem,
- MAO-b: Zaleplon,
Selegiline Eszopiclone
BARBITURATES DRUGS FOR SEIZURES/EPILEPSY DRUGS FOR PAKINSON'S DISEASE
- Ultra Short-Acting: Carbamazepine, Levodopa,
Thiopental, Thiamylal, Methohexital Ethosuximide Carbidopa
Valproic Acid,
- Short-Acting: Lamotrignine,
Pentobarbital, Hexobarbital, Secobarbital Topiramate,
Phenytoin
- Intermediate-Acting:
Amobarbital, Butobarbital
- Long-Acting:
Phenobarbital, Metharbital,
Mephobarbital
DOPAMINE AGONISTS (PD) COMT INHIBITORS (PD) OTHERS (PD)
Ergot: Bromocriptine, Pergolide, Entacaqpone, Amantadine
Cabergoline Tolcapone Anticholinergic
> Non-Ergot: Pramipexole, Ropinirole MAO-b Inhibitors
GENERAL ANESTHESIA LOCAL ANESTHESIA
Inhaled Anesthetics Ester (Short-Acting)
- Nitrous Oxide, Cocaine,
Methoxyflurane, Procaine,
Enflurane, Chlorprocaine
Sevoflurane,
Halothane Amide (Long-Acting)
Lidocaine,
IV Anesthetics Bupivacaine,
- Propofol, Prilocaine
Etomidate,
Ketamine, BDZs, Barbiturates, Opioids
ANTIBACTERIAL AGENTS
CELL-WALL SYNTHESIS INHIBITORS
BETA-LACTAMS PENICILLINS BETA-LACTAM - CEPHALOSPORINS POLYPEPTIDES
Natural: 1st Gen: Vancomycin,
Pen G, Cefazolin, Cephalexin, Cefadroxil, Bacitracin,
Pen V Cephradine, Cephalotin Fosfomycin,
Teicoplanin,
> Anti-Staph: > 2nd Gen: Daptomycin,
Methicillin, Cefaclor, Cefoxitin, Cefotetan, Gramicidin A
Nafcillin, Cefamandole, Cefuroxime, Cefprozil,
Isoxazoyl Penicillins (Oxacillin, Cloxacillin, Cefpodoxime, Loracarbacef - Polymyxin:
Dicloxacillin) Polymyxin B,
> 3rd Gen: Colistin
> Broad-spectrum: Ampicillin, Amoxcillin Ceftriaxone, Cefoperazone, Cefdinir,
Ceftibuten, Ceftidoxime, Cefofaxime,
> Anti-Pseudomonal Ceftazidime, Cefotaxime, Moxolactam
- Carboxypenicillin:
Carbenicillin, Ticarcillin > 4th Gen:
Cefepime, Cefpirome
- Ureidopenicillin:
Azlocillin, Piperacillin, Mezlocillin > 5th Gen:
Ceftaroline, Ceftobiprole
PROTEIN SYNTHESIS INHIBITORS
30S - AMINOGLYCOSIDES 30S - TETRACYCLINE
Neomycin, > Short-Acting:
Tobramycin, Chlortetracycline, Tetracycline, Oxytetracycline
Gentamicin,
Amikacin, > Intermediate-Acting:
Kanamycin, Metacycline, Demeclocycline
Steptomycin
> Long-Acting:
Minocycline, Doxycycline
2. Sulfonamide
- Sulfasalazine, Sulfamethoxazole,
Sulfadiazine, Sulfadoxine, Silver
sulfadiazene, Sulfacetamide, Mafenide
3. Sulfones –
Dapsone
4. Methenamine
(Urothropin)