HiralOT_ADRENERGIC DRUGS Cheat Sheet

by Hiral OT (Hiral) via cheatography.com/31053/cs/9375/

Beta 1 Selective Agonists Beta 2 Selective Agonists (cont) Adrenergic Drugs (cont)

Located at Myocardium Another Uterine Muscle (When Adrenergic Stimulate activity in tissues that

Stimul​ation Increased Heart rate and
results in increased force of myocardial
contra​ction (Increased Cardiac
output)
USED FOR To increase cardiac output in
emergency situations such as
CVS shock or to treat
compli​cations in Cardiac
Surgery.
LOCATION stimul​ate​d--​>cause inhibition or
relaxation of the uterus)
Beta 2 Albuterol (Provv​entil, Ventolin),
Selective Metapr​ote​renol (Alupe​nt,),
Bronch​odi​al Pirbuterol (Maxair), Salmeterol
ators (Servent), and Terbut​aline
(Breth​aire, bricanyl).
what it Bronch​odi​lat​ation at pulmonary
causes smooth muscles - Asthma.
Drugs respond to Epi and NorEpi
(Adren​ergic agonists) OR inhibit
epinep​hrine and norepi​nep​hrine
influence (adren​ergic
antago​nists)
From Adrenal gland and reach to
where they Heart, Kidneys, and various other
release? tissues and organs via systemic
circul​ation.

also USED To increase cardiac function in Isopro​teren can be the same but: less beta 2 Where it is Junction between sympat​hetic
found postga​ngl​ionic neurons and
FOR the short-term treatment of ol (Isuprel) selective and affects beta 1
certain type of heart disease, - receptor too. peripheral tissues

heart failure Adm Oral inhalation so that affects on Adrenergic Sympat​hom​imetic

Dobutamine Use: Short term mx of Cardiac the bronchial membranes. agonists

(Dobutrex) decomp​ens​ation that occurs Adverse nervou​sness, restle​ssness, Adrenergic sypath​olytic

during heart disease or heart Effect trembling. sometimes fatal antago​nists
surgery. How: Increase force of
asthamatic attaacks.
cardiac contra​ction. Adm: IV Subcla​ssi​fic​ation of Adrenergic Drugs
When used Terbut​aline - increase in
pump infusion (to stable plasma
to treat maternal heart rate and systolic Adrenergic Alpha and Beta receptors
levels)
premature blood pressure, as well as receptors
Dopamine directly stimulates Beta 1. Low labor, maternal pulmonary edema. can be
(Intropin) DOSE: cause peripheral
Sometimes fatal to mother. divided
vasodi​lat​ation. Adm: IV drip to
into two
maintain stable plasma levels
Adrenergic Drugs Five Alph 1 (a, b, d) 2 (a, b, c) beta
ADVERSE Chest pain, difficulty in breathing
Adrenergic Refers physio​logical responses receptor 1,2,3,
Effects
subtypes
related to adrenaline and
noradr​enaline Alpha 1 or Located at specific tissues
Beta 2 Selective Agonists
alpha 2 throughout the body--> the
Other Adrenaline and NorAdr​enalin =
Location on bronchiole smooth muscle responsed depend upon
names Epinep​hrine and
intera​ction between that receptor
How Stimulated Beta 2 --> mediates NonEpi​nep​hrine
andthe reseptive tissue
relaxation of bronch​ioles
Agonist Increase or mimic the receptor
Treat Bronch​ospasm associated with
respir​atory ailments such as mediated response

asthama, bronch​itis, emphysema. Antagonist decrease the receptor mediated

Treats ALSO Cardiac Arrythmias or resonce
heart failure
Epinep​hrin affects alpha and beta receptors
e drug Equally

Receptor select​ivity

By Hiral OT (Hiral) Published 6th October, 2016. Sponsored by Readability-Score.com

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 HiralOT_ADRENERGIC DRUGS Cheat Sheet
by Hiral OT (Hiral) via cheatography.com/31053/cs/9375/

MIX ALPHA AND BETA MIX ALPHA AND BETA (cont) MIX ALPHA AND BETA (cont)

Amphat​ami Drugs:​Am Increase Norepi As Narcolepsy treatment Metara​min act like Directly stimulates
nes p​het​amine release and Bronch​od ol Epinep​hrin alpha 1, 2 and
(generic), decrease NorEpi i​lator (aramine) e beta1
dextro​amp​ reuptake and
Epinphrine All Antias​thmatic Treat shock or general
het​amine breakdown at
(Adren​alin, receptors inhalation products. - anasthesia
(Dexed​rin adrenergic
Bronkaid are primary stimulate B2 NorEpi​Nep​ Stimul​ates displays little
e) and synapses - so
Mist, stimul​ate bronchii. hrine : Alpha 1, agonistic activity
metham​ph Increase activity at Primatene d.
(Levophed) 2 and toward beta2.
a​tamine synapses with Mist, )
Beta 1.
(Desoxyn) Norepi sesitive
Effect of vasoco​nst​irction and
receptors - Alpha Adm IV Treat: Hypote​nsion
Alpha 1 control of bleeding injection during shock or
1,2 and Beta1)
vascular during minor surgical general
Used to The use to
procedures (sutures). anasth​esia.
treat suppress appetite or
Prolongs effects of
attent​ion​- to combat normal Adverse Nervou​sn Prolonged use
the anasth​etics
de​ficit sleepiness is Effect ess, Causes-
B1 effect reesta​blish normal restle​ssne hypert​ension,
disorder discou​rage- as they
on heart cardiac rhythm during ss, arrhyt​hmias, cardiac
in have high potential
cardiac arrest. anxiety. arrest.
children, of abuse
to Drug of hypers​ens​itive Prolonged Use in
increase choice in allergic reaction inhala​tion: Cause
mental Anaphy​la marked by CVS bronchial irrita​tion.
alertness ctic collapse (decreased
in adults shock cardiac output,
ALPHA 1 SELECTIVE AGONISTS
with hypote​nsion) and
narcol​eps severe Alpha 1 or Contra​ction and
y. bronch​oco​nst​ric​tion. alpha 2 VasoCo​nst​riction : Increase BP

Ephendrine Stimulate Use: Primarily for why Becase Stimulate heart (b1), Mephen​ter Mainta​in/​restore BP during
(Generic) Alpha 1, 2 Alpha 1 effects: ability to vasoco​nst​riction mine hypote​nsive episodes.
and beta treat hypote​nsion. periphery (alpha 1) (Wyamine) Admini​stered: IV or IM
1 and also and Dilate bronchi inject​ions.
stimulate (beta2).
the same
by
increasing
release of
norepi at
synapses

IV ALSO a nasal
injection decong​enstant -
stimulate alpha 1:
combined with other
agents
(antit​uss​ives,
antihi​sta​mines) to
form cough and
cold products

By Hiral OT (Hiral) Published 6th October, 2016. Sponsored by Readability-Score.com

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 HiralOT_ADRENERGIC DRUGS Cheat Sheet
by Hiral OT (Hiral) via cheatography.com/31053/cs/9375/

ALPHA 1 SELECTIVE AGONISTS (cont) ALPHA 1 SELECTIVE AGONISTS (cont) ALHA 2 SELECTIVE AGONISTS (cont)

Methox​am Increase and maintain BP in
i​ne(​Vas​ox severe hypote​nsion- during
yl) general anesthesia and spinal
anesth​esia. Treats: Paroxymal
syprav​ent​ricular tachyc​ardia by
causing peripheral
vasoco​nst​ric​tion, activation of
barore​ceptor reflex. Adm : IV
injection
Midodrine Treat: orthos​tatic hypote​nsion
(ProAm​ati Adm: Orally Also: treat
ne) hypote​nsion in patients who go
under dialysis, offset the
hypote​nsive effects of
psycho​tropic drugs like
antips​ychotic medica​tions
Oxymet​az Adm: naslal drops and nasal
oline sprays. Treat: Decrease nasal
(Afrin, congestion and decrease redness
OcuClear, and minor eye irritation
Many
others)
Phenyl​eph Treat: hypote​nsion, treat certain
rine (Neo- episodes of suprav​ent​ricular
S​yne​phrin tachyc​ardia. Adm: Orally a lso or
e, Others) nasal spray, or topically as eye
Adverse increased BP, headache, Clonidine Antihy​per​tensive and analgesic,
Effect: abnormally slow heart rate, (Catapres, It does not effect ALONE. so
sometimes chest pain, difficulty in Duraclon) given with PRAZOSIN (Minipress
breathing, feelings of nervou​sness - alpha antago​nists). also useful
to treat severe pain in cancer.
ALHA 2 SELECTIVE AGONISTS Guanabenz decrease BP (same as
(Wytensin) Clonidine)
Primary Hypert​ension, spasti​city..
use Guanfacine similar to Guanabenz
(Tenex)
How Drug stimulate alpha-2 receptors
located at brain and brainstem -- Methyldopa Antihy​per​ten​sive.
> cebtral alpha2 exert an (Aldomet)
inhibitory effect on sympat​hetic Tizanidine To treat spasti​city. Similar to
discharge from the vasomotor (Zanaflex) Clonidine but has fewer
center in the brainstem ---> vasomotor effects and less likey
diminished sympat​hetic to cause hypote​nsion and other
discharge results in decreased CVS problems.
BP.
Adverse Hypote​nsion, dizziness,
Also Stimul​ation of Alpha 2 --> causes Effects drowsi​ness, dry mouth. Difficulty
effective intern​euron inhibition and a in breathing, slow heart rate,
on Spinal subsequent decrease in persistent fainting - overdose of
cord excita​bility of motor neurons drugs.
supplied by intern​eurons. USE
TO normalize the neuronal
activity in Spasticity
Brimon​idin Adm: local to eye to treat

drops. e glaucoma. (Decreases vitreous

(Alphagan) humor production and increasing
Pseudo​ep Adm: Orally - relieve cold
drainage of vitreous humor from
h​edrine symptoms
the eye)
(Drixoral,
Sudafed,
etc)

Xylome​taz​ nasal spray to decrease

oline congestion during cold and
(Otrivin) alergies.

By Hiral OT (Hiral) Published 6th October, 2016. Sponsored by Readability-Score.com

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